DE60204633T2 - Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel - Google Patents
Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel Download PDFInfo
- Publication number
- DE60204633T2 DE60204633T2 DE60204633T DE60204633T DE60204633T2 DE 60204633 T2 DE60204633 T2 DE 60204633T2 DE 60204633 T DE60204633 T DE 60204633T DE 60204633 T DE60204633 T DE 60204633T DE 60204633 T2 DE60204633 T2 DE 60204633T2
- Authority
- DE
- Germany
- Prior art keywords
- triazoles
- sulfonyl
- heteroaryl
- inflammatory
- analgesic agents
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Dermatology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Heart & Thoracic Surgery (AREA)
- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Virology (AREA)
- Immunology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US30323201P | 2001-07-05 | 2001-07-05 |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60204633D1 DE60204633D1 (de) | 2005-07-21 |
DE60204633T2 true DE60204633T2 (de) | 2006-06-14 |
Family
ID=23171118
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60204633T Expired - Fee Related DE60204633T2 (de) | 2001-07-05 | 2002-07-01 | Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel |
Country Status (9)
Country | Link |
---|---|
US (2) | US6753332B2 (de) |
EP (1) | EP1273580B1 (de) |
JP (1) | JP2003040887A (de) |
AT (1) | ATE297913T1 (de) |
BR (1) | BR0202546A (de) |
CA (1) | CA2392271C (de) |
DE (1) | DE60204633T2 (de) |
ES (1) | ES2240661T3 (de) |
MX (1) | MXPA02006723A (de) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100686537B1 (ko) * | 2001-12-28 | 2007-02-27 | 씨제이 주식회사 | 사이클로옥시게나제-2 의 저해제로서 선택성이 뛰어난디아릴 1,2,4-트리아졸 유도체 |
KR100467668B1 (ko) * | 2002-08-07 | 2005-01-24 | 씨제이 주식회사 | 1,2,4-트리아졸 유도체, 그 제조방법 및 약제학적 조성물 |
US7074809B2 (en) * | 2002-08-09 | 2006-07-11 | Astrazeneca Ab | Compounds |
KR100491317B1 (ko) * | 2002-11-26 | 2005-05-24 | 씨제이 주식회사 | 1,2,4-트리아졸 유도체, 그 제조방법 및 약제학적 조성물 |
BRPI0414663A (pt) * | 2003-09-22 | 2006-11-21 | Pfizer | derivados triazol substituìdos como antagonistas de oxitocina |
TW200835487A (en) * | 2006-12-28 | 2008-09-01 | Basf Ag | 2-substituted pyridines I in therapy |
DE112010001898T5 (de) | 2009-04-27 | 2012-08-02 | Dow Agrosciences Llc | Insektizide Pyridinverbindungen |
EP2527335B1 (de) | 2011-04-26 | 2013-09-18 | King Saud University | Triazolderivate als Entzündungshemmer |
US8853248B2 (en) * | 2012-04-05 | 2014-10-07 | Hubert Maehr | (1,2,3-triazolyl)sulfonyl derivatives |
CN112142716B (zh) * | 2020-10-29 | 2021-08-31 | 山东新时代药业有限公司 | 一种5元杂芳基取代的吡嗪衍生物及其应用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3169966A (en) * | 1961-01-24 | 1965-02-16 | Ciba Geigy Corp | Aminopyrazoles |
EP0003895A1 (de) | 1978-02-16 | 1979-09-05 | E.R. Squibb & Sons, Inc. | 1-Acyl-3(5)-alkyl-5(3)-phenyl-1,2,4-triazole, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen |
US4259504A (en) | 1979-08-27 | 1981-03-31 | American Cyanamid Company | Substituted 1H-1,2,4-triazoles |
HU193891B (en) | 1984-02-07 | 1987-12-28 | Gyogyszerkutato Intezet | Process for production of new derivatives of 1,2,4-triasole |
US5256680A (en) | 1988-11-29 | 1993-10-26 | Warner-Lambert Company | 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents |
US5066668A (en) | 1989-06-09 | 1991-11-19 | Warner-Lambert Co. | Triazole derivatives of fenamates as antiinflammatory agents |
US4962119A (en) | 1989-06-09 | 1990-10-09 | Warner-Lambert Company | Triazole derivatives of fenamates as antiinflammatory agents |
CA2327185A1 (en) * | 1998-04-08 | 1999-10-14 | Abbott Laboratories | Pyrazole inhibitors of cytokine production |
EP1099695A1 (de) * | 1999-11-09 | 2001-05-16 | Laboratoire Theramex S.A. | 5-Aryl-1H-1,2,4-triazolverbindungen als Cyclooxygenase-2 Inhibitoren und diese enthaltende pharmazeutische Zusammensetzungen |
DE60001623T2 (de) | 1999-12-03 | 2003-12-18 | Pfizer Products Inc., Groton | Sulfamoylheteroarylpyrazolverbindungen zur Verwendung als analgetisches/entzündungshemmendes Mittel |
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2002
- 2002-07-01 DE DE60204633T patent/DE60204633T2/de not_active Expired - Fee Related
- 2002-07-01 EP EP02254275A patent/EP1273580B1/de not_active Expired - Lifetime
- 2002-07-01 AT AT02254275T patent/ATE297913T1/de not_active IP Right Cessation
- 2002-07-01 ES ES02254275T patent/ES2240661T3/es not_active Expired - Lifetime
- 2002-07-03 CA CA002392271A patent/CA2392271C/en not_active Expired - Fee Related
- 2002-07-03 US US10/188,511 patent/US6753332B2/en not_active Expired - Fee Related
- 2002-07-04 BR BR0202546-9A patent/BR0202546A/pt not_active IP Right Cessation
- 2002-07-04 JP JP2002196419A patent/JP2003040887A/ja active Pending
- 2002-07-04 MX MXPA02006723A patent/MXPA02006723A/es not_active Application Discontinuation
-
2004
- 2004-04-22 US US10/829,882 patent/US6875779B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
ES2240661T3 (es) | 2005-10-16 |
ATE297913T1 (de) | 2005-07-15 |
US6753332B2 (en) | 2004-06-22 |
US6875779B2 (en) | 2005-04-05 |
DE60204633D1 (de) | 2005-07-21 |
MXPA02006723A (es) | 2003-01-23 |
US20040198735A1 (en) | 2004-10-07 |
CA2392271A1 (en) | 2003-01-05 |
JP2003040887A (ja) | 2003-02-13 |
BR0202546A (pt) | 2003-05-13 |
CA2392271C (en) | 2006-08-29 |
EP1273580B1 (de) | 2005-06-15 |
US20030119835A1 (en) | 2003-06-26 |
EP1273580A1 (de) | 2003-01-08 |
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