DE3873862T2 - 17-substituierte androsta-1,4-dien-3-on-derivate. - Google Patents

17-substituierte androsta-1,4-dien-3-on-derivate.

Info

Publication number
DE3873862T2
DE3873862T2 DE8888308104T DE3873862T DE3873862T2 DE 3873862 T2 DE3873862 T2 DE 3873862T2 DE 8888308104 T DE8888308104 T DE 8888308104T DE 3873862 T DE3873862 T DE 3873862T DE 3873862 T2 DE3873862 T2 DE 3873862T2
Authority
DE
Germany
Prior art keywords
alkyl
hydrogen
derivatives
dien
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE8888308104T
Other languages
English (en)
Other versions
DE3873862D1 (de
Inventor
Vittoria Villa
Salle Enrico Di
Paolo Lombardi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL, Carlo Erba SpA filed Critical Farmitalia Carlo Erba SRL
Publication of DE3873862D1 publication Critical patent/DE3873862D1/de
Application granted granted Critical
Publication of DE3873862T2 publication Critical patent/DE3873862T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0018—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Superconductors And Manufacturing Methods Therefor (AREA)
  • Mounting, Exchange, And Manufacturing Of Dies (AREA)
  • Catalysts (AREA)
DE8888308104T 1987-09-11 1988-09-01 17-substituierte androsta-1,4-dien-3-on-derivate. Expired - Fee Related DE3873862T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB878721384A GB8721384D0 (en) 1987-09-11 1987-09-11 17-substituted andro-sta-1 4-dien-3-one derivatives

Publications (2)

Publication Number Publication Date
DE3873862D1 DE3873862D1 (de) 1992-09-24
DE3873862T2 true DE3873862T2 (de) 1993-01-14

Family

ID=10623619

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8888308104T Expired - Fee Related DE3873862T2 (de) 1987-09-11 1988-09-01 17-substituierte androsta-1,4-dien-3-on-derivate.

Country Status (14)

Country Link
US (1) US4873233A (de)
EP (1) EP0307135B1 (de)
JP (1) JP2677626B2 (de)
KR (1) KR970007948B1 (de)
AT (1) ATE79629T1 (de)
AU (1) AU602607B2 (de)
CA (1) CA1305699C (de)
DE (1) DE3873862T2 (de)
ES (1) ES2043834T3 (de)
FI (1) FI88393C (de)
GB (1) GB8721384D0 (de)
GR (1) GR3005961T3 (de)
IL (1) IL87656A (de)
SU (1) SU1750431A3 (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH683151A5 (de) * 1991-04-24 1994-01-31 Ciba Geigy Ag Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.
FR2681069B1 (fr) * 1991-09-06 1995-04-28 Roussel Uclaf Nouveau procede de preparation de l'hydrocortisone et nouveaux intermediaires.
GB9201224D0 (en) * 1992-01-21 1992-03-11 Erba Carlo Spa Difluoromethylenandrostenone derivatives and process for their preparation
GB9217035D0 (en) * 1992-08-11 1992-09-23 Erba Carlo Spa Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation
NZ261123A (en) * 1993-02-18 1996-08-27 Erba Carlo Spa Fluorinated 4-aminoandrostadienone derivatives
DE10104327A1 (de) * 2001-01-24 2002-07-25 Schering Ag 11beta-Halogensteroide, deren Herstellung und Verwendung zur Herstellung von Arzneimitteln sowie 11beta-Halogensteroide enthaltende pharmazeutische Präparate
WO2003032961A2 (en) * 2001-10-10 2003-04-24 Pharmacia Italia Spa Methods for preventing and treating bone loss with steroid compounds
US7435757B2 (en) * 2004-07-02 2008-10-14 Schering Ag 2-substituted D-homo-estra-1,3,5(10)-trienes as inhibitors of 17β-hydroxy steroid dehydrogenase type 1
US20060211667A1 (en) * 2005-03-21 2006-09-21 Eric Marchewitz Use of pregnane steroid derivatives for enhancing physical performance
EP1854465A1 (de) 2006-05-12 2007-11-14 Alexander Tobias Teichmann Verwendung von 4,17 beta-dihydroxyandrost-4-ene-3-one zur Behandlung von Krebs
ES2547339T3 (es) 2007-11-13 2015-10-05 Curadis Gmbh Esteroides C-19 para usos terapéuticos específicos
ES2574933T3 (es) 2007-11-13 2016-06-23 Athenion Ag Esteroides de C-19 para usos cosméticos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB929985A (de) *
GB8517360D0 (en) * 1985-07-09 1985-08-14 Erba Farmitalia Substituted androsta-1,4-diene-3,17-diones

Also Published As

Publication number Publication date
FI88393C (fi) 1993-05-10
CA1305699C (en) 1992-07-28
IL87656A0 (en) 1989-02-28
ES2043834T3 (es) 1994-01-01
EP0307135A1 (de) 1989-03-15
AU2197988A (en) 1989-03-16
KR970007948B1 (ko) 1997-05-19
ATE79629T1 (de) 1992-09-15
JP2677626B2 (ja) 1997-11-17
US4873233A (en) 1989-10-10
JPH01104096A (ja) 1989-04-21
SU1750431A3 (ru) 1992-07-23
FI884088A (fi) 1989-03-12
AU602607B2 (en) 1990-10-18
GR3005961T3 (de) 1993-06-07
GB8721384D0 (en) 1987-10-21
FI884088A0 (fi) 1988-09-06
KR890005142A (ko) 1989-05-13
FI88393B (fi) 1993-01-29
EP0307135B1 (de) 1992-08-19
DE3873862D1 (de) 1992-09-24
IL87656A (en) 1993-02-21

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ATE168367T1 (de) Vitamin-d-derivate und verfahren zu deren herstellung
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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8327 Change in the person/name/address of the patent owner

Owner name: PHARMACIA & UPJOHN S.P.A., MAILAND/MILANO, IT

8327 Change in the person/name/address of the patent owner

Owner name: PHARMACIA ITALIA S.P.A., MAILAND/MILANO, IT

8339 Ceased/non-payment of the annual fee