DE3468024D1 - Benzofuran- and benzopyran-carboxamide derivatives - Google Patents
Benzofuran- and benzopyran-carboxamide derivativesInfo
- Publication number
- DE3468024D1 DE3468024D1 DE8484103843T DE3468024T DE3468024D1 DE 3468024 D1 DE3468024 D1 DE 3468024D1 DE 8484103843 T DE8484103843 T DE 8484103843T DE 3468024 T DE3468024 T DE 3468024T DE 3468024 D1 DE3468024 D1 DE 3468024D1
- Authority
- DE
- Germany
- Prior art keywords
- lower alkyl
- group
- alkyl group
- hydrogen atom
- image
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Otolaryngology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Furan Compounds (AREA)
- Pyrane Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Detergent Compositions (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP58062554A JPS59186969A (ja) | 1983-04-08 | 1983-04-08 | ベンゾフラン−およびベンゾピランカルボキサミド誘導体 |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3468024D1 true DE3468024D1 (de) | 1988-01-21 |
Family
ID=13203591
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8484103843T Expired DE3468024D1 (de) | 1983-04-08 | 1984-04-06 | Benzofuran- and benzopyran-carboxamide derivatives |
Country Status (8)
Country | Link |
---|---|
US (1) | US4617314A (de) |
EP (1) | EP0124783B1 (de) |
JP (1) | JPS59186969A (de) |
KR (1) | KR910002883B1 (de) |
AT (1) | ATE31307T1 (de) |
CA (1) | CA1238906A (de) |
DE (1) | DE3468024D1 (de) |
ES (1) | ES8507135A1 (de) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5122528A (en) * | 1983-12-22 | 1992-06-16 | Erbamont, Inc. | Analgesic use of benzobicyclic carboxamides |
CA1297877C (en) * | 1983-12-22 | 1992-03-24 | Daniel Lednicer | Benzofurancarboxamides useful as antiemetic or antipsychotic agents |
US4888353A (en) * | 1986-02-28 | 1989-12-19 | Erbamont, Inc. | Carboxamides useful as antiemetic or antipsychotic agents |
US5175173A (en) * | 1983-12-22 | 1992-12-29 | Sun Jung Hui | Carboxamides useful as antiemetic or antipsychotic agents |
SE8503055D0 (sv) * | 1985-06-19 | 1985-06-19 | Astra Laekemedel Ab | Piperonylcarboxamido derivatives |
FR2593504B1 (fr) * | 1986-01-30 | 1988-12-09 | Ile De France | Nouveaux derives de dihydrobenzofuranne - et de chromane - carboxamides, leurs procedes de preparation et leur utilisation comme neuroleptiques |
JPS62234083A (ja) * | 1986-02-28 | 1987-10-14 | アーバモント インク ディビーエイ アドリヤ ラボラトリーズ | 鎮吐薬または精神病治療薬として有用なカルボキサミド類 |
US4772459A (en) * | 1986-09-09 | 1988-09-20 | Erbamont, Inc. | Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein |
DE3724756A1 (de) * | 1987-07-25 | 1989-02-09 | Basf Ag | Basisch substituierte benzofurancarbonsaeureamide, verfahren zu ihrer herstellung und sie enthaltende therapeutische mittel |
EP0314483A1 (de) * | 1987-10-29 | 1989-05-03 | Erbamont, Inc. | Herstellung von Benzamiden |
US5374637A (en) * | 1989-03-22 | 1994-12-20 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
US5122361A (en) * | 1989-04-17 | 1992-06-16 | Trustees Of The University Of Pennsylvania | Dopamine receptor ligands and imaging agents |
GB9005014D0 (en) * | 1990-03-06 | 1990-05-02 | Janssen Pharmaceutica Nv | N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives |
AU667874B2 (en) * | 1992-02-06 | 1996-04-18 | Smithkline Beecham Plc | Benzopyran, benzothiopyran and benzofuran derivatives as 5-HT4 antagonists |
FR2699533A1 (fr) * | 1992-12-21 | 1994-06-24 | Mouhtaram Mohamed | Dérivés de N-((1,4-dialkyl-6-arylpipérazine-2-yl)méthyl)benzamides. (Isomères cis et trans) Propriétés pharmacologiques et applications. |
GB9317987D0 (en) * | 1993-08-26 | 1993-10-13 | Glaxo Group Ltd | Chemical compounds |
CZ20011760A3 (cs) * | 1998-11-20 | 2001-12-12 | F. Hoffmann-La Roche Ag | Pyrrolidinové deriváty jako antagonisty CCR-3 receptorů |
DE60234057D1 (de) | 2001-07-25 | 2009-11-26 | Raptor Pharmaceutical Inc | Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke |
US7728155B2 (en) | 2003-10-24 | 2010-06-01 | Wyeth Llc | Dihydrobenzofuranyl alkanamines and methods for using same as cns agents |
CA2604915A1 (en) * | 2005-04-22 | 2006-11-02 | Wyeth | New therapeutic combinations for the treatment or prevention of depression |
CA2789262C (en) | 2005-04-28 | 2016-10-04 | Proteus Digital Health, Inc. | Pharma-informatics system |
EP2063905B1 (de) | 2006-09-18 | 2014-07-30 | Raptor Pharmaceutical Inc | Behandlungen von lebererkrankungen durch verabreichung von konjugaten aus rezeptor-assoziierten proteinen |
PL2398500T3 (pl) | 2009-02-20 | 2019-09-30 | 2-Bbb Medicines B.V. | System dostarczania leków na bazie glutationu |
KR101741629B1 (ko) | 2009-05-06 | 2017-05-31 | 라보라토리 스킨 케어, 인크. | 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법 |
US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
CN103908548A (zh) * | 2014-04-02 | 2014-07-09 | 郭卫杰 | 一种用于治疗躁狂抑郁性精神病的中药及其制备方法 |
WO2017066705A1 (en) * | 2015-10-14 | 2017-04-20 | Aquinnah Pharmaceuticals, Inc. | Compounds, compositions and methods of use against stress granules |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL281394A (de) * | 1961-07-25 | |||
US3342826A (en) * | 1964-01-13 | 1967-09-19 | Ile De France | Heterocyclic aminoalkyl benzamides |
MC807A1 (fr) * | 1968-07-29 | 1970-07-30 | Soc Et Scient Et Ind De L Ile | Procédé de préparation de 3-alcoxy-thianaphtene-carboxamide substituées ou non |
US3860619A (en) * | 1969-05-09 | 1975-01-14 | Novo Terapeutisk Labor As | Sulphonylurea derivatives |
GB1358684A (en) * | 1970-06-15 | 1974-07-03 | Novo Terapeutisk Labor As | Carboxylic acids |
DE2152230A1 (de) * | 1971-10-20 | 1973-04-26 | Boehringer Mannheim Gmbh | Blutzuckersenkende sulfonylaminopyrimidine und verfahren zu deren herstellung |
US3953462A (en) * | 1973-10-29 | 1976-04-27 | Xeerox Corporation | Imaging process |
US4205080A (en) * | 1977-07-21 | 1980-05-27 | Shell Oil Company | 2,3-Dihydro benzofuran carboxamides |
EP0108986A1 (de) * | 1982-11-02 | 1984-05-23 | Hokuriku Pharmaceutical Co.,Ltd | N-substituierte Flavon-8-karbonsäure-amide |
-
1983
- 1983-04-08 JP JP58062554A patent/JPS59186969A/ja active Granted
-
1984
- 1984-03-20 US US06/591,363 patent/US4617314A/en not_active Expired - Fee Related
- 1984-03-21 CA CA000450167A patent/CA1238906A/en not_active Expired
- 1984-03-29 ES ES531121A patent/ES8507135A1/es not_active Expired
- 1984-04-06 EP EP84103843A patent/EP0124783B1/de not_active Expired
- 1984-04-06 DE DE8484103843T patent/DE3468024D1/de not_active Expired
- 1984-04-06 AT AT84103843T patent/ATE31307T1/de not_active IP Right Cessation
- 1984-04-07 KR KR1019840001850A patent/KR910002883B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ES531121A0 (es) | 1985-09-01 |
ATE31307T1 (de) | 1987-12-15 |
JPS6119630B2 (de) | 1986-05-17 |
KR840009092A (ko) | 1984-12-24 |
US4617314A (en) | 1986-10-14 |
KR910002883B1 (ko) | 1991-05-09 |
JPS59186969A (ja) | 1984-10-23 |
EP0124783A1 (de) | 1984-11-14 |
EP0124783B1 (de) | 1987-12-09 |
ES8507135A1 (es) | 1985-09-01 |
CA1238906A (en) | 1988-07-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |