CY2502B1 - Novel tetrazoles. - Google Patents

Novel tetrazoles.

Info

Publication number
CY2502B1
CY2502B1 CY0500012A CY0500012A CY2502B1 CY 2502 B1 CY2502 B1 CY 2502B1 CY 0500012 A CY0500012 A CY 0500012A CY 0500012 A CY0500012 A CY 0500012A CY 2502 B1 CY2502 B1 CY 2502B1
Authority
CY
Cyprus
Prior art keywords
pct
novel
tetrazoles
radical
sec
Prior art date
Application number
CY0500012A
Other languages
English (en)
Inventor
Beate Schmidt
Hermann Amschler
Wolf-Ruediger Ulrich
Thomas Martin
Thomas Baer
Rolf-Peter Hummel
Armin Hatzelmann
Hildegard Boss
Rolf Beume
Hans-Peter Kley
Dietrich Haefner
Karl-Josef Goebel
Dieter Flockerzi
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of CY2502B1 publication Critical patent/CY2502B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
CY0500012A 1997-03-07 2005-02-15 Novel tetrazoles. CY2502B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19709293 1997-03-07
EP97103924 1997-03-08

Publications (1)

Publication Number Publication Date
CY2502B1 true CY2502B1 (en) 2005-09-02

Family

ID=26034595

Family Applications (1)

Application Number Title Priority Date Filing Date
CY0500012A CY2502B1 (en) 1997-03-07 2005-02-15 Novel tetrazoles.

Country Status (12)

Country Link
US (1) US6143759A (da)
EP (1) EP0968211B1 (da)
JP (1) JP2001514640A (da)
AT (1) ATE248167T1 (da)
AU (1) AU6825898A (da)
CY (1) CY2502B1 (da)
DE (1) DE69817548T2 (da)
DK (1) DK0968211T3 (da)
ES (1) ES2206909T3 (da)
PT (1) PT968211E (da)
SI (1) SI0968211T1 (da)
WO (1) WO1998040382A1 (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR015966A1 (es) * 1997-10-17 2001-05-30 Smithkline Beecham Corp Uso de un compuesto inhibidor de pde4 para la preparacion de un medicamento util para el tratamiento de prurito
DK1109810T3 (da) * 1998-08-31 2004-10-18 Altana Pharma Ag Benzonaphthydin-N-oxider med PDE3- og PDE4-inhiberende aktivitet
WO2000042034A1 (en) * 1999-01-15 2000-07-20 Byk Gulden Phenanthridine-n-oxides with pde-iv inhibiting activity
ATE356810T1 (de) 1999-01-15 2007-04-15 Altana Pharma Ag Polysubstituted 6-phenylphenanthridines mit pde- iv hemmender wirkung
AU774868B2 (en) 1999-01-15 2004-07-08 Takeda Gmbh Phenylphenanthridines with PDE-IV inhibiting activity
CA2359404A1 (en) 1999-01-15 2000-07-20 Beate Gutterer Phenanthridine-n-oxides with pde-iv inhibiting activity
DE60026855T2 (de) 1999-08-21 2006-12-07 Altana Pharma Ag Synergistische kombination von roflumilast und salmeterol
ATE287403T1 (de) 2001-02-21 2005-02-15 Byk Gulden Lomberg Chem Fab 6-phenylbenzonaphthyidine
US6479493B1 (en) 2001-08-23 2002-11-12 Cell Pathways, Inc. Methods for treatment of type I diabetes
AU2003241903A1 (en) * 2002-05-31 2003-12-19 Takeda Pharmaceutical Company Limited Piperidine derivative, process for producing the same, and use
EP1581533A2 (en) * 2002-08-17 2005-10-05 ALTANA Pharma AG Novel benzonaphthyridines
US7470704B2 (en) * 2002-09-04 2008-12-30 Nycomed Gmbh Benzonaphthyridines
DK1723135T5 (da) 2004-03-03 2013-09-16 Takeda Gmbh Ukendte hydroxy-6-heteroarylphenanthridiner og deres anvendelse som pde4-inhibitorer
AU2005223386A1 (en) * 2004-03-17 2005-09-29 Nycomed Gmbh Novel N- (alkoxyalkyl) carbamoyl - substituted 6-phenyl-benzonaphthyridine derivatives and their use as PDE3/4 inhibitors
WO2006027345A2 (en) * 2004-09-08 2006-03-16 Altana Pharma Ag Novel 3-thia-10-aza-phenanthrene derivatives
JP5009799B2 (ja) * 2004-09-08 2012-08-22 ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規の3−オキサ−10−アザ−フェナントレン
NZ560268A (en) 2005-03-02 2010-12-24 Nycomed Gmbh Novel salts of 6-heterocyclyl substituted hexahydrophenanthridine derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3899494A (en) * 1970-05-13 1975-08-12 Sandoz Ltd Substituted 6-phenyl benzo-naphthyridines
EP0247971A3 (en) * 1986-05-29 1990-01-17 Sandoz Ag Novel pharmaceutical compositions comprising and use of cis-6-(4-acetanilido)-8,9-dimethoxy-2-methyl-1,2,3,4,4a,10b-hexahydrobenzo[c][1,6]naphthyridin
MY105344A (en) * 1990-05-16 1994-09-30 Byk Gulden Lomberg Chemische Fabrik New sulphonyl compounds

Also Published As

Publication number Publication date
DE69817548T2 (de) 2004-06-17
EP0968211B1 (en) 2003-08-27
PT968211E (pt) 2004-01-30
DE69817548D1 (de) 2003-10-02
ATE248167T1 (de) 2003-09-15
AU6825898A (en) 1998-09-29
WO1998040382A1 (en) 1998-09-17
SI0968211T1 (en) 2004-02-29
DK0968211T3 (da) 2003-12-08
US6143759A (en) 2000-11-07
JP2001514640A (ja) 2001-09-11
EP0968211A1 (en) 2000-01-05
ES2206909T3 (es) 2004-05-16

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