CY1111048T1 - Ενωσεις που εμφανιζουν αντικαρκινικη δραστηριοτητα - Google Patents

Ενωσεις που εμφανιζουν αντικαρκινικη δραστηριοτητα

Info

Publication number
CY1111048T1
CY1111048T1 CY20101100990T CY101100990T CY1111048T1 CY 1111048 T1 CY1111048 T1 CY 1111048T1 CY 20101100990 T CY20101100990 T CY 20101100990T CY 101100990 T CY101100990 T CY 101100990T CY 1111048 T1 CY1111048 T1 CY 1111048T1
Authority
CY
Cyprus
Prior art keywords
unions
cancer activity
displaying anti
displaying
cancer
Prior art date
Application number
CY20101100990T
Other languages
English (en)
Inventor
Gianfranco Peluso
Menotti Calvani
Original Assignee
Defiante Farmacêutica, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Defiante Farmacêutica, S.A. filed Critical Defiante Farmacêutica, S.A.
Publication of CY1111048T1 publication Critical patent/CY1111048T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A61K31/704Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Αποκαλύπτεται η χρήση ενώσεων του χημικού τύπου (I), όπου τα Χ, Υ και Ζ είναι όπως ορίζονται στην περιγραφή της εφεύρεσης, για την παρασκευή αντικαρκινικού φαρμάκου, προαιρετικά σε συνδυασμό με κατά διαφορετικό τρόπο βιολογικά ενεργές ουσίες.
CY20101100990T 2004-02-12 2010-11-03 Ενωσεις που εμφανιζουν αντικαρκινικη δραστηριοτητα CY1111048T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000230A ITMI20040230A1 (it) 2004-02-12 2004-02-12 Composti ad attivita' antitumorale
EP05707260A EP1713461B1 (en) 2004-02-12 2005-02-08 Compounds having antitumor activity

Publications (1)

Publication Number Publication Date
CY1111048T1 true CY1111048T1 (el) 2015-06-11

Family

ID=34856910

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20101100990T CY1111048T1 (el) 2004-02-12 2010-11-03 Ενωσεις που εμφανιζουν αντικαρκινικη δραστηριοτητα

Country Status (20)

Country Link
US (1) US7652066B2 (el)
EP (1) EP1713461B1 (el)
JP (1) JP2007522165A (el)
KR (1) KR101220331B1 (el)
CN (1) CN1917867B (el)
AR (1) AR047742A1 (el)
AT (1) ATE476973T1 (el)
AU (1) AU2005211906B2 (el)
BR (1) BRPI0507664A (el)
CA (1) CA2556069C (el)
CY (1) CY1111048T1 (el)
DE (1) DE602005022828D1 (el)
DK (1) DK1713461T3 (el)
ES (1) ES2350695T3 (el)
HK (1) HK1099687A1 (el)
IT (1) ITMI20040230A1 (el)
PL (1) PL1713461T3 (el)
SI (1) SI1713461T1 (el)
TW (1) TWI361802B (el)
WO (1) WO2005077354A1 (el)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8314144B2 (en) * 2004-02-12 2012-11-20 Defiante Farmaceutica, S.A. Compounds having antitumor activity
US8410150B2 (en) 2007-03-09 2013-04-02 University Health Network Inhibitors of carnitine palmitoyltransferase and treating cancer
CA2694724C (en) 2007-08-01 2017-09-12 University Health Network Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer
KR101225223B1 (ko) * 2008-04-29 2013-01-22 에프. 호프만-라 로슈 아게 4-다이메틸아미노부티르산 유도체
US20110230555A1 (en) * 2008-06-24 2011-09-22 David Middlemiss Enzyme Inhibitors and the Use Thereof
JP5746988B2 (ja) * 2012-02-15 2015-07-08 ライオン株式会社 カプセル皮膜及びカプセル

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1299266B1 (it) 1998-05-15 2000-02-29 Sigma Tau Ind Farmaceuti Inibitori reversibili della carnitina palmitoil trasferasi
KR20090130151A (ko) * 1999-11-12 2009-12-17 더 존스 홉킨스 유니버시티 세포내 말로닐 CoA의 수준을 증가시킴에 의한 암의 치료 방법

Also Published As

Publication number Publication date
CN1917867A (zh) 2007-02-21
AR047742A1 (es) 2006-02-15
ES2350695T3 (es) 2011-01-26
JP2007522165A (ja) 2007-08-09
KR20060134059A (ko) 2006-12-27
EP1713461B1 (en) 2010-08-11
PL1713461T3 (pl) 2011-01-31
KR101220331B1 (ko) 2013-01-09
AU2005211906B2 (en) 2009-07-30
DE602005022828D1 (de) 2010-09-23
TWI361802B (en) 2012-04-11
TW200530154A (en) 2005-09-16
CA2556069A1 (en) 2005-08-25
EP1713461A1 (en) 2006-10-25
BRPI0507664A (pt) 2007-07-17
HK1099687A1 (en) 2007-08-24
CN1917867B (zh) 2011-03-16
ATE476973T1 (de) 2010-08-15
WO2005077354A1 (en) 2005-08-25
US7652066B2 (en) 2010-01-26
US20080227683A1 (en) 2008-09-18
AU2005211906A1 (en) 2005-08-25
ITMI20040230A1 (it) 2004-05-12
DK1713461T3 (da) 2010-11-22
CA2556069C (en) 2013-04-23
SI1713461T1 (sl) 2010-12-31

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