CR20150297A - Producto de comicronización que comprende acetato de ulipristal - Google Patents
Producto de comicronización que comprende acetato de ulipristalInfo
- Publication number
- CR20150297A CR20150297A CR20150297A CR20150297A CR20150297A CR 20150297 A CR20150297 A CR 20150297A CR 20150297 A CR20150297 A CR 20150297A CR 20150297 A CR20150297 A CR 20150297A CR 20150297 A CR20150297 A CR 20150297A
- Authority
- CR
- Costa Rica
- Prior art keywords
- ulipristal acetate
- comicronization
- product
- comicronization product
- ulipristal
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Endocrinology (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Thyristors (AREA)
- Circuit Arrangements For Discharge Lamps (AREA)
- Emergency Protection Circuit Devices (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Abstract
La presente invención tiene por objeto un producto de comicronización que comprende una sustancia activa elegida entre el grupo constituido por el acetato de ulipristal, un metabolito del acetato de ulipristal y sus mezclas, y un tensioactivo sólido aceptable desde el punto de vista farmacéutico. La invención se refiere también a una composición farmacéutica que comprende dicho producto de comicronización y sus utilizaciones terapéuticas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1260603A FR2997627B1 (fr) | 2012-11-08 | 2012-11-08 | Produit de co-micronisation comprenant de l'ulipristal acetate |
PCT/FR2013/052670 WO2014072646A1 (fr) | 2012-11-08 | 2013-11-07 | Produit de co-micronisation comprenant de l'ulipristal acetate |
Publications (1)
Publication Number | Publication Date |
---|---|
CR20150297A true CR20150297A (es) | 2015-08-14 |
Family
ID=47878175
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR20150297A CR20150297A (es) | 2012-11-08 | 2015-06-05 | Producto de comicronización que comprende acetato de ulipristal |
Country Status (30)
Country | Link |
---|---|
US (2) | US9610293B2 (es) |
EP (1) | EP2916871B1 (es) |
JP (1) | JP2015536968A (es) |
KR (1) | KR20150093170A (es) |
CN (1) | CN104902928B (es) |
AR (1) | AR093402A1 (es) |
AU (1) | AU2013343320B2 (es) |
BR (1) | BR112015010271B1 (es) |
CA (1) | CA2890272A1 (es) |
CR (1) | CR20150297A (es) |
CY (1) | CY1119542T1 (es) |
DK (1) | DK2916871T3 (es) |
EA (1) | EA027641B1 (es) |
EC (1) | ECSP15022442A (es) |
ES (1) | ES2606307T3 (es) |
FR (1) | FR2997627B1 (es) |
GE (1) | GEP201706637B (es) |
HR (1) | HRP20161624T1 (es) |
HU (1) | HUE031911T2 (es) |
LT (1) | LT2916871T (es) |
MD (1) | MD4563C1 (es) |
MX (1) | MX363699B (es) |
PL (1) | PL2916871T3 (es) |
PT (1) | PT2916871T (es) |
RS (1) | RS55429B1 (es) |
SI (1) | SI2916871T1 (es) |
SM (1) | SMT201600445B (es) |
TW (1) | TWI617325B (es) |
UA (1) | UA117465C2 (es) |
WO (1) | WO2014072646A1 (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2997627B1 (fr) * | 2012-11-08 | 2015-01-16 | Hra Pharma Lab | Produit de co-micronisation comprenant de l'ulipristal acetate |
CN103923154B (zh) * | 2013-01-16 | 2017-09-26 | 杭州容立医药科技有限公司 | 醋酸乌利司他的共晶及制备方法 |
CN105663140A (zh) * | 2014-11-21 | 2016-06-15 | 四川海思科制药有限公司 | 一种含醋酸乌利司他的药物组合物及其制备方法 |
CN104865215A (zh) * | 2015-05-16 | 2015-08-26 | 南京海纳医药科技有限公司 | 一种醋酸乌利司他片剂及其溶出度测定方法 |
CN105919150A (zh) * | 2016-05-12 | 2016-09-07 | 高洁珺 | 一种代替压片工艺中化工添加剂的方法 |
CN106265533A (zh) * | 2016-10-10 | 2017-01-04 | 朱隆娅 | 一种阿德呋啉颗粒剂及其制备方法 |
FR3060389B1 (fr) | 2016-12-20 | 2019-05-31 | Laboratoire Hra-Pharma | Comprime enrobe comprenant de l'ulipristal acetate ou un de ses metabolites |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2627696B1 (fr) | 1988-02-26 | 1991-09-13 | Fournier Innovation Synergie | Nouvelle forme galenique du fenofibrate |
US4954490A (en) | 1988-06-23 | 1990-09-04 | Research Triangle Institute | 11 β-substituted progesterone analogs |
GB9608719D0 (en) | 1996-04-26 | 1996-07-03 | Scherer Ltd R P | Pharmaceutical compositions |
FR2757397B1 (fr) * | 1996-12-23 | 1999-03-05 | Mazal Pharma | Composition pharmaceutique a base de rheine ou de diacerheine a biodisponibilite amelioree |
IL127129A (en) * | 1998-11-18 | 2004-06-01 | Ferring Bv | Method for preparation of progesterone tablets for vaginal delivery and tablets so prepared |
FR2821555B1 (fr) * | 2001-03-01 | 2003-05-16 | Besins Int Lab | Progestatif co-micronise avec un tensioactif, composition pharmaceutique le comprenant, leurs procedes de fabrication et leurs utilisations |
FR2841138B1 (fr) * | 2002-06-25 | 2005-02-25 | Cll Pharma | Composition pharmaceutique solide contenant un principe actif lipophile, son procede de preparation |
ES2212912B1 (es) | 2003-01-22 | 2005-10-01 | Crystal Pharma, S.A. | Procedimiento para la obtencion de 17alfa-acetoxi-11beta-(4-n,n-dimetilaminofenil)-19-norpregna-4,9-dien-3,20-diona. |
WO2006010097A2 (en) | 2004-07-09 | 2006-01-26 | The Population Council, Inc. | Sustained release compositions containing progesterone receptor modulators |
WO2008037044A1 (en) | 2006-09-27 | 2008-04-03 | Medley S.A. Indústria Farmacêutica | Oxcarbazepine-containing oral formulation and a process to obtain the same |
BRPI0719486A2 (pt) | 2006-12-20 | 2014-02-18 | Duramed Pharmaceuticals Inc | "forma farmacêutica sólida oral desitegrante, não-efervescente, métodos para tratar uma mulher que necessite de um contraceptivo de emergência, pacote terapêutico para tratar uma mulher que necessite de contracepção de emergência e processo para a preparação de uma forma sólida de dosagem farmacêutica oral desintegrante, não-efervescente" |
JP2010514793A (ja) * | 2006-12-28 | 2010-05-06 | レプロス セラピューティクス インコーポレイティド | 抗プロゲスチンのバイオアベイラビリティを改善するための方法および製剤 |
EP2062572A1 (en) * | 2007-11-19 | 2009-05-27 | Teva Pharmaceutical Industries Ltd. | Pharmaceutical compositions |
US8299050B2 (en) | 2008-01-29 | 2012-10-30 | Laboratoire Hra-Pharma | Method for treating uterine fibroids |
US8512745B2 (en) * | 2008-12-08 | 2013-08-20 | Laboratoire Hra Pharma | Ulipristal acetate tablets |
ME02548B (me) | 2009-04-14 | 2017-02-20 | Hra Pharma Lab | Postupak za kontracepciju po potrebi |
EP2471537A1 (en) * | 2010-12-30 | 2012-07-04 | PregLem S.A. | Treatment of pain associated with dislocation of basal endometrium |
FR2997627B1 (fr) * | 2012-11-08 | 2015-01-16 | Hra Pharma Lab | Produit de co-micronisation comprenant de l'ulipristal acetate |
-
2012
- 2012-11-08 FR FR1260603A patent/FR2997627B1/fr not_active Expired - Fee Related
-
2013
- 2013-07-11 UA UAA201505665A patent/UA117465C2/uk unknown
- 2013-11-07 RS RS20161080A patent/RS55429B1/sr unknown
- 2013-11-07 WO PCT/FR2013/052670 patent/WO2014072646A1/fr active Application Filing
- 2013-11-07 EA EA201500513A patent/EA027641B1/ru not_active IP Right Cessation
- 2013-11-07 US US14/441,027 patent/US9610293B2/en not_active Expired - Fee Related
- 2013-11-07 GE GEAP201313847A patent/GEP201706637B/en unknown
- 2013-11-07 PT PT138016399T patent/PT2916871T/pt unknown
- 2013-11-07 PL PL13801639T patent/PL2916871T3/pl unknown
- 2013-11-07 EP EP13801639.9A patent/EP2916871B1/fr active Active
- 2013-11-07 KR KR1020157015210A patent/KR20150093170A/ko not_active Application Discontinuation
- 2013-11-07 AR ARP130104089A patent/AR093402A1/es unknown
- 2013-11-07 DK DK13801639.9T patent/DK2916871T3/da active
- 2013-11-07 BR BR112015010271A patent/BR112015010271B1/pt not_active IP Right Cessation
- 2013-11-07 CN CN201380058466.0A patent/CN104902928B/zh not_active Expired - Fee Related
- 2013-11-07 MX MX2015005762A patent/MX363699B/es unknown
- 2013-11-07 SI SI201330409A patent/SI2916871T1/sl unknown
- 2013-11-07 CA CA2890272A patent/CA2890272A1/fr not_active Abandoned
- 2013-11-07 JP JP2015541214A patent/JP2015536968A/ja active Pending
- 2013-11-07 ES ES13801639.9T patent/ES2606307T3/es active Active
- 2013-11-07 HU HUE13801639A patent/HUE031911T2/en unknown
- 2013-11-07 AU AU2013343320A patent/AU2013343320B2/en not_active Ceased
- 2013-11-07 MD MDA20150053A patent/MD4563C1/ro not_active IP Right Cessation
- 2013-11-07 LT LTEP13801639.9T patent/LT2916871T/lt unknown
- 2013-11-08 TW TW102140765A patent/TWI617325B/zh not_active IP Right Cessation
-
2015
- 2015-06-05 CR CR20150297A patent/CR20150297A/es unknown
- 2015-06-05 EC ECIEPI201522442A patent/ECSP15022442A/es unknown
-
2016
- 2016-11-29 CY CY20161101236T patent/CY1119542T1/el unknown
- 2016-12-02 HR HRP20161624TT patent/HRP20161624T1/hr unknown
- 2016-12-07 SM SM201600445T patent/SMT201600445B/it unknown
-
2017
- 2017-02-16 US US15/434,650 patent/US20170157146A1/en not_active Abandoned
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CR20150297A (es) | Producto de comicronización que comprende acetato de ulipristal | |
GT201500053A (es) | Composicion farmaceutica recubierta que contiene regorafenib | |
CL2015002164A1 (es) | Formulación combinada de dos compuesos antivirales. | |
CL2015000295A1 (es) | Compuestos derivados de alquilpirimidina; composicion farmaceutica que los comprende; uso para el tratamiento de infecciones víricas y otras enfermedades. | |
CU24486B1 (es) | Dispersión sólida amorfa que comprende taxano, tabletas comprendiendo la misma y método para prepararla | |
BR112016008576A2 (pt) | Formulações aquosas estáveis de anticorpos e forma farmacêutica de dosagem unitária | |
CL2016002091A1 (es) | Compuesto de triazina y su uso para fines medicinales | |
PE20140255A1 (es) | Tableta dispersable en forma oral | |
CL2016001918A1 (es) | Heteroaril amidas como inhibidores de agregación de proteína | |
CL2014001838A1 (es) | Compuestos derivados de fluormetil-5,6-dihidro-4h-[1,3]oxazin-2-ilamina, como inhibidores de la bace1; su proceso de obtencion; composicion farmaceutica que los contiene; y su uso para el tratamiento terapeutico y/o profilactico de la enfermedad de alzheimer, esclerosis lateral amiotrofica, cancer, enfermedades cardiovasculares y enfermedades gastrointestinales, entre otras. | |
CL2017001483A1 (es) | Formulación de relación fija de insulina glargina/lixisenatida | |
CR20160438A (es) | Dispersión sólida amorfa que comprende taxano, comprimido que comprende la misma, y método para su preparación | |
IN2014MN02236A (es) | ||
CL2015002832A1 (es) | Formulación farmaceutica que comprende fosfatidilcolina para el tratamiento de colitus ulcerosa. | |
BR112014032583A2 (pt) | forma farmacêutica para liberação prolongada de substâncias ativas | |
MX2015016410A (es) | Esteres de acidos oligo-hidroxicarboxilicos y uso de los mismos. | |
MX2017015322A (es) | Composicion farmaceutica oral de isotretinoin. | |
EA201691741A1 (ru) | Фармацевтическая композиция | |
MX2015016490A (es) | Esteres sulfatados de acidos oligohidroxicarboxilicos, y uso de los mismos. | |
AR093252A1 (es) | Composicion farmaceutica oral utilizada como antiparasitaria y antidiarreica y procesos para prepararla | |
CL2015000290A1 (es) | Compuestos derivados de ariletinilo. moduladores alostéricos del receptor de glutamato mglur5; proceso de obtencion; composicion farmaceuticas: y su uso en el tratamiento o prevencon de la esquizofenia, enfermedades cognitivas, sindrome de x fragil o autismo | |
WO2015087343A3 (en) | An improved process for the preparation of nilotinib and pharmaceutically acceptable salts thereof | |
WO2015031198A3 (en) | Bendamustine pharmaceutical compositions | |
BR112015021769A2 (pt) | composições farmacêuticas compreendendo um agente ativo | |
IN2014DN07897A (es) |