CO6700858A2 - Lactams substituted by piperidinyl as modulators of gpr119 - Google Patents

Lactams substituted by piperidinyl as modulators of gpr119

Info

Publication number
CO6700858A2
CO6700858A2 CO13098019A CO13098019A CO6700858A2 CO 6700858 A2 CO6700858 A2 CO 6700858A2 CO 13098019 A CO13098019 A CO 13098019A CO 13098019 A CO13098019 A CO 13098019A CO 6700858 A2 CO6700858 A2 CO 6700858A2
Authority
CO
Colombia
Prior art keywords
gpr119
modulators
piperidinyl
lactams
substituted
Prior art date
Application number
CO13098019A
Other languages
Spanish (es)
Inventor
Thomas Daniel Aicher
Josef Bencsik
Steven A Boyd
Kevin Ronald Condroski
Jay Bradford Fell
John P Fischer
Ronald Hinklin
Scott Alan Pratt
Ajay Singh
Timothy Turner
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Priority to CO13098019A priority Critical patent/CO6700858A2/en
Publication of CO6700858A2 publication Critical patent/CO6700858A2/en

Links

Abstract

Compuestos de Fórmula I:y sales farmacéuticamente aceptables de los mismos donde X, X, L, R, R, R, Ry n tienen los significados dados en la memoria descriptiva, son moduladores de GPR119 y son útiles en el tratamiento o prevención de enfermedades tales como pero sin limitación a, diabetes tipo 2, complicaciones diabéticas, síntomas de diabetes, síndrome metabólico, obesidad, dislipidemia y afecciones relacionadas.Compounds of Formula I: and pharmaceutically acceptable salts thereof where X, X, L, R, R, R, Ry n have the meanings given in the specification, are modulators of GPR119 and are useful in the treatment or prevention of diseases such as but not limited to, type 2 diabetes, diabetic complications, diabetes symptoms, metabolic syndrome, obesity, dyslipidemia and related conditions.

CO13098019A 2013-04-16 2013-04-16 Lactams substituted by piperidinyl as modulators of gpr119 CO6700858A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CO13098019A CO6700858A2 (en) 2013-04-16 2013-04-16 Lactams substituted by piperidinyl as modulators of gpr119

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CO13098019A CO6700858A2 (en) 2013-04-16 2013-04-16 Lactams substituted by piperidinyl as modulators of gpr119

Publications (1)

Publication Number Publication Date
CO6700858A2 true CO6700858A2 (en) 2013-06-28

Family

ID=49118227

Family Applications (1)

Application Number Title Priority Date Filing Date
CO13098019A CO6700858A2 (en) 2013-04-16 2013-04-16 Lactams substituted by piperidinyl as modulators of gpr119

Country Status (1)

Country Link
CO (1) CO6700858A2 (en)

Similar Documents

Publication Publication Date Title
UY33614A (en) READING REPLACED BY PIPERIDINYL AS MODULATORS OF GPR119
CO6670520A2 (en) Lactmas substituted with piperidinium as modulators of gpr119
ECSP22091792A (en) SUBSTITUTED TRICYCLIC COMPOUNDS AS INHIBITORS OF THE FIBROPLAST GROWTH FACTOR RECEPTOR
CY1124000T1 (en) SUBSTITUTED 5-FLUORO-1H-PYRAZOLOPYRIDINES IN CRYSTALLINE FORM
NI201300074A (en) NOVEL DERIVATIVES OF CYCLIC AZABENZIMIDAZOLE USEFUL AS ANTIDIABETIC AGENTS.
CR20150078A (en) 1,4-DISPOSED PIRIDAZINE ANALOGS AND METHODS FOR THE TREATMENT OF CONDITIONS RELATED TO THE DEFICIENCY OF SMN
NI201400043A (en) 4 - PHENYL - PYRIDINES SUBSTITUTED FOR THE TREATMENT OF DISEASES RELATED TO THE NK1 RECEPTOR
CO6771441A2 (en) Triazolopyridine compounds as pim kinase inhibitors
CR20140142A (en) VARIANTS OF THE FIBROBLAST GROWTH 21
EA201690107A1 (en) PHARMACEUTICAL COMPOSITION CONTAINING DIMETHYLFUMATE FOR INTRODUCTION TO LOW DAILY DOSE
BR112013002957A2 (en) 1,4,5,6-tetrahydro-pyrimidin-2-ylamine
EA201491335A1 (en) BIGUANID COMPOSITIONS AND METHODS OF TREATMENT OF METABOLIC DISORDERS
UY35171A (en) DERIVATIVES OF INDANILOXIDIHIDROBENZOFURANILACÉTIC ACIDS AS AGONISTS OF THE GPR40
CR20110255A (en) NEW COMPOUNDS 578
UY34859A (en) Peptide analogs of exendin 4.
EA201690582A1 (en) MODULATORS OF COMPLEMENT FACTOR
EA201590951A1 (en) DIHYDROPYRAZOL GPR40 MODULATORS
EA201491857A1 (en) Α7 nicotinic holinoreceptor allosteric modulators, their derivatives and their application
PE20151595A1 (en) PIRAZOL-AMIDE COMPOUNDS AND THEIR PHARMACEUTICAL USES
EA201590949A1 (en) DIHYDROPYRAZOL GPR40 MODULATORS
EA201590954A1 (en) DIHYDROPYRAZOL GPR40 MODULATORS
BR112014031091A2 (en) PIPERIDINE DERIVATIVES FOR GPR119 AGONIST
UY34964A (en) CHROMAN DERIVATIVES AS INHIBITORS OF THE MELASTATIN POTENTIAL TRANSITORY RECEIVER 8 (TRPM8)
CO6741223A2 (en) Azetidine derivatives useful for the treatment of metabolic and inflammatory diseases
UY33509A (en) METHODS AND COMPOSITIONS FOR ALLERGY TREATMENT

Legal Events

Date Code Title Description
FG Application granted