CO6592108A2 - Agonista alfa -2 adrenergico que tiene larga duración en el efecto reductor de la presión intraocular - Google Patents
Agonista alfa -2 adrenergico que tiene larga duración en el efecto reductor de la presión intraocularInfo
- Publication number
- CO6592108A2 CO6592108A2 CO12140238A CO12140238A CO6592108A2 CO 6592108 A2 CO6592108 A2 CO 6592108A2 CO 12140238 A CO12140238 A CO 12140238A CO 12140238 A CO12140238 A CO 12140238A CO 6592108 A2 CO6592108 A2 CO 6592108A2
- Authority
- CO
- Colombia
- Prior art keywords
- intraocular pressure
- alpha
- long duration
- reducing effect
- adrenergic agonist
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Ophthalmology & Optometry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona un método para reducir la presión intraocular que comprende administrar una cantidad terapéuticamente eficaz de una composición farmacéutica que comprende 4-bromo-5- (2-imidazólin-2-ilamino)bencimidazol o una de sus sales en el ojo afectado de un paciente, en una dosis única, en el cual el ojo afectado tiene una presión intraocular menor que la presión intraocular basal durante al menos ocho (8) horas.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US29691210P | 2010-01-21 | 2010-01-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
CO6592108A2 true CO6592108A2 (es) | 2013-01-02 |
Family
ID=44169074
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO12140238A CO6592108A2 (es) | 2010-01-21 | 2012-08-17 | Agonista alfa -2 adrenergico que tiene larga duración en el efecto reductor de la presión intraocular |
Country Status (17)
Country | Link |
---|---|
US (1) | US9889088B2 (es) |
EP (1) | EP2525793B1 (es) |
JP (3) | JP2013518051A (es) |
KR (1) | KR20120125305A (es) |
CN (1) | CN102770135A (es) |
AU (1) | AU2011207301A1 (es) |
BR (1) | BR112012018154A2 (es) |
CA (1) | CA2787573A1 (es) |
CL (1) | CL2012002038A1 (es) |
CO (1) | CO6592108A2 (es) |
IL (1) | IL221030A0 (es) |
MX (1) | MX2012008516A (es) |
RU (1) | RU2012134065A (es) |
SG (1) | SG182637A1 (es) |
TW (1) | TW201141477A (es) |
WO (1) | WO2011091225A2 (es) |
ZA (1) | ZA201205470B (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013016072A1 (en) * | 2011-07-22 | 2013-01-31 | Allergan, Inc. | Pharmaceutical compositions comprising 4-bromo-n-(imidazolidin-2-ylidene)-1h-benzimidazol-5-amine for treating skin diseases |
EP2734200A1 (en) * | 2011-07-22 | 2014-05-28 | Allergan, Inc. | Alpha-2 adrenergic modulators for treating visual disorders mediated by central visual projections from the eye |
US20130046003A1 (en) * | 2011-07-22 | 2013-02-21 | Mohammed I. Dibas | Pharmaceutical compositions comprising 4-bromo-n-(imidazolidin-2-ylidene)-1h-benzimidazol-5-amine for treating retinal diseases |
CA2900671A1 (en) * | 2013-03-14 | 2014-10-02 | Allergan, Inc. | Alpha-2 adrenergic agonist for treating intraocular pressure and ocular diseases through intravitreal and intracameral routes |
TWI699205B (zh) * | 2014-12-12 | 2020-07-21 | 日商興和股份有限公司 | 用於預防或治療青光眼之藥物療法 |
EP3647420B1 (en) | 2017-06-27 | 2023-08-23 | The University Of Tokyo | Probe and method for detecting transcript resulting from fusion gene and/or exon skipping |
US11077053B2 (en) | 2018-08-21 | 2021-08-03 | Allergan, Inc. | Alpha-2-adrenergic receptor agonists for treatment of presbyopia, visual glare, visual starbursts, visual halos and night myopia |
TW202233170A (zh) * | 2020-11-02 | 2022-09-01 | 美商偉視醫療股份有限公司 | 藥物中的降解化合物 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5478858A (en) * | 1993-12-17 | 1995-12-26 | The Procter & Gamble Company | 5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists |
AU704972B2 (en) * | 1994-08-04 | 1999-05-13 | H. Lundbeck A/S | Novel benzimidazole derivatives |
US6495583B1 (en) * | 1997-03-25 | 2002-12-17 | Synaptic Pharmaceutical Corporation | Benzimidazole derivatives |
US20050244463A1 (en) * | 2004-04-30 | 2005-11-03 | Allergan, Inc. | Sustained release intraocular implants and methods for treating ocular vasculopathies |
CA2603044A1 (en) * | 2005-06-29 | 2007-01-11 | Allergan, Inc. | Alpha-2 adrenergic agonists for the treatment of pain |
EP1981852A1 (en) | 2006-02-06 | 2008-10-22 | NicOx S.A. | Nitrooxy-comprising derivatives of apraclonidine and brimodnidine as al pha2 -adrenergic receptor agonists |
US8821870B2 (en) * | 2008-07-18 | 2014-09-02 | Allergan, Inc. | Method for treating atrophic age related macular degeneration |
-
2011
- 2011-01-21 WO PCT/US2011/022001 patent/WO2011091225A2/en active Application Filing
- 2011-01-21 SG SG2012053815A patent/SG182637A1/en unknown
- 2011-01-21 RU RU2012134065/15A patent/RU2012134065A/ru unknown
- 2011-01-21 KR KR1020127021719A patent/KR20120125305A/ko not_active Application Discontinuation
- 2011-01-21 TW TW100102411A patent/TW201141477A/zh unknown
- 2011-01-21 US US13/010,958 patent/US9889088B2/en active Active
- 2011-01-21 CA CA2787573A patent/CA2787573A1/en not_active Abandoned
- 2011-01-21 BR BR112012018154A patent/BR112012018154A2/pt not_active IP Right Cessation
- 2011-01-21 JP JP2012550140A patent/JP2013518051A/ja active Pending
- 2011-01-21 EP EP11702342.4A patent/EP2525793B1/en active Active
- 2011-01-21 AU AU2011207301A patent/AU2011207301A1/en not_active Abandoned
- 2011-01-21 CN CN2011800111530A patent/CN102770135A/zh active Pending
- 2011-01-21 MX MX2012008516A patent/MX2012008516A/es unknown
-
2012
- 2012-07-19 IL IL221030A patent/IL221030A0/en unknown
- 2012-07-20 CL CL2012002038A patent/CL2012002038A1/es unknown
- 2012-07-20 ZA ZA2012/05470A patent/ZA201205470B/en unknown
- 2012-08-17 CO CO12140238A patent/CO6592108A2/es not_active Application Discontinuation
-
2015
- 2015-10-28 JP JP2015211447A patent/JP2016026206A/ja active Pending
-
2017
- 2017-04-26 JP JP2017086952A patent/JP6466504B2/ja active Active
Also Published As
Publication number | Publication date |
---|---|
TW201141477A (en) | 2011-12-01 |
ZA201205470B (en) | 2013-05-29 |
AU2011207301A1 (en) | 2012-08-09 |
CL2012002038A1 (es) | 2012-11-16 |
IL221030A0 (en) | 2012-09-24 |
WO2011091225A2 (en) | 2011-07-28 |
US9889088B2 (en) | 2018-02-13 |
BR112012018154A2 (pt) | 2016-04-05 |
KR20120125305A (ko) | 2012-11-14 |
SG182637A1 (en) | 2012-08-30 |
MX2012008516A (es) | 2012-10-15 |
JP2017125074A (ja) | 2017-07-20 |
CA2787573A1 (en) | 2011-07-28 |
EP2525793B1 (en) | 2018-09-05 |
JP2016026206A (ja) | 2016-02-12 |
RU2012134065A (ru) | 2014-02-27 |
CN102770135A (zh) | 2012-11-07 |
EP2525793A2 (en) | 2012-11-28 |
US20110178145A1 (en) | 2011-07-21 |
JP6466504B2 (ja) | 2019-02-06 |
WO2011091225A3 (en) | 2012-05-18 |
JP2013518051A (ja) | 2013-05-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CO6592108A2 (es) | Agonista alfa -2 adrenergico que tiene larga duración en el efecto reductor de la presión intraocular | |
DOP2011000104A (es) | Combinacion de una insulina y un agonista de glp-1 | |
CY1121041T1 (el) | Μεθοδοι αγωγης παιδιατρικων ασθενων με τη χρηση δεξμεδετομιδινης | |
CY1122648T1 (el) | Διαδικασια για την παρασκευη συνθεσεων που περιεχουν υαλουρονικο οξυ και υδροχλωρικη μεπιβακαϊνη | |
CL2017000156A1 (es) | Procedimientos para el tratamiento de paramixovirus. | |
GT201200217A (es) | Derivados de 3-hidroxi-5-arilisotiazol novedosos | |
BR112015022972A2 (pt) | composição farmacêutica de cloridrato de s-cetamina | |
CL2011001529A1 (es) | Uso de un modulador o agonista de los receptores s1p derivado de 2-amino-propan-1,3-diol o 2-amino-propanol para tratar una enfermedad cronica larga en un sujeto, de manera de conseguir una disminucion diaria en la frecuencia cardiaca de 2 latidos/minutos o menos; y kit que lo comprende. | |
TN2011000281A1 (en) | Dosage regimen of an s1p receptor agonist | |
BR112015022465A2 (pt) | método para tratamento não-tóxico para síndrome de abstinência de drogas | |
BR112013008601A8 (pt) | Formulações de emulsão de clevidipina contendo agentes antimicrobianos | |
CR20110110A (es) | Composicion farmaceutica | |
ES2721900T3 (es) | Polvo y suspensión acuosa de liberación prolongada que comprende metilfenidato | |
AR089509A1 (es) | Metodo para tratar la perdida osea alveolar, un implante dental, un anticuerpo antiesclerostina, un gel o matriz que comprende dicho anticuerpo y uso | |
CR20120663A (es) | Combinaciones que comprenden antisicóticos atípicos y agonistas taar1 | |
MX2013002422A (es) | Sales de lorcaserina con acidos opticamente activos. | |
AR092993A1 (es) | Laquinimod para reducir el daño talamico en la esclerosis multiple | |
PH12015502282A1 (en) | Alpha-2 adrenoceptor and sigma receptor ligand combinations | |
UA110979C2 (uk) | Рідка фармацевтична композиція, яка включає нітизинон | |
CL2015000434A1 (es) | Metodo para el tratamiento, prevencion o disminucion de la severidad de una condicion o trastorno no neoplasico de la piel que comprende administrar un compuesto derivado de retinoides; composicion dermica que comprende los derivados de retinoide. | |
NZ706990A (en) | A veterinary method of alleviating noise aversion | |
EA201390616A1 (ru) | ЛЕЧЕНИЕ НАРУШЕНИЙ, АССОЦИИРОВАННЫХ С ГЕНОМ MeCP2 | |
CL2012003341A1 (es) | Composicion farmaceutica de administracion oral que compende bendamustina o un ester, una sal o un solvato de la misma, y un excipiente que es un agente tensioactivo no ionico e hidrofilico; combinacion farmaceutica; y su uso para el tratamiento de leucemia linfocitica cronica y el mieloma multiple, entre otras enfermedades. | |
AR090929A1 (es) | Identificacion de la respuesta de un paciente a la administracion del modulador del receptor de s1p | |
AR085523A1 (es) | Mecanismo de establecimiento de dosis y dispositivo de inyeccion |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC | Application refused |