CO6321187A2 - DERIVATIVES OF QUINOLINA AND ITS USE AS A FUNGICIDE - Google Patents

DERIVATIVES OF QUINOLINA AND ITS USE AS A FUNGICIDE

Info

Publication number
CO6321187A2
CO6321187A2 CO10081942A CO10081942A CO6321187A2 CO 6321187 A2 CO6321187 A2 CO 6321187A2 CO 10081942 A CO10081942 A CO 10081942A CO 10081942 A CO10081942 A CO 10081942A CO 6321187 A2 CO6321187 A2 CO 6321187A2
Authority
CO
Colombia
Prior art keywords
alkyl
alkoxy
halo
hydrogen
optionally substituted
Prior art date
Application number
CO10081942A
Other languages
Spanish (es)
Inventor
Fiona Murphy Kessabi
Laura Quaranta
Renaud Beaudegnies
Hans-Georg Brunner
Fredrick Ceberbaum
Original Assignee
Syngenta Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Ltd filed Critical Syngenta Ltd
Publication of CO6321187A2 publication Critical patent/CO6321187A2/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Quinoline Compounds (AREA)

Abstract

1.- Un compuesto de la fórmula general Ien donde Q1 es hidrógeno, alquilo C1-4, trialquilsilanilo C1-4, hidroxi- alquilo C1-6, alcoxi-alquilo C1-6, halo-alquilo C1-6, o halógeno, Q2 y Q3, en forma independiente, son hidrógeno, alquilo C1-3, halo-alquilo C1-3, o halógeno, R1 es alquilo C1-4, halo-alquilo(C1-4), cicloalquilo C3-4, alcoxi C1-4, halo-alcoxi (C1-4), cicloalcoxi C3-4, alquiltio C1-4, alquilsulfinilo C1-4, alquilsulfonilo C1-4, halo-alquiltio(C1-4), halo-alquilsulfinilo(C1-4), halo-alquilsulfonilo(C1-4), cicloalquiltio C3-4, cicloalquilsulfinilo C3-4, o cicloalquilsulfonilo C3-4, R2 es hidrógeno, alquilo C1-6, cicloalquilo C3-4, alquenilo C2-8, ciano, hidroxi, alcoxi C1-4, halo-alquilo(C1-4), ciano- alquilo(C1-4), alcoxi C1-4 alquilo(C1-4), alcoxi C1-4 alcoxi(C1-4)alquilo(C1-4) o benciloxi alquilo(C1-4), en donde el anillo fenilo está opcionalmente sustituido con alcoxi C1-4, R3 es -(CRaRb)p(CRcRd)q(X)r(CReRf)sR4, en dondeRa, Rb, Rc, Rd, Re, y Rf, en forma independiente, son hidrógeno, alquilo C1-6, halógeno, halo alquilo(C1-6), hidroxi alquilo(C1-6), alcoxi C1-4 alquilo(C1-4), alqueniloxi C3-5alquilo(C1-4), alquiniloxi C3-5 -alquilo C1-4, alquenilo C2-5 o alquinilo C2-5, ciano, hidroxi, alcoxi C1-4, alqueniloxi C3-5, alquiniloxi C3-5 o alcoxicarbonilo C1-4, o RaRb, RcRd o ReRf se pueden unir para formar un anillo heterocíclico o carbocíclico de 3 a 8 miembros que contiene un heterátomo seleccionado de azufre, oxígeno y NR0, en donde R0 es hidrógeno o alquilo C1-6 opcionalmente sustituido, donde el anillo heterocíclico o carbocíclico está opcionalmente sustituido con halo o alquilo C1-4, X es (CO), (CO)O, O(CO), O o S(O)t, en donde t es 0, 1 ó 2, o X es NH o N alquilo(C1-6), p, r y s, en forma independiente, son 0 ó 1,Q es 0, 1 ó 2, R4 es hidrógeno, alquilo C1-6 opcionalmente sustituido, formilo, ciano, alquenilo C2-6 opcionalmente sustituido, o -C=C-R5, en donde R5 es hidrógeno, alquilo C1-8 opcionalmente sustituido con halógeno, hidroxi, alcoxi C1-6, alcoxi C1-3alcoxi(C1-3), ciano, alquilcarboniloxi C1-4, aminocarboniloxi, mono- o di-aIquilaminocarboniloxi(C1-4), trialquilsililoxi(C1-4), ...1.- A compound of the general formula Ien wherein Q1 is hydrogen, C1-4 alkyl, C1-4 trialkylsilyl, C1-6 hydroxy alkyl, C1-6 alkoxy alkyl, halo C1-6 alkyl, or halogen, Q2 and Q3, independently, are hydrogen, C1-3 alkyl, halo-C1-3 alkyl, or halogen, R1 is C1-4 alkyl, halo-C1-4 alkyl, C3-4 cycloalkyl, C1-4 alkoxy , halo (C1-4) alkoxy, C3-4 cycloalkoxy, C1-4 alkylthio, C1-4 alkylsulfinyl, C1-4 alkylsulfonyl, halo (C1-4) alkyl, halo (C1-4) alkylsulfinyl, halo- C 1-4 alkylsulfonyl, C 3-4 cycloalkylthio, C 3-4 cycloalkylsulfinyl, or C 3-4 cycloalkylsulfonyl, R 2 is hydrogen, C 1-6 alkyl, C 3-4 cycloalkyl, C 2-8 alkenyl, cyano, hydroxy, C 1-4 alkoxy , halo (C1-4) alkyl, cyano- (C1-4) alkyl, C1-4 alkoxy (C1-4) alkyl, C1-4 alkoxy (C1-4) alkoxy or benzyloxy alkyl ( C1-4), where the phenyl ring is optionally substituted with C1-4 alkoxy, R3 is - (CRaRb) p (CRcRd) q (X) r (CReRf) sR4, whereRa, Rb, Rc, Rd, Re, and Rf, independently e, are hydrogen, C1-6 alkyl, halogen, halo (C1-6) alkyl, hydroxy (C1-6) alkyl, C1-4 alkoxy (C1-4) alkyl, C3-5 alkenyloxy (C1-4) alkyl, alkynyloxy C3-5 -C1-4 alkyl, C2-5 alkenyl or C2-5 alkynyl, cyano, hydroxy, C1-4 alkoxy, C3-5 alkyloxy, C3-5 alkynyloxy or C1-4 alkoxycarbonyl, or RaRb, RcRd or ReRf se they can join to form a 3- to 8-membered heterocyclic or carbocyclic ring containing a heteratome selected from sulfur, oxygen and NR0, wherein R0 is hydrogen or optionally substituted C1-6 alkyl, where the heterocyclic or carbocyclic ring is optionally substituted with halo or C1-4 alkyl, X is (CO), (CO) O, O (CO), O or S (O) t, where t is 0, 1 or 2, or X is NH or N (C1-) alkyl 6), p, rys, independently, are 0 or 1, Q is 0, 1 or 2, R4 is hydrogen, optionally substituted C1-6 alkyl, formyl, cyano, optionally substituted C2-6 alkenyl, or -C = C-R5, wherein R5 is hydrogen, C1-8 alkyl optionally substituted with halogen, hi droxy, C1-6 alkoxy, C1-3 alkoxy (C1-3) alkoxy, cyano, C1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di-alkylaminocarbonyloxy (C1-4), trialkylsilyloxy (C1-4), ...

CO10081942A 2008-01-10 2010-07-07 DERIVATIVES OF QUINOLINA AND ITS USE AS A FUNGICIDE CO6321187A2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0800407.9A GB0800407D0 (en) 2008-01-10 2008-01-10 Fungicides

Publications (1)

Publication Number Publication Date
CO6321187A2 true CO6321187A2 (en) 2011-09-20

Family

ID=39144717

Family Applications (1)

Application Number Title Priority Date Filing Date
CO10081942A CO6321187A2 (en) 2008-01-10 2010-07-07 DERIVATIVES OF QUINOLINA AND ITS USE AS A FUNGICIDE

Country Status (26)

Country Link
US (1) US8415272B2 (en)
EP (1) EP2231614B1 (en)
JP (1) JP2011509271A (en)
KR (1) KR20100109952A (en)
CN (2) CN101910135B (en)
AR (1) AR070135A1 (en)
AT (1) ATE546433T1 (en)
AU (1) AU2009203826B2 (en)
BR (1) BRPI0907184A2 (en)
CA (1) CA2711094A1 (en)
CL (1) CL2009000036A1 (en)
CO (1) CO6321187A2 (en)
DK (1) DK2231614T3 (en)
EA (1) EA201001124A1 (en)
EC (1) ECSP10010334A (en)
ES (1) ES2380186T3 (en)
GB (1) GB0800407D0 (en)
GT (1) GT200900003A (en)
IL (1) IL206360A (en)
PH (1) PH12012501905A1 (en)
PL (1) PL2231614T3 (en)
PT (1) PT2231614E (en)
SV (1) SV2010003617A (en)
TW (1) TW200930294A (en)
WO (1) WO2009087098A2 (en)
ZA (1) ZA201004305B (en)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2343280A1 (en) * 2009-12-10 2011-07-13 Bayer CropScience AG Fungicide quinoline derivatives
WO2011144444A1 (en) * 2010-05-21 2011-11-24 Syngenta Participations Ag Novel amides as fungicides
EP2397467A1 (en) * 2010-06-10 2011-12-21 Syngenta Participations AG Quinoline derivatives as fungicides
TWI504350B (en) 2010-09-01 2015-10-21 Du Pont Fungicidal pyrazoles and their mixtures
TWI568721B (en) 2012-02-01 2017-02-01 杜邦股份有限公司 Fungicidal pyrazole mixtures
WO2013126283A1 (en) 2012-02-20 2013-08-29 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
WO2013156324A1 (en) * 2012-04-16 2013-10-24 Syngenta Participations Ag Use of compounds for the control of cereal diseases
JP6185056B2 (en) 2012-06-22 2017-08-23 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニーE.I.Du Pont De Nemours And Company Bactericidal and fungicidal 4-methylanilinopyrazole
WO2014044642A1 (en) * 2012-09-20 2014-03-27 Syngenta Participations Ag N-cyclopropylmethyl-2-(quinolin-6-yloxy)-acetamide derivatives and their use as fungicides
WO2014060177A1 (en) * 2012-10-16 2014-04-24 Syngenta Participations Ag Fungicidal compositions
WO2014130409A2 (en) 2013-02-21 2014-08-28 E. I. Du Pont De Nemours And Company Fungicidal pyrazole mixtures
WO2014172190A1 (en) 2013-04-15 2014-10-23 E. I. Du Pont De Nemours And Company Fungicidal amides
PL2986601T3 (en) 2013-04-15 2017-10-31 Fmc Corp Fungicidal carboxamides
WO2015123193A1 (en) 2014-02-12 2015-08-20 E. I. Du Pont De Nemours And Company Fungicidal benzodipyrazoles
WO2015157005A1 (en) 2014-04-10 2015-10-15 E I Du Pont De Nemours And Company Substituted tolyl fungicide mixtures
US20170037014A1 (en) 2014-05-06 2017-02-09 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
EP3271336A1 (en) 2015-03-19 2018-01-24 E. I. du Pont de Nemours and Company Fungicidal pyrazoles
PL3558984T3 (en) 2016-12-20 2024-01-15 Fmc Corporation Fungicidal oxadiazoles
TWI772367B (en) * 2017-02-16 2022-08-01 瑞士商先正達合夥公司 Fungicidal compositions
TW202334101A (en) 2017-04-06 2023-09-01 美商富曼西公司 Fungicidal oxadiazoles
AR112221A1 (en) 2017-07-05 2019-10-02 Fmc Corp FUNGICIDE OXADIAZOLES, COMPOSITION THAT INCLUDE THEM AND A METHOD TO CONTROL PHYTO DISEASES THAT USE THEM
TW202400547A (en) 2018-09-06 2024-01-01 美商富曼西公司 Fungicidal nitroanilino substituted pyrazoles
JP2022500434A (en) 2018-09-14 2022-01-04 エフ エム シー コーポレーションFmc Corporation Fungal killing halomethyl ketones and hydrates
TWI832917B (en) 2018-11-06 2024-02-21 美商富曼西公司 Substituted tolyl fungicides
EP4090651A1 (en) 2020-01-15 2022-11-23 Fmc Corporation Fungicidal amides
MX2022009926A (en) 2020-02-14 2022-09-09 Fmc Corp Substituted 5,6-diphenyl-3(2h)-pyridazinones for use as fungicides.
WO2022128746A1 (en) 2020-12-14 2022-06-23 Elanco Tiergesundheit Ag Quinoline derivatives as endoparasiticides

Family Cites Families (8)

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Publication number Priority date Publication date Assignee Title
AU1685999A (en) 1997-12-24 1999-07-19 Ihara Chemical Industry Co. Ltd. Pyridyloxy(thio)alkanoic acid amide derivatives and agricultural/horticultural bactericides
JP2001089453A (en) * 1999-09-21 2001-04-03 Kumiai Chem Ind Co Ltd Heteroaryloxy(thio)alkanoic acid amide derivative and germicide for agriculture and horticulture
GB0129267D0 (en) * 2001-12-06 2002-01-23 Syngenta Ltd Fungicides
GB0227555D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0312863D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0426373D0 (en) * 2004-12-01 2005-01-05 Syngenta Ltd Fungicides
GB0704906D0 (en) * 2007-03-14 2007-04-25 Syngenta Participations Ag Fungicides
GB0717256D0 (en) * 2007-09-05 2007-10-17 Syngenta Participations Ag Novel fungicides

Also Published As

Publication number Publication date
US8415272B2 (en) 2013-04-09
CN103183637A (en) 2013-07-03
PH12012501905A1 (en) 2015-10-19
EA201001124A1 (en) 2011-02-28
CN101910135B (en) 2013-03-13
AU2009203826B2 (en) 2013-08-22
WO2009087098A2 (en) 2009-07-16
GB0800407D0 (en) 2008-02-20
CN101910135A (en) 2010-12-08
TW200930294A (en) 2009-07-16
IL206360A (en) 2013-08-29
ZA201004305B (en) 2011-11-30
AU2009203826A1 (en) 2009-07-16
CA2711094A1 (en) 2009-07-16
WO2009087098A8 (en) 2009-11-26
WO2009087098A3 (en) 2009-10-01
EP2231614A2 (en) 2010-09-29
ES2380186T3 (en) 2012-05-09
US20100280068A1 (en) 2010-11-04
GT200900003A (en) 2009-11-24
ECSP10010334A (en) 2010-08-31
DK2231614T3 (en) 2012-04-23
PL2231614T3 (en) 2012-09-28
ATE546433T1 (en) 2012-03-15
CL2009000036A1 (en) 2009-06-05
PT2231614E (en) 2012-04-03
AR070135A1 (en) 2010-03-17
SV2010003617A (en) 2011-03-23
EP2231614B1 (en) 2012-02-22
IL206360A0 (en) 2010-12-30
BRPI0907184A2 (en) 2019-09-24
JP2011509271A (en) 2011-03-24
KR20100109952A (en) 2010-10-11

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