CO4480099A1 - A PRE-CONCENTRATE OF MICROEMULSION THAT INCLUDES A HARDLY SOLUBLE ACTIVE AGENT AND A CARRIING MEDIA - Google Patents
A PRE-CONCENTRATE OF MICROEMULSION THAT INCLUDES A HARDLY SOLUBLE ACTIVE AGENT AND A CARRIING MEDIAInfo
- Publication number
- CO4480099A1 CO4480099A1 CO95050316A CO95050316A CO4480099A1 CO 4480099 A1 CO4480099 A1 CO 4480099A1 CO 95050316 A CO95050316 A CO 95050316A CO 95050316 A CO95050316 A CO 95050316A CO 4480099 A1 CO4480099 A1 CO 4480099A1
- Authority
- CO
- Colombia
- Prior art keywords
- active agent
- composition
- carriing
- microemulsion
- concentrate
- Prior art date
Links
Abstract
1. UN PRE-CONCENTRADO DE MICROEMULSION QUE COM- PRENDE UN AGENTE ACTIVO DIFICILMENTE SOLUBLE, Y UN MEDIO PORTADOR, QUE COMPRENDE 1) UNA FASE HIDROFILICA LA CUAL COMPRENDE DIMETIL- ISOSORBIDE Y/O ESTER ALCANOICO DE ALQUILO INFE- RIOR,A FSE LIPOFILICA; Y 2) UNA FASE LIPOFILICA; Y 3) UN TENSOACTIVO. 2. UNA COMPOSICION DE LA REIVINDICACION 1, EN LA QUE EL AGENTE ACTIVO ES UNA CICLOSPORINA O UN MA- CROLIDO. 4. UNA COMPOSICION COMO SE REIVINDICA EN CUAL- QUIER REIVINDICACION PRECEDENTE. EN LA QUE LA FASE HIDROFILICA COMPRENDE ACETATO DE ETILO COMO EL ESTER ALCANOICO DE ALQUILO INFERIOR. 5. UNA COMPOSICION COMO SE REIVINDICA EN UNA DE LAS REIVINDICACIONES 1 A 4, PARA ADMINISTRACIN O- RAL O PARENTERAL. 6. UNA COMPOSICION FARMACEUTICA PARA ADMINISTRA- CION ENTERAL O PARENTERAL, QUE COMPRENDE UN MACRO- LIDO Y UN ACIDO. 7. UNA COMPOSICION COMO SE REIVINDICA EN LA REI- VINDICACION 6, EN LA QUE EL ACIDO ES UN ACIDO MO- NO-, DI-, O TRI-CARBOXILICO. FIGURA 11. A PRE-CONCENTRATE OF MICROEMULSION THAT INCLUDES A DIFFICULT SOLUBLE ACTIVE AGENT, AND A CARRIING MEDIUM, WHICH INCLUDES 1) A HYDROPHILIC PHASE WHICH INCLUDES DIMETHYL-ISOSORBIDE AND / OR ALCANOIC STERILE OF ALKYL INFORIORAL, FS ; AND 2) A LIPOPHILIC PHASE; AND 3) A TENSOACTIVE. 2. A COMPOSITION OF CLAIM 1, IN WHICH THE ACTIVE AGENT IS A CYCLOSPORINE OR A MOLECOLID. 4. A COMPOSITION AS CLAIMED IN ANY PRECEDING CLAIM. IN WHICH THE HYDROPHILIC PHASE INCLUDES ETHYL ACETATE AS THE LOWER ALKYL ALCANOIC ESTER. 5. A COMPOSITION AS CLAIMED IN ONE OF CLAIMS 1 TO 4, FOR ORAL OR PARENTERAL ADMINISTRATION. 6. A PHARMACEUTICAL COMPOSITION FOR ENTERAL OR PARENTERAL ADMINISTRATION, WHICH INCLUDES A MACROLID AND AN ACID. 7. A COMPOSITION AS CLAIMED IN CLAIM 6, IN WHICH THE ACID IS A MONO-, DI-, OR TRI-CARBOXYLIC ACID. FIGURE 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9421613A GB9421613D0 (en) | 1994-10-26 | 1994-10-26 | Organic compounds |
GB9422084A GB9422084D0 (en) | 1994-11-02 | 1994-11-02 | Organic compounds |
GBGB9517133.6A GB9517133D0 (en) | 1995-08-22 | 1995-08-22 | Pharmaceutical compositions |
Publications (1)
Publication Number | Publication Date |
---|---|
CO4480099A1 true CO4480099A1 (en) | 1997-07-09 |
Family
ID=40929712
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO95050316A CO4480099A1 (en) | 1994-10-26 | 1995-10-25 | A PRE-CONCENTRATE OF MICROEMULSION THAT INCLUDES A HARDLY SOLUBLE ACTIVE AGENT AND A CARRIING MEDIA |
Country Status (1)
Country | Link |
---|---|
CO (1) | CO4480099A1 (en) |
-
1995
- 1995-10-25 CO CO95050316A patent/CO4480099A1/en unknown
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