CO4370014A1 - Soluciones inyectables estables de diritromicina - Google Patents

Soluciones inyectables estables de diritromicina

Info

Publication number
CO4370014A1
CO4370014A1 CO95011794A CO95011794A CO4370014A1 CO 4370014 A1 CO4370014 A1 CO 4370014A1 CO 95011794 A CO95011794 A CO 95011794A CO 95011794 A CO95011794 A CO 95011794A CO 4370014 A1 CO4370014 A1 CO 4370014A1
Authority
CO
Colombia
Prior art keywords
lipophyl
directromycin
stable
injectable solutions
injectable solution
Prior art date
Application number
CO95011794A
Other languages
English (en)
Inventor
Stefan Leiner
Bernhard Hassel
Original Assignee
Boehringer Ingelheim Vetmed
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Vetmed filed Critical Boehringer Ingelheim Vetmed
Publication of CO4370014A1 publication Critical patent/CO4370014A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

1. SOLUCION INYECTABLE QUE CONTIENE DIRITROMICINA COMO SUSTANCIA ACTIVA EN UNA MEZCLA DE DISOLVENTES FARMACOLOGICAMENTE COMPATIBLE, UNIFASICA, QUE CONTIENE AGUA Y LIPOFILA. 2. SOLUCION INYECTABLE SEGUN LA REIVINDICACION 1, CARACTERIZADA PORQUE LA MEZCLA DE DISOLVENTES LIPOFILA CONSTA DE UN COMPONENTE LIPOFILO Y UN DISOLVENTE ORGANICO ANFIFILO O HIDROFILO. 6. SOLUCION INYECTABLE SEGUN UNA DE LAS PRECEDEN- TES REIVINDICACIONES, CARACTERIZADA PORQUE CONTIE- NE MIRISTATO DE ISOPROPILO COMO COMPONENTE LIPO- FILO Y ETANOL COMO DISOLVENTE HIDROFILO.
CO95011794A 1994-03-26 1995-03-23 Soluciones inyectables estables de diritromicina CO4370014A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4410637A DE4410637C1 (de) 1994-03-26 1994-03-26 Injizierbare Lösungen von Dirithromycin

Publications (1)

Publication Number Publication Date
CO4370014A1 true CO4370014A1 (es) 1996-10-07

Family

ID=6514000

Family Applications (1)

Application Number Title Priority Date Filing Date
CO95011794A CO4370014A1 (es) 1994-03-26 1995-03-23 Soluciones inyectables estables de diritromicina

Country Status (7)

Country Link
EP (1) EP0754047A1 (es)
JP (1) JPH09510722A (es)
AU (1) AU2214195A (es)
CO (1) CO4370014A1 (es)
DE (1) DE4410637C1 (es)
WO (1) WO1995026191A1 (es)
ZA (1) ZA952405B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19518917A1 (de) * 1995-05-23 1996-11-28 Boehringer Ingelheim Vetmed Stabile, konzentrierte lokalverträgliche Erythromycylamin-Lösungen
DE19701949A1 (de) * 1997-01-13 1998-07-16 Jenapharm Gmbh Transdermales therapeutisches System
KR101805087B1 (ko) * 2010-09-16 2017-12-05 주식회사 엘지화학 높은 방부력을 제공하는 오일 주사 제형

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
US4918108A (en) * 1982-03-16 1990-04-17 Boehringer Ingelheim Vetmedica Gmbh Method of improving the absorption of injected antibacterial substances
DE3209429A1 (de) * 1982-03-16 1983-10-06 Boehringer Ingelheim Vetmed Mittel zur verbesserung der resorption von injizierten antibakteriell wirksamen substanzen und kombinationen, enthaltend ein benzyaminderivat
AU630469B2 (en) * 1989-05-26 1992-10-29 Abbott Laboratories Injectable clarithromycin composition

Also Published As

Publication number Publication date
JPH09510722A (ja) 1997-10-28
EP0754047A1 (de) 1997-01-22
DE4410637C1 (de) 1995-09-21
WO1995026191A1 (de) 1995-10-05
ZA952405B (en) 1995-09-26
AU2214195A (en) 1995-10-17

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