CN1297439A - 4-(氨基)-(乙氨基)-羟吲哚多巴胺自身受体激动剂 - Google Patents
4-(氨基)-(乙氨基)-羟吲哚多巴胺自身受体激动剂 Download PDFInfo
- Publication number
- CN1297439A CN1297439A CN99805030A CN99805030A CN1297439A CN 1297439 A CN1297439 A CN 1297439A CN 99805030 A CN99805030 A CN 99805030A CN 99805030 A CN99805030 A CN 99805030A CN 1297439 A CN1297439 A CN 1297439A
- Authority
- CN
- China
- Prior art keywords
- alkyl
- hydrogen
- compound
- formula
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5883498A | 1998-04-13 | 1998-04-13 | |
US09/058,834 | 1998-04-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
CN1297439A true CN1297439A (zh) | 2001-05-30 |
Family
ID=22019205
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN99805030A Pending CN1297439A (zh) | 1998-04-13 | 1999-04-12 | 4-(氨基)-(乙氨基)-羟吲哚多巴胺自身受体激动剂 |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1073636A1 (es) |
JP (1) | JP2002511450A (es) |
CN (1) | CN1297439A (es) |
AR (1) | AR014847A1 (es) |
AU (1) | AU3555099A (es) |
CA (1) | CA2327477A1 (es) |
WO (1) | WO1999052870A1 (es) |
ZA (1) | ZA992670B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR032641A1 (es) * | 2001-01-29 | 2003-11-19 | Otsuka Pharma Co Ltd | Agonista de subtipo de receptor 5-ht 1a. |
US7053092B2 (en) | 2001-01-29 | 2006-05-30 | Otsuka Pharmaceutical Co., Ltd. | 5-HT1a receptor subtype agonist |
US8703772B2 (en) | 2001-09-25 | 2014-04-22 | Otsuka Pharmaceutical Co., Ltd. | Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
AR033485A1 (es) | 2001-09-25 | 2003-12-26 | Otsuka Pharma Co Ltd | Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4452808A (en) * | 1982-12-07 | 1984-06-05 | Smithkline Beckman Corporation | 4-Aminoalkyl-2(3H)-indolones |
GB8712073D0 (en) * | 1987-05-21 | 1987-06-24 | Smith Kline French Lab | Medicament |
AU4312593A (en) * | 1992-05-18 | 1993-12-13 | Smithkline Beecham Plc | Use of indolone derivatives for the treatment of memory disorders, sexual dysfunction and Parkinson's disease |
AU4088897A (en) * | 1996-08-27 | 1998-03-19 | American Home Products Corporation | 4-aminoethoxy indolone derivatives |
-
1999
- 1999-04-12 CA CA002327477A patent/CA2327477A1/en not_active Abandoned
- 1999-04-12 JP JP2000543433A patent/JP2002511450A/ja active Pending
- 1999-04-12 CN CN99805030A patent/CN1297439A/zh active Pending
- 1999-04-12 WO PCT/US1999/007967 patent/WO1999052870A1/en not_active Application Discontinuation
- 1999-04-12 ZA ZA9902670A patent/ZA992670B/xx unknown
- 1999-04-12 EP EP99917423A patent/EP1073636A1/en not_active Withdrawn
- 1999-04-12 AU AU35550/99A patent/AU3555099A/en not_active Abandoned
- 1999-04-12 AR ARP990101678A patent/AR014847A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
ZA992670B (en) | 2000-10-12 |
EP1073636A1 (en) | 2001-02-07 |
AU3555099A (en) | 1999-11-01 |
WO1999052870A1 (en) | 1999-10-21 |
JP2002511450A (ja) | 2002-04-16 |
CA2327477A1 (en) | 1999-10-21 |
AR014847A1 (es) | 2001-03-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
WD01 | Invention patent application deemed withdrawn after publication |