CL2022000790A1 - Método para tratar vih con cabotegravir y rilpivirina - Google Patents

Método para tratar vih con cabotegravir y rilpivirina

Info

Publication number
CL2022000790A1
CL2022000790A1 CL2022000790A CL2022000790A CL2022000790A1 CL 2022000790 A1 CL2022000790 A1 CL 2022000790A1 CL 2022000790 A CL2022000790 A CL 2022000790A CL 2022000790 A CL2022000790 A CL 2022000790A CL 2022000790 A1 CL2022000790 A1 CL 2022000790A1
Authority
CL
Chile
Prior art keywords
cabotegravir
rilpivirine
treat hiv
human
pharmaceutically acceptable
Prior art date
Application number
CL2022000790A
Other languages
English (en)
Inventor
Herta Maria Ludovica Crauwels
Susan L Ford
David Andrew Margolis
Stefaan Louis F Rossenu
William Robert Spreen
Solingen-Ristea Rodica Mihaela Van
Peter Evan Owen Williams
Original Assignee
Viiv Healthcare Co
Janssen Sciences Ireland Unlimited Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Viiv Healthcare Co, Janssen Sciences Ireland Unlimited Co filed Critical Viiv Healthcare Co
Publication of CL2022000790A1 publication Critical patent/CL2022000790A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Abstract

La invención consiste en métodos para tratar VIH en un humano que los necesita, los cuales comprenden la administración de una cantidad terapéuticamente eficaz de una combinación de cabotegravir o una sal farmacéuticamente aceptable del mismo y rilpivirina o una sal farmacéuticamente aceptable de la misma, a dicho humano.
CL2022000790A 2019-10-01 2022-03-30 Método para tratar vih con cabotegravir y rilpivirina CL2022000790A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201962908882P 2019-10-01 2019-10-01
US201962908995P 2019-10-01 2019-10-01
US202063037782P 2020-06-11 2020-06-11
US202063052214P 2020-07-15 2020-07-15

Publications (1)

Publication Number Publication Date
CL2022000790A1 true CL2022000790A1 (es) 2022-11-25

Family

ID=72826936

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2022000790A CL2022000790A1 (es) 2019-10-01 2022-03-30 Método para tratar vih con cabotegravir y rilpivirina

Country Status (11)

Country Link
US (1) US20220347174A1 (es)
EP (1) EP4037661A1 (es)
JP (1) JP2022550828A (es)
KR (1) KR20220074880A (es)
CN (1) CN114502166A (es)
AU (1) AU2020358156A1 (es)
CA (1) CA3155587A1 (es)
CL (1) CL2022000790A1 (es)
IL (1) IL290716A (es)
MX (1) MX2022003945A (es)
WO (1) WO2021064618A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023222755A1 (en) * 2022-05-17 2023-11-23 Janssen Sciences Ireland Unlimited Company Treatment or prevention of hiv infection
WO2023222754A1 (en) * 2022-05-17 2023-11-23 Janssen Sciences Ireland Unlimited Company Rilpivirine for use in the treatment or prevention of hiv infection

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010299959B2 (en) * 2009-09-22 2016-07-21 Tibotec Pharmaceuticals Treatment and prevention of HIV infection
JP7384783B2 (ja) * 2017-07-21 2023-11-21 ヴィーブ ヘルスケア カンパニー Hiv感染症及びaidsを治療するためのレジメン
CN109568328A (zh) * 2017-09-29 2019-04-05 重庆药友制药有限责任公司 一种用于预防和治疗hiv感染的药物组合物

Also Published As

Publication number Publication date
MX2022003945A (es) 2022-04-25
US20220347174A1 (en) 2022-11-03
CN114502166A (zh) 2022-05-13
CA3155587A1 (en) 2021-04-08
EP4037661A1 (en) 2022-08-10
JP2022550828A (ja) 2022-12-05
KR20220074880A (ko) 2022-06-03
IL290716A (en) 2022-04-01
AU2020358156A1 (en) 2022-04-21
WO2021064618A1 (en) 2021-04-08

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