CH484161A - Verfahren zur Herstellung von Pyrazinoylguanidinen und Pyrazinamidoguanidinen - Google Patents

Verfahren zur Herstellung von Pyrazinoylguanidinen und Pyrazinamidoguanidinen

Info

Publication number
CH484161A
CH484161A CH803667A CH803667A CH484161A CH 484161 A CH484161 A CH 484161A CH 803667 A CH803667 A CH 803667A CH 803667 A CH803667 A CH 803667A CH 484161 A CH484161 A CH 484161A
Authority
CH
Switzerland
Prior art keywords
pyrazinamidoguanidines
pyrazinoylguanidines
preparation
Prior art date
Application number
CH803667A
Other languages
English (en)
Inventor
Immanuel Pollak Peter
James Tull Roger
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CH484161A publication Critical patent/CH484161A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CH803667A 1966-08-25 1967-06-07 Verfahren zur Herstellung von Pyrazinoylguanidinen und Pyrazinamidoguanidinen CH484161A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57490966A 1966-08-25 1966-08-25

Publications (1)

Publication Number Publication Date
CH484161A true CH484161A (de) 1970-01-15

Family

ID=24298146

Family Applications (1)

Application Number Title Priority Date Filing Date
CH803667A CH484161A (de) 1966-08-25 1967-06-07 Verfahren zur Herstellung von Pyrazinoylguanidinen und Pyrazinamidoguanidinen

Country Status (7)

Country Link
US (1) US3432502A (de)
BE (1) BE699435A (de)
CH (1) CH484161A (de)
DK (1) DK115771B (de)
ES (1) ES341321A1 (de)
GB (1) GB1184709A (de)
NL (1) NL6707563A (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3506662A (en) * 1968-04-30 1970-04-14 Merck & Co Inc Process for preparation of pyrazinoyland pyrazinamidoguanidines
US4224447A (en) * 1979-03-27 1980-09-23 Merck & Co., Inc. Novel pyrazinecarboxamides and processes for preparing same
US4246406A (en) * 1979-03-27 1981-01-20 Merck & Co., Inc. Heterocyclic substituted pyrazinoylguanidines
TWI439462B (zh) 2007-12-10 2014-06-01 Novartis Ag 作為enac阻抑劑之螺環胍化合物

Also Published As

Publication number Publication date
NL6707563A (de) 1968-02-26
GB1184709A (en) 1970-03-18
BE699435A (de) 1967-12-04
ES341321A1 (es) 1968-10-16
US3432502A (en) 1969-03-11
DK115771B (da) 1969-11-10

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Legal Events

Date Code Title Description
PL Patent ceased