CA2616915A1 - Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire - Google Patents

Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire Download PDF

Info

Publication number: CA2616915A1
Authority: CA; Canada
Prior art keywords: depigmenting; adapalene; agent; skin; composition
Prior art date: 2005-09-02
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002616915A

Other languages

English (en)

Inventor

Isabelle Pelisson

Andre Jomard

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Galderma Research and Development SNC

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-09-02

Filing date

2006-08-31

Publication date

2007-05-10

2005-09-02 Priority claimed from FR0509003A external-priority patent/FR2890314B1/fr

2006-08-31 Application filed by Individual filed Critical Individual

2007-05-10 Publication of CA2616915A1 publication Critical patent/CA2616915A1/fr

Status Abandoned legal-status Critical Current

Links

229960002916 adapalene Drugs 0.000 title claims abstract description 43
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239000000203 mixture Substances 0.000 title claims abstract description 43
239000007854 depigmenting agent Substances 0.000 title claims abstract description 21
229940121363 anti-inflammatory agent Drugs 0.000 title claims abstract description 13
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239000002537 cosmetic Substances 0.000 claims abstract description 7
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229940100460 peg-100 stearate Drugs 0.000 description 2
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WZNJWVWKTVETCG-UHFFFAOYSA-N kojic acid Natural products OC(=O)C(N)CN1C=CC(=O)C(O)=C1 WZNJWVWKTVETCG-UHFFFAOYSA-N 0.000 description 1
FAARLWTXUUQFSN-UHFFFAOYSA-N methylellagic acid Natural products O1C(=O)C2=CC(O)=C(O)C3=C2C2=C1C(OC)=C(O)C=C2C(=O)O3 FAARLWTXUUQFSN-UHFFFAOYSA-N 0.000 description 1
229960004584 methylprednisolone Drugs 0.000 description 1
229960002509 miconazole Drugs 0.000 description 1
239000002480 mineral oil Substances 0.000 description 1
235000010446 mineral oil Nutrition 0.000 description 1
230000001333 moisturizer Effects 0.000 description 1
VYQNWZOUAUKGHI-UHFFFAOYSA-N monobenzone Chemical compound C1=CC(O)=CC=C1OCC1=CC=CC=C1 VYQNWZOUAUKGHI-UHFFFAOYSA-N 0.000 description 1
229960000990 monobenzone Drugs 0.000 description 1
210000004400 mucous membrane Anatomy 0.000 description 1
230000037311 normal skin Effects 0.000 description 1
150000007530 organic bases Chemical class 0.000 description 1
229960005323 phenoxyethanol Drugs 0.000 description 1
WVDDGKGOMKODPV-ZQBYOMGUSA-N phenyl(114C)methanol Chemical compound O[14CH2]C1=CC=CC=C1 WVDDGKGOMKODPV-ZQBYOMGUSA-N 0.000 description 1
229960005205 prednisolone Drugs 0.000 description 1
OIGNJSKKLXVSLS-VWUMJDOOSA-N prednisolone Chemical compound O=C1C=C[C@]2(C)[C@H]3[C@@H](O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 OIGNJSKKLXVSLS-VWUMJDOOSA-N 0.000 description 1
229960004618 prednisone Drugs 0.000 description 1
XOFYZVNMUHMLCC-ZPOLXVRWSA-N prednisone Chemical compound O=C1C=C[C@]2(C)[C@H]3C(=O)C[C@](C)([C@@](CC4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 XOFYZVNMUHMLCC-ZPOLXVRWSA-N 0.000 description 1
239000003223 protective agent Substances 0.000 description 1
150000003217 pyrazoles Chemical class 0.000 description 1
230000004044 response Effects 0.000 description 1
150000003839 salts Chemical class 0.000 description 1
235000010265 sodium sulphite Nutrition 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
150000003408 sphingolipids Chemical class 0.000 description 1
229940098760 steareth-2 Drugs 0.000 description 1
229940100458 steareth-21 Drugs 0.000 description 1
230000003637 steroidlike Effects 0.000 description 1
230000000475 sunscreen effect Effects 0.000 description 1
239000000516 sunscreening agent Substances 0.000 description 1
239000011975 tartaric acid Substances 0.000 description 1
235000002906 tartaric acid Nutrition 0.000 description 1
230000000699 topical effect Effects 0.000 description 1
229960002117 triamcinolone acetonide Drugs 0.000 description 1
YNDXUCZADRHECN-JNQJZLCISA-N triamcinolone acetonide Chemical compound C1CC2=CC(=O)C=C[C@]2(C)[C@]2(F)[C@@H]1[C@@H]1C[C@H]3OC(C)(C)O[C@@]3(C(=O)CO)[C@@]1(C)C[C@@H]2O YNDXUCZADRHECN-JNQJZLCISA-N 0.000 description 1
229930003231 vitamin Natural products 0.000 description 1
239000011782 vitamin Substances 0.000 description 1
229940088594 vitamin Drugs 0.000 description 1
235000013343 vitamin Nutrition 0.000 description 1
239000000341 volatile oil Substances 0.000 description 1
229940105296 zinc peroxide Drugs 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/02—Preparations for care of the skin for chemically bleaching or whitening the skin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/34—Alcohols
- A61K8/347—Phenols
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/36—Carboxylic acids; Salts or anhydrides thereof
- A61K8/368—Carboxylic acids; Salts or anhydrides thereof with carboxyl groups directly bound to carbon atoms of aromatic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/63—Steroids; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Chemical & Material Sciences (AREA)
Birds (AREA)
Emergency Medicine (AREA)
Dermatology (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

CA002616915A 2005-09-02 2006-08-31 Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire Abandoned CA2616915A1 (fr)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
FR0509003		2005-09-02
FR0509003A FR2890314B1 (fr)	2005-09-02	2005-09-02	Compositiondepigmentante de la peau comprenant de l'adapalene au moins un agent depigmentant et au moins un agent anti-inflammatoire
US71776705P	2005-09-19	2005-09-19
US60/717,767		2005-09-19
PCT/IB2006/003725 WO2007052157A2 (fr)	2005-09-02	2006-08-31	Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire

Publications (1)

Publication Number	Publication Date
CA2616915A1 true CA2616915A1 (fr)	2007-05-10

Family

ID=38006259

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002616915A Abandoned CA2616915A1 (fr)	2005-09-02	2006-08-31	Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire

Country Status (3)

Country	Link
EP (1)	EP1926484A2 (fr)
CA (1)	CA2616915A1 (fr)
WO (1)	WO2007052157A2 (fr)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3856934A (en) *	1970-06-24	1974-12-24	A Kligman	Skin depigmentation
US6358541B1 (en) *	2000-05-03	2002-03-19	David S. Goodman	Topical preparation for the treatment of hair loss
FR2833841B1 (fr) *	2001-12-21	2005-07-22	Galderma Res & Dev	Gel comprenant au moins un retinoide et du peroxyde de benzoyle
ES2289315T3 (es) *	2002-09-05	2008-02-01	GALDERMA RESEARCH & DEVELOPMENT	Composicion despigmentante para la piel que contiene adapaleno y al menos un agente despigmentante.

2006
- 2006-08-31 CA CA002616915A patent/CA2616915A1/fr not_active Abandoned
- 2006-08-31 EP EP06842260A patent/EP1926484A2/fr not_active Withdrawn
- 2006-08-31 WO PCT/IB2006/003725 patent/WO2007052157A2/fr active Application Filing

Also Published As

Publication number	Publication date
WO2007052157A2 (fr)	2007-05-10
WO2007052157A3 (fr)	2007-10-04
EP1926484A2 (fr)	2008-06-04

Legal Events

Date	Code	Title	Description
2011-08-30	EEER	Examination request
2014-06-24	FZDE	Dead	Effective date: 20140429

Publication	Publication Date	Title
US20050163731A1 (en)	2005-07-28	Skin depigmenting compositions comprising adapalene and at least one depigmenting active agent
JP3500154B2 (ja)	2004-02-23	皮膚美白組成物
JPH07501541A (ja)	1995-02-16	皮膚シワ及び／又は皮膚萎縮を調節するためのサリチル酸の用法
US20060029556A1 (en)	2006-02-09	Aqueous-alcoholic depigmenting gels
Dessinioti et al.	2017	Melasma
MX2010012753A (es)	2010-12-21	Composiciones despigmentantes anhidras que comprenden, dentro de la fase grasa, un derivado fenolico solubilizado y un retinoide.
US20100124538A1 (en)	2010-05-20	Topical application of fluocinolone acetonide for depigmentation of the skin
US20080219936A1 (en)	2008-09-11	Skin depigmenting compositions comprising adapalene, at least one depigmenting agent and at least one anti-inflammatory agent
CA2022917C (fr)	1995-04-18	Compose synergique pour la depigmentation de la peau
CA2616915A1 (fr)	2007-05-10	Composition de depigmentation destinee a la peau et comprenant de l'adapalene, au moins un agent de depigmentation et au moins un agent anti-inflammatoire
US20080305060A1 (en)	2008-12-11	Aqueous-alcoholic depigmenting gels
Mashhood	2006	Treatment of hyperpigmentation disorders
EP1477157B1 (fr)	2008-03-19	Compositions conprenant une amidine et un alkane polyol
Westerhof et al.	1999	Bleaching agents
EP1813312A2 (fr)	2007-08-01	Composition de dépigmentation pour la peau comportant de l'adapalène et au moins un agent de dépigmentation
US20140005276A1 (en)	2014-01-02	Compositions comprising substituted phenols and topical application thereof
JP2009519304A (ja)	2009-05-14	乾癬または湿疹に引き続く皮膚の過剰色素沈着を処理するための、ヒドロキノン、フルオシノロンアセトニド、及びトレチノインの組み合わせを含む皮膚科学用組成物の使用
ZA200504037B (en)	2006-04-26	Aqueous-alchoholic depigmenting gel
JP2003292413A (ja)	2003-10-15	皮膚外用剤
Selleri	0	Managing Hyperpigmentation
OA12083A (en)	2006-05-04	A method of treating and lightening hyperpigmentation in black skin with a retinoid.