BRPI0917519A2 - Processo para preparacao de um polimorfo de 7-cloro-n,n,5-trimetil-4-oxo-3-fenil-3,5-di-hidro-4h-pir idazino[4,5-b]indol-1-acetamida - Google Patents

Processo para preparacao de um polimorfo de 7-cloro-n,n,5-trimetil-4-oxo-3-fenil-3,5-di-hidro-4h-pir idazino[4,5-b]indol-1-acetamida

Info

Publication number
BRPI0917519A2
BRPI0917519A2 BRPI0917519-9A BRPI0917519A BRPI0917519A2 BR PI0917519 A2 BRPI0917519 A2 BR PI0917519A2 BR PI0917519 A BRPI0917519 A BR PI0917519A BR PI0917519 A2 BRPI0917519 A2 BR PI0917519A2
Authority
BR
Brazil
Prior art keywords
polymorph
indol
pyridazine
acetamide
dihydro
Prior art date
Application number
BRPI0917519-9A
Other languages
English (en)
Inventor
William L Rocco
Original Assignee
Sanofi Aventis Us Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis Us Llc filed Critical Sanofi Aventis Us Llc
Publication of BRPI0917519A2 publication Critical patent/BRPI0917519A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
BRPI0917519-9A 2008-08-18 2009-08-13 Processo para preparacao de um polimorfo de 7-cloro-n,n,5-trimetil-4-oxo-3-fenil-3,5-di-hidro-4h-pir idazino[4,5-b]indol-1-acetamida BRPI0917519A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8964808P 2008-08-18 2008-08-18
PCT/US2009/053698 WO2010021905A1 (en) 2008-08-18 2009-08-13 Process for preparing polymorph of 7-chloro-n, n,5-trimethyl-4-oxo-3-phenyl-3,5-dihydr0-4h-pyridazin0[4,5-b]indole-1-acetamide

Publications (1)

Publication Number Publication Date
BRPI0917519A2 true BRPI0917519A2 (pt) 2015-08-04

Family

ID=41131790

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0917519-9A BRPI0917519A2 (pt) 2008-08-18 2009-08-13 Processo para preparacao de um polimorfo de 7-cloro-n,n,5-trimetil-4-oxo-3-fenil-3,5-di-hidro-4h-pir idazino[4,5-b]indol-1-acetamida

Country Status (12)

Country Link
US (1) US20110224214A1 (pt)
EP (1) EP2364315A1 (pt)
JP (1) JP2012500268A (pt)
KR (1) KR20110052640A (pt)
CN (1) CN102186854A (pt)
AU (1) AU2009283039A1 (pt)
BR (1) BRPI0917519A2 (pt)
CA (1) CA2734448A1 (pt)
IL (1) IL211221A0 (pt)
MX (1) MX2011001474A (pt)
RU (1) RU2011110241A (pt)
WO (1) WO2010021905A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7303772B2 (en) 2005-11-10 2007-12-04 Olalde Rangel Jose Angel Synergistic phytoceutical compositions

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2766823B1 (fr) * 1997-07-30 1999-10-08 Synthelabo Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique
FR2788696B1 (fr) * 1999-01-26 2004-03-05 Synthelabo Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central
WO2007027525A1 (en) * 2005-08-29 2007-03-08 Sanofi-Aventis U.S. Llc Novel crystalline form of a pyridazino [4 , 5-b] indole derivative
SI1926476T1 (sl) * 2005-08-29 2013-07-31 Sanofi-Aventis U.S. Llc Amorfne trdne disperzije 7-kloro-N,N,5-trimetil-4-okso-3-fenil-3,5- dihidro-4H-piridazino/4,5-b/indol-1-acetamida

Also Published As

Publication number Publication date
CA2734448A1 (en) 2010-02-25
CN102186854A (zh) 2011-09-14
EP2364315A1 (en) 2011-09-14
IL211221A0 (en) 2011-04-28
MX2011001474A (es) 2011-03-25
WO2010021905A1 (en) 2010-02-25
RU2011110241A (ru) 2012-09-27
AU2009283039A1 (en) 2010-02-25
JP2012500268A (ja) 2012-01-05
US20110224214A1 (en) 2011-09-15
KR20110052640A (ko) 2011-05-18

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 4A, 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.