BRPI0912512A2 - Processo para a preparação de compostos - Google Patents

Processo para a preparação de compostos

Info

Publication number
BRPI0912512A2
BRPI0912512A2 BRPI0912512-4A BRPI0912512A BRPI0912512A2 BR PI0912512 A2 BRPI0912512 A2 BR PI0912512A2 BR PI0912512 A BRPI0912512 A BR PI0912512A BR PI0912512 A2 BRPI0912512 A2 BR PI0912512A2
Authority
BR
Brazil
Prior art keywords
compounds
preparation
Prior art date
Application number
BRPI0912512-4A
Other languages
English (en)
Inventor
Stéphanie AUBOURG
Bernard Boudet
Daniel Cravo
Matthias Helmreich
Original Assignee
Poxel Sas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poxel Sas filed Critical Poxel Sas
Publication of BRPI0912512A2 publication Critical patent/BRPI0912512A2/pt
Publication of BRPI0912512B1 publication Critical patent/BRPI0912512B1/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D251/00Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/10Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BRPI0912512A 2008-05-23 2009-04-24 processo para a preparação de compostos 3,6-diidro-1,3,5-triazina BRPI0912512B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08009483 2008-05-23
PCT/EP2009/002997 WO2009141040A2 (en) 2008-05-23 2009-04-24 Process for the synthesis of 3,6-dihydro-1,3,5-triazine derivatives

Publications (2)

Publication Number Publication Date
BRPI0912512A2 true BRPI0912512A2 (pt) 2015-07-28
BRPI0912512B1 BRPI0912512B1 (pt) 2018-09-11

Family

ID=40791625

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0912512A BRPI0912512B1 (pt) 2008-05-23 2009-04-24 processo para a preparação de compostos 3,6-diidro-1,3,5-triazina

Country Status (21)

Country Link
US (1) US20110124860A1 (pt)
EP (1) EP2300444B1 (pt)
JP (1) JP5458093B2 (pt)
KR (1) KR101618198B1 (pt)
CN (1) CN102036970A (pt)
AU (1) AU2009250149B2 (pt)
BR (1) BRPI0912512B1 (pt)
CA (1) CA2725011A1 (pt)
CY (1) CY1117855T1 (pt)
DK (1) DK2300444T3 (pt)
EA (1) EA018921B1 (pt)
ES (1) ES2571793T3 (pt)
HR (1) HRP20160414T1 (pt)
HU (1) HUE027532T2 (pt)
IL (1) IL209198A (pt)
MX (1) MX2010012741A (pt)
PL (1) PL2300444T3 (pt)
RS (1) RS54736B1 (pt)
SI (1) SI2300444T1 (pt)
WO (1) WO2009141040A2 (pt)
ZA (1) ZA201009160B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2646422T3 (pl) 2010-12-01 2015-12-31 Poxel Rozdział enancjomerów pochodnych triazyny z zastosowaniem kwasu winowego
CN105753801B (zh) * 2016-03-25 2018-06-01 浙江工业大学 一种均三嗪类化合物的制备方法
US11617754B2 (en) 2017-10-02 2023-04-04 Poxel Sa Methods of treating heart failure with preserved ejection fraction
CN112218623A (zh) 2018-06-14 2021-01-12 博希尔公司 用于治疗糖尿病的包含三嗪衍生物的薄膜包衣片剂
CN114681464A (zh) * 2020-12-28 2022-07-01 南京理工大学 二甲双胍类似物在制备脑缺血再灌注损伤预防和治疗药物中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2804113B1 (fr) * 2000-01-26 2004-06-18 Lipha Derives animes de dihydro-1,3,5-triazine et leurs applications en therapeutique
AU2003289375A1 (en) * 2002-12-17 2004-07-09 Hamari Chemicals, Ltd Novel 2,4-diamino-1,3,5-triazine derivative
FR2853650B1 (fr) * 2003-04-10 2006-07-07 Merck Sante Sas Procede de dedoublement d'amines utiles pour le traitement de desordres associes au syndrome d'insulino-resistance
DE102007054416A1 (de) * 2007-11-13 2009-05-14 Studiengesellschaft Kohle Mbh Verfahren zur Herstellung von 3,6-Dihydro-1,3,5- Triazin-Derivaten für die Behandlungen von Erkrankungen, die mit dem Insulinresistenz-Syndrom assoziiert sind

Also Published As

Publication number Publication date
RS54736B1 (sr) 2016-10-31
IL209198A0 (en) 2011-01-31
CN102036970A (zh) 2011-04-27
AU2009250149A1 (en) 2009-11-26
EA201001828A1 (ru) 2011-04-29
EP2300444A2 (en) 2011-03-30
HUE027532T2 (en) 2016-10-28
HRP20160414T1 (hr) 2016-05-20
MX2010012741A (es) 2010-12-21
CY1117855T1 (el) 2017-05-17
US20110124860A1 (en) 2011-05-26
ES2571793T3 (es) 2016-05-26
IL209198A (en) 2013-11-28
KR101618198B1 (ko) 2016-05-04
EA018921B1 (ru) 2013-11-29
WO2009141040A2 (en) 2009-11-26
EP2300444B1 (en) 2016-04-13
WO2009141040A3 (en) 2010-01-21
ZA201009160B (en) 2011-10-26
KR20110013498A (ko) 2011-02-09
DK2300444T3 (en) 2016-05-23
AU2009250149B2 (en) 2013-05-23
JP5458093B2 (ja) 2014-04-02
SI2300444T1 (sl) 2016-10-28
CA2725011A1 (en) 2009-11-26
BRPI0912512B1 (pt) 2018-09-11
JP2011520930A (ja) 2011-07-21
PL2300444T3 (pl) 2016-08-31

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 24/04/2009, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 13A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2667 DE 15-02-2022 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.