BRPI0606606A2 - composições estáveis contendo prostaglandina - Google Patents

composições estáveis contendo prostaglandina

Info

Publication number
BRPI0606606A2
BRPI0606606A2 BRPI0606606-2A BRPI0606606A BRPI0606606A2 BR PI0606606 A2 BRPI0606606 A2 BR PI0606606A2 BR PI0606606 A BRPI0606606 A BR PI0606606A BR PI0606606 A2 BRPI0606606 A2 BR PI0606606A2
Authority
BR
Brazil
Prior art keywords
prostaglandin
containing compositions
acid ester
chemical stability
alkanoic acid
Prior art date
Application number
BRPI0606606-2A
Other languages
English (en)
Inventor
Victor Deaciuc
Michael Hagan
Hashem Heiati
Karem Kostick Jette
Gregory C Visor
Ian G C Mcaffer
Peter Tasko
Original Assignee
Breath Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Breath Ltd filed Critical Breath Ltd
Publication of BRPI0606606A2 publication Critical patent/BRPI0606606A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

COMPOSIçõES ESTáVEIS CONTENDO PROSTAGLANDINA. A presente invenção se refere à composição farmacêutica contendo uma prostaglandina e um éster de ácido alcanóico de um sorbitol polietoxilado em uma quantidade eficaz para intensificar a estabilidade química da prostaglandina e o uso da mesma para o tratamento de condições oftálmicas. Também divulgados são métodos para intensificação da estabilidade química de uma composição contendo prostaglandina através de uso de um éster de ácido alcanóico de um sorbitol polietoxilado.
BRPI0606606-2A 2005-01-20 2006-01-18 composições estáveis contendo prostaglandina BRPI0606606A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0501192.9A GB0501192D0 (en) 2005-01-20 2005-01-20 Stable prostaglandin-containing compositions
PCT/US2006/001626 WO2006078659A2 (en) 2005-01-20 2006-01-18 Stable prostaglandin-containing compositions

Publications (1)

Publication Number Publication Date
BRPI0606606A2 true BRPI0606606A2 (pt) 2009-07-07

Family

ID=34259405

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0606606-2A BRPI0606606A2 (pt) 2005-01-20 2006-01-18 composições estáveis contendo prostaglandina

Country Status (16)

Country Link
US (2) US8084501B2 (pt)
EP (1) EP1843744A2 (pt)
JP (2) JP2008528490A (pt)
KR (1) KR20070094793A (pt)
CN (1) CN101106973A (pt)
AU (1) AU2006206649B2 (pt)
BR (1) BRPI0606606A2 (pt)
CA (1) CA2595237A1 (pt)
CZ (1) CZ2007555A3 (pt)
GB (1) GB0501192D0 (pt)
IL (1) IL184111A0 (pt)
IS (1) IS8665A (pt)
NO (1) NO20073699L (pt)
NZ (1) NZ556117A (pt)
WO (1) WO2006078659A2 (pt)
ZA (1) ZA200705428B (pt)

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ES2394130T3 (es) 2007-11-30 2013-01-22 Toltec Pharmaceuticals, Llc Composiciones y métodos para tratar infecciones vaginales y biopelículas vaginales patógenas
TWI544927B (zh) 2008-03-17 2016-08-11 愛爾康研究有限公司 具有低濃度的表面活性劑以促進治療劑之生物可利用性的藥學組成物
EP2127638A1 (en) 2008-05-30 2009-12-02 Santen Pharmaceutical Co., Ltd Method and composition for treating ocular hypertension and glaucoma
EP2328574A1 (en) * 2008-08-05 2011-06-08 University College Cork-National University of Ireland, Cork Treatment of retinal degeneration
US20100087540A1 (en) * 2008-10-07 2010-04-08 R-Tech Ueno, Ltd. Pharmaceutical composition
US20120232139A1 (en) * 2009-09-01 2012-09-13 Ryuji Ueno Composition for ocular topical administration treatment ocular hypertension and glaucoma
AU2010314863A1 (en) * 2009-11-09 2012-06-14 Allergan, Inc. Compositions for enhancing hair growth
TWI478730B (zh) * 2009-12-03 2015-04-01 Alcon Res Ltd 眼科乳劑
WO2012141334A1 (en) * 2011-04-12 2012-10-18 R-Tech Ueno, Ltd. Aqueous ophthalmic composition
DE102011108948A1 (de) * 2011-07-29 2013-01-31 Achim Göpferich Wässrige, kolloidale Lösungen von lipophilen Substanzen,insbesondere Arzneistofflösungen
CN104208015A (zh) * 2013-05-29 2014-12-17 天津金耀集团有限公司 含有曲伏***素和防腐剂的眼部制剂
EP3103439B1 (en) * 2015-06-09 2019-08-07 MEDproject Pharma-Entwicklungs- und Vertriebsgesellschaft mbH Drippable ophthalmic bimatoprost gel
EP3643297A4 (en) 2017-06-22 2021-03-17 Yonsung Fine Chemical Co., Ltd. OPHTHALMIC COMPOSITION FOR GLUCOMA TREATMENT
EP4331600A1 (en) * 2021-04-30 2024-03-06 Innovent Biologics (Suzhou) Co., Ltd. Oxm3 storage agent, oxm3 preparation, and preparation method

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Also Published As

Publication number Publication date
AU2006206649B2 (en) 2010-05-27
CN101106973A (zh) 2008-01-16
WO2006078659A3 (en) 2006-11-16
WO2006078659A2 (en) 2006-07-27
ZA200705428B (en) 2008-09-25
EP1843744A2 (en) 2007-10-17
US20060270735A1 (en) 2006-11-30
AU2006206649A1 (en) 2006-07-27
JP2013056948A (ja) 2013-03-28
JP2008528490A (ja) 2008-07-31
KR20070094793A (ko) 2007-09-21
WO2006078659A8 (en) 2007-08-30
IS8665A (is) 2007-08-02
CA2595237A1 (en) 2006-07-27
NO20073699L (no) 2007-10-19
IL184111A0 (en) 2007-10-31
CZ2007555A3 (cs) 2007-10-10
US20120065258A1 (en) 2012-03-15
US8084501B2 (en) 2011-12-27
NZ556117A (en) 2009-10-30
GB0501192D0 (en) 2005-03-02

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 9A E 10A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.