BR9709065A - Alkylaminobenzothiazole derivatives e-benzoxazole - Google Patents

Alkylaminobenzothiazole derivatives e-benzoxazole

Info

Publication number: BR9709065A
Authority: BR; Brazil
Prior art keywords: alkylaminobenzothiazole; benzoxazole; derivatives; alkylaminobenzothiazole derivatives
Prior art date: 1996-05-10

Application number

BR9709065A

Other languages

Portuguese (pt)

Inventor

Ludo Edmond Josephine Kennis

Josephus Carolus Mertens

Serge Maria Aloysius Pieters

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-05-10

Filing date

1997-05-02

Publication date

1999-08-03

1997-05-02 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1999-08-03 Publication of BR9709065A publication Critical patent/BR9709065A/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/002—Heterocyclic compounds
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms

BR9709065A 1996-05-10 1997-05-02 Alkylaminobenzothiazole derivatives e-benzoxazole BR9709065A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP96201282		1996-05-10
PCT/EP1997/002505 WO1997043271A1 (en)	1996-05-10	1997-05-02	Alkylaminobenzothiazole and -benzoxazole derivatives

Publications (1)

Publication Number	Publication Date
BR9709065A true BR9709065A (en)	1999-08-03

Family

ID=8223970

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9709065A BR9709065A (en)	1996-05-10	1997-05-02	Alkylaminobenzothiazole derivatives e-benzoxazole

Country Status (29)

Country	Link
US (2)	US6103725A (en)
EP (2)	EP1325917B1 (en)
JP (1)	JP3237759B2 (en)
KR (1)	KR100330699B1 (en)
CN (1)	CN1074766C (en)
AR (1)	AR007079A1 (en)
AT (2)	ATE350373T1 (en)
AU (1)	AU710175B2 (en)
BG (1)	BG64097B1 (en)
BR (1)	BR9709065A (en)
CA (1)	CA2253453C (en)
CZ (1)	CZ295639B6 (en)
DE (2)	DE69737217T2 (en)
EA (1)	EA001360B1 (en)
EE (1)	EE03563B1 (en)
ES (2)	ES2230605T3 (en)
HK (2)	HK1057044A1 (en)
HU (1)	HUP9902993A3 (en)
ID (1)	ID16889A (en)
IL (1)	IL126968A0 (en)
MY (1)	MY117852A (en)
NO (1)	NO311027B1 (en)
NZ (1)	NZ332309A (en)
PL (1)	PL190721B1 (en)
SK (1)	SK282919B6 (en)
TR (1)	TR199802253T2 (en)
TW (1)	TW593290B (en)
WO (1)	WO1997043271A1 (en)
ZA (1)	ZA974053B (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1293804B1 (en)	1997-08-01	1999-03-10	Recordati Chem Pharm	DIARYLALKYL PIPERAZINS ACTIVE ON LOW URINARY TRACT
US6281216B1 (en) *	1998-02-09	2001-08-28	Duphar International Research B.V.	2-aminoquinoline derivatives having d4-agonistic activity
EP0982030A3 (en) *	1998-08-17	2000-05-10	Pfizer Products Inc.	2,7-substituted octahydro-pyrrolo 1,2-a]pyrazine derivatives as 5ht 1a ligands
WO2000018767A2 (en) *	1998-09-30	2000-04-06	Neurogen Corporation	2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
US6284759B1 (en)	1998-09-30	2001-09-04	Neurogen Corporation	2-piperazinoalkylaminobenzo-azole derivatives: dopamine receptor subtype specific ligands
US6107313A (en) *	1998-10-02	2000-08-22	Combichem, Inc.	Dopamine receptor antagonists
AU5569800A (en) *	1999-06-30	2001-01-31	Santen Pharmaceutical Co. Ltd.	Brain sigma-1 receptor-binding ligand
US6908929B2 (en)	2000-03-31	2005-06-21	Ortho-Mcneil Pharmaceutical, Inc.	Phenyl-substituted imidazopyridines
US6436939B2 (en)	2000-03-31	2002-08-20	Ortho-Mcneil Pharmaceutical, Inc.	Method for using 2-aryloxyalkylaminobenzoxazoles and 2-aryloxyalkylaminobenzothiazoles as H3 antagonists
GB0203299D0 (en) *	2002-02-12	2002-03-27	Glaxo Group Ltd	Novel compounds
KR20050033662A (en) *	2002-09-06	2005-04-12	얀센 파마슈티카 엔.브이.	Heterocyclic compounds
US8257680B1 (en)	2004-02-24	2012-09-04	The General Hospital Corporation	Catalytic radiofluorination
EP2388017B1 (en) *	2004-02-24	2014-12-24	The General Hospital Corporation	Catalytic radiofluorination
US9017724B2 (en)	2004-02-24	2015-04-28	The General Hospital Corporation	Catalytic radiofluorination
FR2877005A1 (en) *	2004-10-22	2006-04-28	Bioprojet Soc Civ Ile	NEW ARYLPIPERAZINE DERIVATIVES
US7731940B2 (en)	2006-01-25	2010-06-08	The Regents Of The University Of California	Compositions and methods related to serotonin 5-HT1A receptors
JP5501339B2 (en)	2008-03-21	2014-05-21	ザジェネラルホスピタルコーポレイション	Compounds and compositions for detection and treatment of Alzheimer's disease and related diseases
US11337970B2 (en) *	2016-08-26	2022-05-24	Bristol-Myers Squibb Company	Inhibitors of indoleamine 2,3-dioxygenase and methods of their use
PT109740B (en)	2016-11-14	2020-07-30	Hovione Farmaciencia Sa	PROCESS FOR THE PREPARATION OF UMECLIDINUM BROMIDE
KR20210091865A (en) *	2020-01-14	2021-07-23	서울대학교산학협력단	N-phenylbenzothiazol-2-amine Compounds Having Vascular Tube Formation Inhibition Effect and Pharmaceutical Composition Comprising the Same

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1985005359A1 (en) *	1984-05-22	1985-12-05	Sumitomo Chemical Company, Limited	Novel radioactive iodospiroperidol and process for its preparation
DE3874187T2 (en) *	1987-04-08	1993-04-08	Salutar Inc	PROOF FOR AMYLOIDOSE AND ALZHEIMER'S DISEASE AND REAGENT HERE.
US4929618A (en) *	1988-03-25	1990-05-29	Ube Industries, Ltd.	Piperdine and piperazine derivatives, and antihistaminic pharmaceutical compositions containing the same
FR2656609B1 (en) *	1989-12-28	1992-03-27	Synthelabo	2-AMINOPYRIMIDINE-4-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
US5731438A (en) *	1996-08-01	1998-03-24	Isis Pharmaceuticals, Inc.	N-(aminoalkyl)-and/or N-(amidoalkyl)-dinitrogen heterocycles

1997
- 1997-05-01 TW TW086105767A patent/TW593290B/en not_active IP Right Cessation
- 1997-05-02 EP EP03075959A patent/EP1325917B1/en not_active Expired - Lifetime
- 1997-05-02 ES ES97923913T patent/ES2230605T3/en not_active Expired - Lifetime
- 1997-05-02 JP JP54053597A patent/JP3237759B2/en not_active Expired - Lifetime
- 1997-05-02 DE DE69737217T patent/DE69737217T2/en not_active Expired - Lifetime
- 1997-05-02 DE DE69730962T patent/DE69730962T2/en not_active Expired - Lifetime
- 1997-05-02 HU HU9902993A patent/HUP9902993A3/en unknown
- 1997-05-02 US US09/180,369 patent/US6103725A/en not_active Expired - Lifetime
- 1997-05-02 PL PL97329849A patent/PL190721B1/en not_active IP Right Cessation
- 1997-05-02 EE EE9800378A patent/EE03563B1/en not_active IP Right Cessation
- 1997-05-02 NZ NZ332309A patent/NZ332309A/en unknown
- 1997-05-02 AT AT03075959T patent/ATE350373T1/en not_active IP Right Cessation
- 1997-05-02 EA EA199801000A patent/EA001360B1/en not_active IP Right Cessation
- 1997-05-02 ES ES03075959T patent/ES2279923T3/en not_active Expired - Lifetime
- 1997-05-02 TR TR1998/02253T patent/TR199802253T2/en unknown
- 1997-05-02 AU AU29560/97A patent/AU710175B2/en not_active Ceased
- 1997-05-02 EP EP97923913A patent/EP0912533B1/en not_active Expired - Lifetime
- 1997-05-02 BR BR9709065A patent/BR9709065A/en not_active IP Right Cessation
- 1997-05-02 WO PCT/EP1997/002505 patent/WO1997043271A1/en active IP Right Grant
- 1997-05-02 IL IL12696897A patent/IL126968A0/en not_active IP Right Cessation
- 1997-05-02 CN CN97194515A patent/CN1074766C/en not_active Expired - Lifetime
- 1997-05-02 SK SK1532-98A patent/SK282919B6/en not_active IP Right Cessation
- 1997-05-02 CZ CZ19983553A patent/CZ295639B6/en not_active IP Right Cessation
- 1997-05-02 KR KR1019980707914A patent/KR100330699B1/en not_active IP Right Cessation
- 1997-05-02 CA CA002253453A patent/CA2253453C/en not_active Expired - Fee Related
- 1997-05-02 AT AT97923913T patent/ATE277917T1/en not_active IP Right Cessation
- 1997-05-07 MY MYPI97002022A patent/MY117852A/en unknown
- 1997-05-09 AR ARP970101955A patent/AR007079A1/en active IP Right Grant
- 1997-05-09 ZA ZA974053A patent/ZA974053B/en unknown
- 1997-05-09 ID IDP971546A patent/ID16889A/en unknown
1998
- 1998-10-07 BG BG102819A patent/BG64097B1/en unknown
- 1998-11-09 NO NO19985227A patent/NO311027B1/en unknown
1999
- 1999-08-16 HK HK03109371A patent/HK1057044A1/en not_active IP Right Cessation
- 1999-08-16 HK HK99103545A patent/HK1018457A1/en not_active IP Right Cessation
2000
- 2000-06-27 US US09/604,427 patent/US6224849B1/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
KR20000005227A (en)	2000-01-25
CN1074766C (en)	2001-11-14
TW593290B (en)	2004-06-21
PL190721B1 (en)	2005-12-30
ATE277917T1 (en)	2004-10-15
ATE350373T1 (en)	2007-01-15
ID16889A (en)	1997-11-20
EA199801000A1 (en)	1999-04-29
EP0912533A1 (en)	1999-05-06
DE69737217D1 (en)	2007-02-15
NO985227L (en)	1999-01-11
KR100330699B1 (en)	2002-08-27
CN1218461A (en)	1999-06-02
CA2253453A1 (en)	1997-11-20
BG102819A (en)	1999-08-31
DE69730962T2 (en)	2006-03-30
EP1325917B1 (en)	2007-01-03
JP2000503667A (en)	2000-03-28
EE03563B1 (en)	2001-12-17
US6103725A (en)	2000-08-15
CA2253453C (en)	2007-01-16
ES2279923T3 (en)	2007-09-01
SK153298A3 (en)	1999-03-12
HK1018457A1 (en)	1999-12-24
HK1057044A1 (en)	2004-03-12
US6224849B1 (en)	2001-05-01
NO985227D0 (en)	1998-11-09
BG64097B1 (en)	2003-12-31
AU710175B2 (en)	1999-09-16
AR007079A1 (en)	1999-10-13
HUP9902993A3 (en)	2002-01-28
EP0912533B1 (en)	2004-09-29
EE9800378A (en)	1999-04-15
DE69737217T2 (en)	2007-11-08
CZ355398A3 (en)	1999-02-17
AU2956097A (en)	1997-12-05
ZA974053B (en)	1998-11-09
JP3237759B2 (en)	2001-12-10
WO1997043271A1 (en)	1997-11-20
PL329849A1 (en)	1999-04-12
TR199802253T2 (en)	1999-02-22
SK282919B6 (en)	2003-01-09
HUP9902993A2 (en)	2000-05-28
CZ295639B6 (en)	2005-09-14
NZ332309A (en)	1999-08-30
MY117852A (en)	2004-08-30
NO311027B1 (en)	2001-10-01
DE69730962D1 (en)	2004-11-04
EP1325917A1 (en)	2003-07-09
EA001360B1 (en)	2001-02-26
ES2230605T3 (en)	2005-05-01
IL126968A0 (en)	1999-09-22

Legal Events

Date	Code	Title	Description
2008-03-11	B06A	Patent application procedure suspended [chapter 6.1 patent gazette]
2012-06-19	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE AS 13A, 14A E 15A ANUIDADES.
2012-11-20	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 13A, 14A E 15A ANUIDADES.

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ATE323682T1 (en)	2006-05-15	ARYL-PYRIMIDINE DERIVATIVES
PT1005446E (en)	2004-06-30	N-AROYLPHENYLALANINE DERIVATIVES
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ATE208395T1 (en)	2001-11-15	THIOPHENOPYRIMIDINES
ATE262512T1 (en)	2004-04-15	ARYLALKANOYLPYRIDAZINE
DE69732576D1 (en)	2005-03-31	TETRAHYDROBENZINDOLON DERIVATIVES
BR9709065A (en)	1999-08-03	Alkylaminobenzothiazole derivatives e-benzoxazole
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