BR8103216A - 2-nitroimidazois,sua preparacao,composicao filaricida e uso - Google Patents

2-nitroimidazois,sua preparacao,composicao filaricida e uso

Info

Publication number
BR8103216A
BR8103216A BR8103216A BR8103216A BR8103216A BR 8103216 A BR8103216 A BR 8103216A BR 8103216 A BR8103216 A BR 8103216A BR 8103216 A BR8103216 A BR 8103216A BR 8103216 A BR8103216 A BR 8103216A
Authority
BR
Brazil
Prior art keywords
philaricide
nitroimidazois
preparation
composition
philaricide composition
Prior art date
Application number
BR8103216A
Other languages
English (en)
Inventor
H Stohler
W Hofheinz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR8103216A publication Critical patent/BR8103216A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91Nitro radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR8103216A 1980-05-23 1981-05-22 2-nitroimidazois,sua preparacao,composicao filaricida e uso BR8103216A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH405780 1980-05-23

Publications (1)

Publication Number Publication Date
BR8103216A true BR8103216A (pt) 1982-02-16

Family

ID=4269011

Family Applications (1)

Application Number Title Priority Date Filing Date
BR8103216A BR8103216A (pt) 1980-05-23 1981-05-22 2-nitroimidazois,sua preparacao,composicao filaricida e uso

Country Status (11)

Country Link
US (2) US4366166A (pt)
EP (1) EP0040761A1 (pt)
JP (1) JPS5711969A (pt)
AU (1) AU541912B2 (pt)
BR (1) BR8103216A (pt)
GB (1) GB2076402B (pt)
IN (1) IN155338B (pt)
MW (1) MW1681A1 (pt)
OA (1) OA06794A (pt)
PH (1) PH16858A (pt)
ZW (1) ZW8781A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE19071T1 (de) * 1982-02-19 1986-04-15 Ciba Geigy Ag Mikrobizide und wuchsregulierende mittel.
US4568111A (en) * 1983-08-29 1986-02-04 The United States Of America As Represented By The United States Department Of Energy Detachable connection for a nuclear reactor fuel assembly
AU4327585A (en) * 1984-06-21 1986-01-02 Imperial Chemical Industries Plc Antifungal azole compounds
CA1329206C (en) * 1987-06-10 1994-05-03 Tsutomu Kagiya Fluorine-containing nitroazole derivatives and radiosensitizer comprising the same
FR2684382B1 (fr) * 1991-12-02 1994-10-21 Rhone Merieux Medicaments et preparations pures de dichlorhydrate de melarsomine, leur procede d'obtention et produits intermediaires obtenus.
JP3577079B2 (ja) * 1992-12-18 2004-10-13 ポーラ化成工業株式会社 光学活性2−ニトロイミダゾール誘導体
AU8074294A (en) * 1993-10-04 1995-05-01 Board Of Regents, The University Of Texas System Rapid synthesis and use of 18f-fluoromisonidazole and analogs
US6060604A (en) * 1995-03-31 2000-05-09 Florida State University Pharmaceutical compounds comprising polyamines substituted with electron-affinic groups
US5700825A (en) * 1995-03-31 1997-12-23 Florida State University Radiosensitizing diamines and their pharmaceutical preparations
US6423707B1 (en) 2000-08-28 2002-07-23 California Pacific Medical Center Nitroimidazole ester analogues and therapeutic applications
WO2005041853A2 (en) * 2003-10-28 2005-05-12 Ems S.A. Antibacterial and/or antiprotozoal nitroimidazole derivative compounds with urease inhibitor activity, process for preparing these compounds and use in pharmaceutical compositions and medicines.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3255201A (en) * 1965-04-09 1966-06-07 Hoffmann La Roche 2-nitroimidazoles
US3505349A (en) * 1966-04-18 1970-04-07 Hoffmann La Roche 2-nitro-imidazolyl-1-acetamides
US3641047A (en) * 1970-08-05 1972-02-08 Hoffmann La Roche 2-nitroimidazole derivatives substituted in the 1-position with a 2-oxo-propyl or semicarbazone group
CA1034126A (en) * 1974-01-17 1978-07-04 Alden G. Beaman 2-nitroimidazoles
IE47132B1 (en) * 1977-08-19 1983-12-28 Roche Products Ltd Novel nitroimidazoles and pharmaceutical preparations containing these as well as their manufacture

Also Published As

Publication number Publication date
GB2076402B (en) 1984-05-02
US4366166A (en) 1982-12-28
AU7064081A (en) 1981-11-26
JPS5711969A (en) 1982-01-21
IN155338B (pt) 1985-01-19
EP0040761A1 (de) 1981-12-02
ZW8781A1 (en) 1981-12-16
US4456610A (en) 1984-06-26
MW1681A1 (en) 1982-08-11
PH16858A (en) 1984-03-22
AU541912B2 (en) 1985-01-31
OA06794A (fr) 1982-12-31
GB2076402A (en) 1981-12-02

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