BR112019007980A2 - método para produzir 3-alquilsulfanil-2-cloro-n-(1-alquil-1h-tetrazol-5-il)-4-trifluorometil-benzamidas - Google Patents

método para produzir 3-alquilsulfanil-2-cloro-n-(1-alquil-1h-tetrazol-5-il)-4-trifluorometil-benzamidas

Info

Publication number
BR112019007980A2
BR112019007980A2 BR112019007980A BR112019007980A BR112019007980A2 BR 112019007980 A2 BR112019007980 A2 BR 112019007980A2 BR 112019007980 A BR112019007980 A BR 112019007980A BR 112019007980 A BR112019007980 A BR 112019007980A BR 112019007980 A2 BR112019007980 A2 BR 112019007980A2
Authority
BR
Brazil
Prior art keywords
alkyl
alkylsulfanyl
tetrazol
chloro
benzamides
Prior art date
Application number
BR112019007980A
Other languages
English (en)
Other versions
BR112019007980B1 (pt
Inventor
Gallenkamp Daniel
James Ford Mark
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112019007980A2 publication Critical patent/BR112019007980A2/pt
Publication of BR112019007980B1 publication Critical patent/BR112019007980B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • C07D257/06—Five-membered rings with nitrogen atoms directly attached to the ring carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/01—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton
    • C07C323/09—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C323/18—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C07C323/20—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton with singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton

Abstract

trata-se de um método para preparar 3-alquilsulfanil-2-cloro-n-(1-alquil-1h-tetrazol-5-il)-4-trifluorometilbenzamidas da fórmula (i). os substituintes r1 e r2 nas mesmas são radicais como alquila e fenila substituída.
BR112019007980-7A 2016-10-20 2017-10-16 Método para produzir 3-alquilsulfanil-2-cloro-n-(1-alquil1h-tetrazol-5-il)-4- trifluorometil-benzamidas e compostos intermediários BR112019007980B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16194840.1 2016-10-20
EP16194840 2016-10-20
PCT/EP2017/076307 WO2018073157A1 (de) 2016-10-20 2017-10-16 Verfahren zur herstellung von 3-alkylsulfanyl-2-chlor-n-(1-alkyl-1h-tetrazol-5-yl)-4-trifluoromethyl-benzamiden

Publications (2)

Publication Number Publication Date
BR112019007980A2 true BR112019007980A2 (pt) 2019-07-09
BR112019007980B1 BR112019007980B1 (pt) 2022-06-28

Family

ID=57184339

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112019007980-7A BR112019007980B1 (pt) 2016-10-20 2017-10-16 Método para produzir 3-alquilsulfanil-2-cloro-n-(1-alquil1h-tetrazol-5-il)-4- trifluorometil-benzamidas e compostos intermediários

Country Status (12)

Country Link
US (1) US10457651B2 (pt)
EP (1) EP3529233B1 (pt)
JP (1) JP6925418B2 (pt)
KR (1) KR102517500B1 (pt)
CN (1) CN109790109B (pt)
BR (1) BR112019007980B1 (pt)
DK (1) DK3529233T3 (pt)
ES (1) ES2824698T3 (pt)
IL (1) IL266044B (pt)
MX (1) MX2019004569A (pt)
TW (1) TWI741040B (pt)
WO (1) WO2018073157A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022194841A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194843A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194842A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
AU2022329086A1 (en) 2021-08-17 2024-02-08 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
WO2023020962A1 (en) 2021-08-17 2023-02-23 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
AU2022330302A1 (en) 2021-08-17 2024-02-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
EP4238972A1 (en) 2022-03-04 2023-09-06 Bayer AG Substituted 1,2,4-thiadiazolyl picolinamides, salts or n-oxides thereof and their use as herbicidally active substances
EP4238973A1 (en) 2022-03-04 2023-09-06 Bayer AG Substituted 1,2,4-thiadiazolyl isonicotinamides, salts or n-oxides thereof and their use as herbicidally active substances

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5618981A (en) * 1995-05-19 1997-04-08 Phillips Petroleum Company Process for producing aromatic sulfides
TWI319387B (en) * 2002-04-05 2010-01-11 Astrazeneca Ab Benzamide derivatives
EP2038264B1 (en) * 2006-06-29 2016-10-26 F.Hoffmann-La Roche Ag Tetrazole-substituted arylamides
EP2127521A1 (de) * 2008-05-29 2009-12-02 Bayer CropScience Aktiengesellschaft Herbizid wirksame 4-(3-Alkylsulfinylbenzoyl)pyrazole
AU2010278334A1 (en) * 2009-07-29 2012-03-08 Bayer Cropscience Ag 4-(3-alkylthiobenzoyl)pyrazoles and use thereof as herbicides
WO2012028579A1 (de) * 2010-09-01 2012-03-08 Bayer Cropscience Ag N-(tetrazol-5-yl)- und n-(triazol-5-yl)arylcarbonsäureamide und ihre verwendung als herbizide
EP2765128A1 (en) * 2013-02-07 2014-08-13 Almirall, S.A. Substituted benzamides with activity towards EP4 receptors
JP2018522870A (ja) 2015-07-03 2018-08-16 バイエル・クロップサイエンス・アクチェンゲゼルシャフト ２−クロロ−３−（メチルスルファニル）−ｎ−（１−メチル−１ｈ−テトラゾール−５−イル）−４−（トリフルオロメチル）ベンズアミドの熱力学的に安定な結晶変態

Also Published As

Publication number Publication date
TW201815772A (zh) 2018-05-01
BR112019007980B1 (pt) 2022-06-28
WO2018073157A1 (de) 2018-04-26
EP3529233A1 (de) 2019-08-28
ES2824698T3 (es) 2021-05-13
CN109790109B (zh) 2021-10-22
KR20190066051A (ko) 2019-06-12
EP3529233B1 (de) 2020-08-12
IL266044B (en) 2021-03-25
TWI741040B (zh) 2021-10-01
CN109790109A (zh) 2019-05-21
MX2019004569A (es) 2019-08-21
JP2019532963A (ja) 2019-11-14
IL266044A (en) 2019-06-30
DK3529233T3 (da) 2020-10-12
US20190233382A1 (en) 2019-08-01
US10457651B2 (en) 2019-10-29
JP6925418B2 (ja) 2021-08-25
KR102517500B1 (ko) 2023-04-03

Similar Documents

Publication Publication Date Title
BR112019007980A2 (pt) método para produzir 3-alquilsulfanil-2-cloro-n-(1-alquil-1h-tetrazol-5-il)-4-trifluorometil-benzamidas
SV2018005722A (es) Nuevos derivados de amonio, un proceso para su preparacion y composiciones farmaceuticas que los contienen
CY1120188T1 (el) ΠΑΡΑΓΩΓΑ ΝΑΦΘΥΡΙΔΙΝΗΣ ΧΡΗΣΙΜΑ ΩΣ ΑΝΤΑΓΩΝΙΣΤΕΣ ΙΝΤΕΓΚΡΙΝΗΣ αvβ6
TR201906366T4 (tr) Polisiklik-karbamoilpiridon bileşiklerinin sentezi.
UY36999A (es) Derivados de aryl oxadiazol fungicidas
UY35915A (es) Nuevos derivados tienopirimidina, un proceso para su preparación y composiciones farmacéuticas que los contienen
CU20180144A7 (es) Derivados de carbonucleósidos sustituidos útiles como agentes antineoplásicos
CR20170118A (es) Derivados espirodiamina como inhibidores de la aldosterona sintasa
EA201691799A1 (ru) Бициклические соединения в качестве ингибиторов продукции аутотаксина (atx) и лизофосфатидиловой кислоты (lpa)
EA201600091A1 (ru) 4-членные кольцевые карбоксамиды, применяемые в качестве нематоцидов
CU20180001A7 (es) Derivados de oxopiridina sustituidos y procesos para su preparación
CR20150470A (es) Derivados de triazolona de piridinilo y piridinilo fusionado
EA201790395A1 (ru) Производные аминотриазина, подходящие для применения в качестве соединений-ингибиторов tank-связывающей киназы
EA201691272A1 (ru) Тетрагидропиридопиразины в качестве модуляторов gpr6
UY35447A (es) Moduladores de p2x7
CR20170008A (es) Compuestos de [1,2,4] triazol e imidazol sustituidos
CO2017001528A2 (es) Compuestos novedosos de pirimidina sustituidos
PE20170440A1 (es) Derivados de isoindolina
CR20160198A (es) Derivados de etinilo-imidazolidín-2, 4-diona como moduladore mglur4
UY36221A (es) Derivados de isoindolinona
CY1120763T1 (el) Νεες ενωσεις σουλφονυλαμινοβενζαμιδιου
UY35997A (es) Derivados de isoquinoleína, su procedimiento de preparación y las composiciones farmacéuticas que los contienen
BR112019025028A2 (pt) Método para preparar um composto.
ECSP16074207A (es) Pirazinas moduladoras de gpr6
BR112016027455A2 (pt) moduladores ppar

Legal Events

Date Code Title Description
B350 Update of information on the portal [chapter 15.35 patent gazette]
B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 16/10/2017, OBSERVADAS AS CONDICOES LEGAIS