BR0004066A - Composto ou um éster ou sal deste farmaceuticamente aceitáveis, uso do mesmo, composição farmacêutica, e, composto ou um derivado de acetal deste - Google Patents

Composto ou um éster ou sal deste farmaceuticamente aceitáveis, uso do mesmo, composição farmacêutica, e, composto ou um derivado de acetal deste

Info

Publication number
BR0004066A
BR0004066A BR0004066-5A BR0004066A BR0004066A BR 0004066 A BR0004066 A BR 0004066A BR 0004066 A BR0004066 A BR 0004066A BR 0004066 A BR0004066 A BR 0004066A
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutically acceptable
salt
pharmaceutical composition
acetal derivative
Prior art date
Application number
BR0004066-5A
Other languages
English (en)
Inventor
Toshiyuki Konosu
Sadao Oida
Makoto Mori
Takuya Uchida
Satoshi Ohya
Akihiko Nakagawa
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of BR0004066A publication Critical patent/BR0004066A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/56—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and doubly-bound oxygen atoms bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"COMPOSTO OU UM éSTER OU SAL DESTE FARMACEUTICAMENTE ACEITáVEIS, USO DO MESMO, COMPOSIçãO FARMACêUTICA, E, COMPOSTO OU UM DERIVADO DE ACETAL DESTE". Compostos da seguinte fórmula (I) e seus sais e derivados de éster farmaceuticamente aceitáveis: em que Ar é um grupo fenila que pode ser opcionalmente substituído por 1 a 3 substituintes selecionados do grupo que consiste de átomos halógenos e de grupos trifluorometila, têm excelente atividade anti-fúngica.
BR0004066-5A 1999-09-09 2000-09-08 Composto ou um éster ou sal deste farmaceuticamente aceitáveis, uso do mesmo, composição farmacêutica, e, composto ou um derivado de acetal deste BR0004066A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP25570299 1999-09-09
JP2000103826 2000-04-05

Publications (1)

Publication Number Publication Date
BR0004066A true BR0004066A (pt) 2001-04-17

Family

ID=26542380

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0004066-5A BR0004066A (pt) 1999-09-09 2000-09-08 Composto ou um éster ou sal deste farmaceuticamente aceitáveis, uso do mesmo, composição farmacêutica, e, composto ou um derivado de acetal deste

Country Status (23)

Country Link
US (3) US6391903B1 (pt)
EP (1) EP1083175B1 (pt)
KR (1) KR100592201B1 (pt)
CN (1) CN1167700C (pt)
AR (1) AR025610A1 (pt)
AT (1) ATE244238T1 (pt)
AU (1) AU778073B2 (pt)
BR (1) BR0004066A (pt)
CA (1) CA2317691C (pt)
DE (1) DE60003618T2 (pt)
DK (1) DK1083175T3 (pt)
ES (1) ES2200786T3 (pt)
HK (1) HK1034259A1 (pt)
HU (1) HU224699B1 (pt)
ID (1) ID27234A (pt)
IL (1) IL138329A0 (pt)
NO (1) NO318352B1 (pt)
NZ (1) NZ506818A (pt)
PT (1) PT1083175E (pt)
RU (1) RU2203280C2 (pt)
SA (1) SA00210602B1 (pt)
TR (1) TR200002610A3 (pt)
TW (1) TW530057B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI334866B (en) 2002-05-29 2010-12-21 Mercian Corp Novel physiologically active substances
WO2004108134A1 (ja) * 2003-06-06 2004-12-16 Sankyo Company, Limited トリアゾール化合物を含有する医薬組成物
KR101191682B1 (ko) * 2005-12-01 2012-10-16 바실리어 파마슈티카 아게 에폭시부탄올 중간체의 제조 방법
EP2116542A4 (en) 2007-01-29 2011-05-04 Eisai R&D Man Co Ltd SOLID OF A MAKROLIDE COMPOUND, METHOD OF MANUFACTURING THEREOF AND PHARMACEUTICAL COMPOSITION THEREWITH

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8322983D0 (en) * 1983-08-26 1983-09-28 Pfizer Ltd Triazole antifungal agents
US4483863A (en) * 1984-01-20 1984-11-20 Pfizer Inc. Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
CA2049802A1 (en) * 1990-08-26 1992-02-27 Sadao Oida Anti-fungal triazole derivatives, their preparation and uses
HU227320B1 (en) 1995-04-06 2011-03-28 Daiichi Sankyo Co Ltd 1,2,4-triazole-derivatives, fungicide compositions containing these compounds as active ingredients
JP2902345B2 (ja) 1995-04-06 1999-06-07 三共株式会社 トリアゾール抗真菌剤
EP0780380B1 (en) * 1995-12-22 2001-06-13 Ss Pharmaceutical Co., Ltd. Triazole derivatives with antimycotic action and intermediates
JP3622882B2 (ja) 1996-10-04 2005-02-23 三共株式会社 トリアゾール誘導体を含有する医薬
AU5779598A (en) 1997-02-04 1998-08-25 Sankyo Company Limited Triazole derivatives
AU7937998A (en) 1997-07-08 1999-02-08 Sankyo Company Limited Antifungal triazole compounds
US6303728B1 (en) 1997-07-08 2001-10-16 Kaneka Corporation Hydrosilylation process and polymers produced by the process
JPH1180135A (ja) 1997-07-08 1999-03-26 Sankyo Co Ltd 抗真菌トリアゾール化合物

Also Published As

Publication number Publication date
TR200002610A2 (tr) 2001-06-21
AU5657500A (en) 2001-03-15
US6392082B1 (en) 2002-05-21
CN1291610A (zh) 2001-04-18
IL138329A0 (en) 2001-10-31
EP1083175A2 (en) 2001-03-14
NZ506818A (en) 2001-07-27
NO20004511L (no) 2001-03-12
US6337403B1 (en) 2002-01-08
HUP0003555A2 (hu) 2002-05-29
TR200002610A3 (tr) 2001-06-21
EP1083175A3 (en) 2001-04-11
ID27234A (id) 2001-03-15
CA2317691C (en) 2009-02-17
DK1083175T3 (da) 2003-10-06
CA2317691A1 (en) 2001-03-09
AU778073B2 (en) 2004-11-11
RU2203280C2 (ru) 2003-04-27
PT1083175E (pt) 2003-09-30
KR20010067169A (ko) 2001-07-12
TW530057B (en) 2003-05-01
HU0003555D0 (en) 2000-09-08
DE60003618D1 (de) 2003-08-07
CN1167700C (zh) 2004-09-22
US6391903B1 (en) 2002-05-21
SA00210602B1 (ar) 2006-06-04
HK1034259A1 (en) 2001-10-19
AR025610A1 (es) 2002-12-04
KR100592201B1 (ko) 2006-06-23
ATE244238T1 (de) 2003-07-15
HU224699B1 (en) 2006-01-30
NO20004511D0 (no) 2000-09-08
DE60003618T2 (de) 2004-04-15
NO318352B1 (no) 2005-03-07
EP1083175B1 (en) 2003-07-02
ES2200786T3 (es) 2004-03-16

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements