BE865182A - Derives de la morphine, leur procede de preparation et leur application comme medicament - Google Patents

Derives de la morphine, leur procede de preparation et leur application comme medicament

Info

Publication number
BE865182A
BE865182A BE186173A BE186173A BE865182A BE 865182 A BE865182 A BE 865182A BE 186173 A BE186173 A BE 186173A BE 186173 A BE186173 A BE 186173A BE 865182 A BE865182 A BE 865182A
Authority
BE
Belgium
Prior art keywords
preparation
application
medicinal product
morphine derivatives
morphine
Prior art date
Application number
BE186173A
Other languages
English (en)
French (fr)
Original Assignee
Reckitt & Colmann Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt & Colmann Prod Ltd filed Critical Reckitt & Colmann Prod Ltd
Publication of BE865182A publication Critical patent/BE865182A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BE186173A 1977-03-23 1978-03-22 Derives de la morphine, leur procede de preparation et leur application comme medicament BE865182A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB12342/77A GB1587831A (en) 1977-03-23 1977-03-23 Morphine derivatives

Publications (1)

Publication Number Publication Date
BE865182A true BE865182A (fr) 1978-09-22

Family

ID=10002756

Family Applications (1)

Application Number Title Priority Date Filing Date
BE186173A BE865182A (fr) 1977-03-23 1978-03-22 Derives de la morphine, leur procede de preparation et leur application comme medicament

Country Status (25)

Country Link
US (1) US4241067A (ru)
JP (1) JPS53121798A (ru)
AR (1) AR218296A1 (ru)
AT (1) AT360664B (ru)
AU (1) AU518614B2 (ru)
BE (1) BE865182A (ru)
CA (1) CA1089455A (ru)
CH (1) CH630629A5 (ru)
CS (1) CS199522B2 (ru)
DD (1) DD135081A5 (ru)
DE (1) DE2812581A1 (ru)
DK (1) DK149753C (ru)
ES (1) ES468170A1 (ru)
FR (1) FR2384775A1 (ru)
GB (1) GB1587831A (ru)
HU (1) HU177722B (ru)
IE (1) IE46442B1 (ru)
IT (1) IT1105172B (ru)
LU (1) LU79295A1 (ru)
NL (1) NL7803084A (ru)
NZ (1) NZ186693A (ru)
PL (1) PL111722B1 (ru)
SE (1) SE436132B (ru)
SU (1) SU856381A3 (ru)
ZA (1) ZA781525B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4362870A (en) * 1980-01-16 1982-12-07 Regents Of The University Of Minnesota Selective opioid receptor alkylating agents
US4401672A (en) * 1981-10-13 1983-08-30 Regents Of The University Of Minnesota Non-addictive narcotic antitussive preparation
DE3381877D1 (de) * 1982-03-16 1990-10-18 Univ Rockefeller Verwendung von opium antagonisten zur herstellung von arzneimitteln zur behebung gastro-intestinaler stoerungen.
GB8711558D0 (en) * 1987-05-15 1987-06-17 Reckitt & Colmann Prod Ltd Derivative of codeine
AU666702B2 (en) 1992-01-23 1996-02-22 Toray Industries, Inc. Morphinan derivative and medicinal use
DE69414085T2 (de) * 1993-07-19 1999-03-18 Toray Industries, Inc., Tokio/Tokyo Wirkstoff zum schutze von gehirnzellen
AU686203B2 (en) * 1993-07-23 1998-02-05 Toray Industries, Inc. Morphinan derivative and medicinal use
US20060063792A1 (en) * 2004-09-17 2006-03-23 Adolor Corporation Substituted morphinans and methods of their use
MX2007015789A (es) 2005-06-16 2008-02-15 Mallinckrodt Inc Nueva ruta de sintesis para opiatos de 14-hidroxilo a traves de 1-halo-tebaina o analogos.
WO2015082932A1 (en) 2013-12-05 2015-06-11 The University Of Bath Novel opioid compounds and their uses

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3332950A (en) * 1963-03-23 1967-07-25 Endo Lab 14-hydroxydihydronormorphinone derivatives
IL26896A (en) * 1966-01-19 1970-11-30 Endo Lab 14 - Hydroxynormorphinins and 14 - Hydroxynormorphinones
BE788478A (fr) * 1971-09-08 1973-03-06 Bristol Myers Co Procede de preparation de composes analgesiques
US4017497A (en) * 1975-11-18 1977-04-12 Bristol-Myers Company Process for the preparation of 14-hydroxymorphinan derivatives

Also Published As

Publication number Publication date
IE46442B1 (en) 1983-06-15
ATA204378A (de) 1980-06-15
NL7803084A (nl) 1978-09-26
PL205497A1 (pl) 1979-06-04
IE780514L (en) 1978-09-23
DE2812581A1 (de) 1978-09-28
US4241067A (en) 1980-12-23
SU856381A3 (ru) 1981-08-15
CA1089455A (en) 1980-11-11
SE7803329L (sv) 1978-09-24
LU79295A1 (fr) 1979-10-29
GB1587831A (en) 1981-04-08
FR2384775B1 (ru) 1981-04-30
AT360664B (de) 1981-01-26
DD135081A5 (de) 1979-04-11
PL111722B1 (en) 1980-09-30
FR2384775A1 (fr) 1978-10-20
AU3435678A (en) 1979-09-27
IT7848545A0 (it) 1978-03-22
DK149753C (da) 1987-07-06
CS199522B2 (en) 1980-07-31
AR218296A1 (es) 1980-05-30
NZ186693A (en) 1979-10-25
ZA781525B (en) 1979-04-25
AU518614B2 (en) 1981-10-08
JPS53121798A (en) 1978-10-24
CH630629A5 (fr) 1982-06-30
DK129978A (da) 1978-09-24
ES468170A1 (es) 1979-01-01
SE436132B (sv) 1984-11-12
JPS6259112B2 (ru) 1987-12-09
IT1105172B (it) 1985-10-28
DK149753B (da) 1986-09-22
HU177722B (en) 1981-12-28

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: RECKITT & COLMAN PRODUCTS LTD

Effective date: 19930331