BE854268A - PYRROLIDONS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION - Google Patents
PYRROLIDONS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATIONInfo
- Publication number
- BE854268A BE854268A BE177278A BE177278A BE854268A BE 854268 A BE854268 A BE 854268A BE 177278 A BE177278 A BE 177278A BE 177278 A BE177278 A BE 177278A BE 854268 A BE854268 A BE 854268A
- Authority
- BE
- Belgium
- Prior art keywords
- pyrrolidons
- preparation process
- therapeutic application
- therapeutic
- application
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19762619638 DE2619638A1 (en) | 1976-05-04 | 1976-05-04 | PYRROLIDONE AND THE METHOD FOR MANUFACTURING THEIR |
Publications (1)
Publication Number | Publication Date |
---|---|
BE854268A true BE854268A (en) | 1977-11-04 |
Family
ID=5977020
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE177278A BE854268A (en) | 1976-05-04 | 1977-05-04 | PYRROLIDONS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
Country Status (9)
Country | Link |
---|---|
JP (1) | JPS52133975A (en) |
BE (1) | BE854268A (en) |
DE (1) | DE2619638A1 (en) |
DK (1) | DK194377A (en) |
ES (1) | ES458264A1 (en) |
FR (1) | FR2372806A1 (en) |
GB (1) | GB1583163A (en) |
IT (1) | IT1086223B (en) |
NL (1) | NL7704739A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4320136A (en) | 1980-08-11 | 1982-03-16 | E. I. Du Pont De Nemours And Company | 8-Aza-16,16-difluoroprostanoids |
WO2003074483A1 (en) | 2002-03-05 | 2003-09-12 | Ono Pharmaceutical Co., Ltd. | 8-azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4321201A (en) | 1980-09-22 | 1982-03-23 | E. I. Du Pont De Nemours And Company | Optically active tert-alkyl 7-(2-oxo-5-carbonyloxypyrrolidinyl) heptanoates |
EP0440789A1 (en) * | 1988-04-22 | 1991-08-14 | 2-i MOSKOVSKY GOSUDARSTVENNY MEDITSINSKY INSTITUT IMENI N.I. PIROGOVA | Carbalkoxymethyl ethers of lactam-1-acetic acid and method of obtaining them |
AU1293101A (en) | 1999-12-22 | 2001-07-03 | Pfizer Products Inc. | Ep4 receptor selective agonists in the treatment of osteoporosis |
WO2002024647A1 (en) * | 2000-09-21 | 2002-03-28 | Ono Pharmaceutical Co., Ltd. | Ep4 receptor agonists containing 8-azaprostaglandin derivatives as the active ingredient |
CA2429850C (en) * | 2000-11-27 | 2008-12-30 | Pfizer Products Inc. | Ep4 receptor selective agonists in the treatment of osteoporosis |
KR20040015364A (en) * | 2001-07-16 | 2004-02-18 | 에프. 호프만-라 로슈 아게 | Prostaglandin analogues as ep4 receptor agonists |
BR0211167A (en) | 2001-07-16 | 2004-08-10 | Hoffmann La Roche | 2-Pyrrolidone derivatives as prostanoid agonists |
MXPA04000757A (en) | 2001-07-23 | 2004-07-08 | Ono Pharmaceutical Co | Remedies for diseases with bone mass loss having ep4. |
EP1556347A4 (en) * | 2002-06-10 | 2006-08-09 | Applied Research Systems | Gamma lactams as prostaglandin agonists and use thereof |
CA2511255C (en) | 2003-01-10 | 2009-04-07 | F. Hoffmann-La Roche Ag | 2-piperidone derivatives as prostaglandin agonists |
WO2004065365A1 (en) * | 2003-01-21 | 2004-08-05 | Ono Pharmaceutical Co., Ltd. | 8-azaprostaglandin derivatives and medicinal uses thereof |
US7179820B2 (en) | 2003-06-06 | 2007-02-20 | Allergan, Inc. | Piperidinyl prostaglandin E analogs |
WO2006043655A1 (en) | 2004-10-22 | 2006-04-27 | Ono Pharmaceutical Co., Ltd. | Medicinal composition for inhalation |
CA2879506C (en) | 2012-07-19 | 2020-10-27 | Cayman Chemical Company, Inc. | Difluorolactam compositions for ep4-mediated osteo related diseases and conditions |
US9676712B2 (en) | 2013-03-15 | 2017-06-13 | Cayman Chemical Company, Inc. | Lactam compounds as EP4 receptor-selective agonists for use in the treatment of EP4-mediated diseases and conditions |
CA2903314C (en) | 2013-03-15 | 2023-02-14 | Cayman Chemical Company, Inc. | Methods of synthesizing a difluorolactam analog |
EA201591793A1 (en) * | 2013-03-15 | 2016-01-29 | Кайман Кемикал Компани, Инк. | LACTAM COMPOUNDS AS SELECTIVE AGONISTS OF EP4 RECEPTORS FOR USE IN THE TREATMENT OF EP4-MEDIATED DISEASES AND STATES |
EP3021879A2 (en) | 2013-07-19 | 2016-05-25 | Cayman Chemical Company, Incorporated | Methods, systems, and compositions for promoting bone growth |
-
1976
- 1976-05-04 DE DE19762619638 patent/DE2619638A1/en active Pending
-
1977
- 1977-04-28 ES ES458264A patent/ES458264A1/en not_active Expired
- 1977-04-29 NL NL7704739A patent/NL7704739A/en not_active Application Discontinuation
- 1977-05-02 IT IT23096/77A patent/IT1086223B/en active
- 1977-05-03 GB GB18427/77A patent/GB1583163A/en not_active Expired
- 1977-05-03 DK DK194377A patent/DK194377A/en unknown
- 1977-05-04 BE BE177278A patent/BE854268A/en unknown
- 1977-05-04 FR FR7713518A patent/FR2372806A1/en active Granted
- 1977-05-04 JP JP5194577A patent/JPS52133975A/en active Pending
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4320136A (en) | 1980-08-11 | 1982-03-16 | E. I. Du Pont De Nemours And Company | 8-Aza-16,16-difluoroprostanoids |
WO2003074483A1 (en) | 2002-03-05 | 2003-09-12 | Ono Pharmaceutical Co., Ltd. | 8-azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient |
Also Published As
Publication number | Publication date |
---|---|
JPS52133975A (en) | 1977-11-09 |
FR2372806A1 (en) | 1978-06-30 |
DE2619638A1 (en) | 1977-11-17 |
IT1086223B (en) | 1985-05-28 |
ES458264A1 (en) | 1978-07-16 |
DK194377A (en) | 1977-11-05 |
FR2372806B1 (en) | 1980-02-29 |
NL7704739A (en) | 1977-11-08 |
GB1583163A (en) | 1981-01-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
LU80081A1 (en) | NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE878723A (en) | 4-ANILINOQUINAZOLINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
FR2383157B1 (en) | CHALCON DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE867421A (en) | MEVALONOLACTONE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
FR2393795B1 (en) | CARBOSTYRYL DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATIONS | |
FR2340950A1 (en) | CEFUROXIME ESTERS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE854268A (en) | PYRROLIDONS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE851893A (en) | NEW ARYL-3 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE846452A (en) | NEW PYRIMIDONS, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE847090A (en) | 15-STEROIDS, AND THEIR PREPARATION PROCESS | |
FR2458547B2 (en) | NOVEL AZOLONES N-ARYLE, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE864312A (en) | NEW PYRROLIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
FR2349587A1 (en) | 1,3-DIHYDRO-HETEROARYLSPIRO (ISOBENZOFURANNES), THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE865805A (en) | 1,2,3-THIADIAZOL-3-IN-5-YLIDENE-UREES, THEIR PREPARATION PROCESS AND THEIR USE | |
FR2351965A1 (en) | BENZENESULFONYLUREES, THEIR PROCESS FOR PREPARATION AND THEIR THERAPEUTIC APPLICATION | |
LU79606A1 (en) | BISAMIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
FR2353520A1 (en) | 1-ARYLOXY-2-HYDROXY-3-AMINOPROPANES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATIONS | |
BE866928A (en) | BENZENE-SULFONYL UREES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
LU78873A1 (en) | ALKYLTHIO-7,8-DIHYDROXY-1-PHENYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINES, THEIR PREPARATION PROCESS AND THERAPEUTIC APPLICATION | |
FR2351098A1 (en) | ISOTHIOUREA DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE860773A (en) | MONOCYCLIC BETA-LACTAMES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE868659A (en) | NEW BENZAMIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATIONS | |
BE835828A (en) | NEW 1,4-BENZODIOXANES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION | |
BE866648A (en) | TRIAZOLOTHIADIAZINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATIONS | |
FR2340951A1 (en) | CEFUROXIME DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |