BE798677A - Derives de benzodiazepine, leur preparation et leurs applications - Google Patents

Derives de benzodiazepine, leur preparation et leurs applications

Info

Publication number
BE798677A
BE798677A BE130386A BE130386A BE798677A BE 798677 A BE798677 A BE 798677A BE 130386 A BE130386 A BE 130386A BE 130386 A BE130386 A BE 130386A BE 798677 A BE798677 A BE 798677A
Authority
BE
Belgium
Prior art keywords
applications
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
BE130386A
Other languages
English (en)
Original Assignee
Centre Etd Ind Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centre Etd Ind Pharma filed Critical Centre Etd Ind Pharma
Publication of BE798677A publication Critical patent/BE798677A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BE130386A 1972-05-05 1973-04-25 Derives de benzodiazepine, leur preparation et leurs applications BE798677A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB2114172 1972-05-05
CH581473A CH571001A5 (fr) 1972-05-05 1973-04-24

Publications (1)

Publication Number Publication Date
BE798677A true BE798677A (fr) 1973-08-16

Family

ID=25698412

Family Applications (1)

Application Number Title Priority Date Filing Date
BE130386A BE798677A (fr) 1972-05-05 1973-04-25 Derives de benzodiazepine, leur preparation et leurs applications

Country Status (6)

Country Link
JP (1) JPS4947391A (fr)
BE (1) BE798677A (fr)
CA (1) CA999860A (fr)
CH (1) CH571001A5 (fr)
DE (1) DE2321705A1 (fr)
FR (1) FR2183716A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0518484A3 (en) * 1991-05-14 1993-03-17 Merck & Co. Inc. 1,4-benzodiazepines condesed with 5- and 6-membered heterocyclic rings to treat anxiety, pain, pupil constriction, withdrawal-syndrome or oncologic disorders

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
DE2547652A1 (de) * 1974-11-15 1976-05-20 Upjohn Co Pharmazeutische zubereitung
US4044142A (en) 1975-02-03 1977-08-23 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
US4134976A (en) * 1975-02-15 1979-01-16 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
AT361486B (de) * 1975-08-07 1981-03-10 Hoffmann La Roche Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen
US4185102A (en) 1975-11-04 1980-01-22 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
JPS60202096A (ja) * 1984-03-22 1985-10-12 日産自動車株式会社 フオ−クリフトのフオ−ク移動装置
DE3610848A1 (de) * 1986-04-01 1987-10-15 Boehringer Ingelheim Kg Neue 1,4-diazepine
YU136287A (en) * 1986-07-25 1990-06-30 Boehringer Kg Process for preparing new 1,4 benzodiazepines
AU6909194A (en) * 1993-05-14 1994-12-12 Board Of Regents, The University Of Texas System Preparation of n-cyanodithioimino-carbonates and 3-mercapto-5-amino-1h-1,2,4-triazole
US7160880B1 (en) 1999-05-14 2007-01-09 Cenes Limited Short-acting benzodiazepines
GB9911152D0 (en) * 1999-05-14 1999-07-14 Glaxo Group Ltd Short-acting benzodiazepines
CN104059071B (zh) 2006-07-10 2016-06-22 Paion英国有限公司 短效苯并二氮杂*盐及其多晶型
EP2450039A1 (fr) 2010-11-08 2012-05-09 PAION UK Ltd. Régime de dosage permettant la sédation avec CNS 7056 (Remimazolam)
CN108033964B (zh) 2017-12-28 2021-02-09 杭州奥默医药股份有限公司 一种吡啶基咪唑并苯并二氮杂卓丙酸酯化合物及其合成和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE787251A (fr) * 1971-08-04 1973-02-05 Upjohn Co Nouvelles benzodiazepines et leur preparation

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0518484A3 (en) * 1991-05-14 1993-03-17 Merck & Co. Inc. 1,4-benzodiazepines condesed with 5- and 6-membered heterocyclic rings to treat anxiety, pain, pupil constriction, withdrawal-syndrome or oncologic disorders

Also Published As

Publication number Publication date
CA999860A (en) 1976-11-16
CH571001A5 (fr) 1975-12-31
FR2183716A1 (en) 1973-12-21
DE2321705A1 (de) 1973-11-15
JPS4947391A (fr) 1974-05-08
FR2183716B1 (fr) 1976-12-03

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