AU7732691A - Hiv protease inhibitors and processes for their preparation - Google Patents

Hiv protease inhibitors and processes for their preparation

Info

Publication number: AU7732691A
Authority: AU; Australia
Prior art keywords: processes; preparation; protease inhibitors; hiv protease; hiv
Prior art date: 1990-06-01
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU77326/91A

Inventor

Not Given Name

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novartis AG

Original Assignee

Ciba Geigy AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-06-01

Filing date

1991-05-24

Publication date

1991-12-05

1991-05-24 Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG

1991-12-05 Publication of AU7732691A publication Critical patent/AU7732691A/en

Status Abandoned legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K17/00—Carrier-bound or immobilised peptides; Preparation thereof
- C07K17/02—Peptides being immobilised on, or in, an organic carrier
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0207—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

AU77326/91A 1990-06-01 1991-05-24 Hiv protease inhibitors and processes for their preparation Abandoned AU7732691A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH1860/90		1990-06-01
CH186090		1990-06-01

Publications (1)

Publication Number	Publication Date
AU7732691A true AU7732691A (en)	1991-12-05

Family

ID=4220305

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU77326/91A Abandoned AU7732691A (en)	1990-06-01	1991-05-24	Hiv protease inhibitors and processes for their preparation

Country Status (9)

Country	Link
EP (1)	EP0459465A3 (en)
JP (1)	JPH04235999A (en)
KR (1)	KR920000790A (en)
AU (1)	AU7732691A (en)
CA (1)	CA2043603A1 (en)
IE (1)	IE911873A1 (en)
IL (1)	IL98260A0 (en)
PT (1)	PT97782A (en)
ZA (1)	ZA914136B (en)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1995007269A1 (en) *	1993-09-10	1995-03-16	Narhex Limited	Polar-substituted hydrocarbons
US5679688A (en) *	1992-03-11	1997-10-21	Narhex Limited	Quinaldoyl-amine derivatives of oxo-and hydroxy-substituted hydrocarbons
US5888992A (en) *	1992-03-11	1999-03-30	Narhex Limited	Polar substituted hydrocarbons
US6071895A (en) *	1992-03-11	2000-06-06	Narhex Limited	Polar-substituted hydrocarbons
US6258806B1 (en)	1992-03-11	2001-07-10	Narhex Limited	Amine derivatives of oxo- and hydroxy- substituted hydrocarbons

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5643878A (en) *	1991-09-12	1997-07-01	Ciba-Geigy Corporation	5-amino-4-hydroxyhexanoic acid derivatives
TW217410B (en) *	1992-04-01	1993-12-11	Ciba Geigy
DE4215874A1 (en) *	1992-05-14	1993-11-18	Bayer Ag	Dithiolanylglycine-containing HIV protease inhibitors of the hydroxyethylene isostear type
US5559256A (en) *	1992-07-20	1996-09-24	E. R. Squibb & Sons, Inc.	Aminediol protease inhibitors
EP0626178A1 (en) *	1993-05-17	1994-11-30	Ciba-Geigy Ag	Use of inhibitors of HIV-protease for the treatment of tumorous diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4727060A (en) *	1984-11-13	1988-02-23	Ciba-Geigy Corporation	Novel 5-amino-4-hydroxyvaleryl derivatives
EP0374097A3 (en) *	1988-12-15	1991-06-12	Ciba-Geigy Ag	Use of peptide isosteres as retroviral protease inhibitors
EP0374098A3 (en) *	1988-12-15	1991-05-02	Ciba-Geigy Ag	Inhibitors of retroviral proteases

1991
- 1991-05-24 AU AU77326/91A patent/AU7732691A/en not_active Abandoned
- 1991-05-24 IL IL98260A patent/IL98260A0/en unknown
- 1991-05-29 PT PT97782A patent/PT97782A/en not_active Application Discontinuation
- 1991-05-29 EP EP19910108828 patent/EP0459465A3/en not_active Withdrawn
- 1991-05-30 ZA ZA914136A patent/ZA914136B/en unknown
- 1991-05-30 CA CA002043603A patent/CA2043603A1/en not_active Abandoned
- 1991-05-31 KR KR1019910009007A patent/KR920000790A/en not_active Application Discontinuation
- 1991-05-31 IE IE187391A patent/IE911873A1/en unknown
- 1991-06-01 JP JP3130116A patent/JPH04235999A/en active Pending

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5679688A (en) *	1992-03-11	1997-10-21	Narhex Limited	Quinaldoyl-amine derivatives of oxo-and hydroxy-substituted hydrocarbons
US5888992A (en) *	1992-03-11	1999-03-30	Narhex Limited	Polar substituted hydrocarbons
US5942504A (en) *	1992-03-11	1999-08-24	Narhex Limited	Amine derivatives of oxo- and hydroxy- substituted hydrocarbons
US6071895A (en) *	1992-03-11	2000-06-06	Narhex Limited	Polar-substituted hydrocarbons
US6258806B1 (en)	1992-03-11	2001-07-10	Narhex Limited	Amine derivatives of oxo- and hydroxy- substituted hydrocarbons
WO1995007269A1 (en) *	1993-09-10	1995-03-16	Narhex Limited	Polar-substituted hydrocarbons

Also Published As

Publication number	Publication date
IE911873A1 (en)	1991-12-04
CA2043603A1 (en)	1991-12-02
KR920000790A (en)	1992-01-29
ZA914136B (en)	1992-02-26
EP0459465A3 (en)	1992-12-23
IL98260A0 (en)	1992-06-21
PT97782A (en)	1992-02-28
EP0459465A2 (en)	1991-12-04
JPH04235999A (en)	1992-08-25

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