AU7329394A - A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library - Google Patents

A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library

Info

Publication number
AU7329394A
AU7329394A AU73293/94A AU7329394A AU7329394A AU 7329394 A AU7329394 A AU 7329394A AU 73293/94 A AU73293/94 A AU 73293/94A AU 7329394 A AU7329394 A AU 7329394A AU 7329394 A AU7329394 A AU 7329394A
Authority
AU
Australia
Prior art keywords
preparing
pharmaceutically useful
peptide compounds
useful non
structurally diverse
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU73293/94A
Inventor
David Garry Hangauer Jr.
Mark Edward Hediger
Michael Raymond Pavia
George Mcclelland Whitesides
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Sphinx Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sphinx Pharmaceuticals Corp filed Critical Sphinx Pharmaceuticals Corp
Publication of AU7329394A publication Critical patent/AU7329394A/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/04Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
    • C07C279/08Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/21Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
    • C07C65/24Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
AU73293/94A 1993-08-03 1994-07-07 A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library Abandoned AU7329394A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US10107493A 1993-08-03 1993-08-03
US101074 1993-08-03
US23954294A 1994-05-08 1994-05-08
US239542 1994-05-08
PCT/US1994/007780 WO1995004277A1 (en) 1993-08-03 1994-07-07 A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library

Publications (1)

Publication Number Publication Date
AU7329394A true AU7329394A (en) 1995-02-28

Family

ID=26797874

Family Applications (1)

Application Number Title Priority Date Filing Date
AU73293/94A Abandoned AU7329394A (en) 1993-08-03 1994-07-07 A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library

Country Status (6)

Country Link
EP (1) EP0712493A4 (en)
JP (1) JPH09504511A (en)
AU (1) AU7329394A (en)
CA (1) CA2168886A1 (en)
PE (1) PE14895A1 (en)
WO (1) WO1995004277A1 (en)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5811241A (en) * 1995-09-13 1998-09-22 Cortech, Inc. Method for preparing and identifying N-substitued 1,4-piperazines and N-substituted 1,4-piperazinediones
US5874443A (en) * 1995-10-19 1999-02-23 Trega Biosciences, Inc. Isoquinoline derivatives and isoquinoline combinatorial libraries
US5840500A (en) * 1996-07-11 1998-11-24 Trega Biosciences, Inc. Quinoline derivatives and quinoline combinatorial libraries
GB9616563D0 (en) * 1996-08-07 1996-09-25 Oxford Asymmetry Ltd Compounds and methods
US5916899A (en) * 1996-10-18 1999-06-29 Trega Biosciences, Inc. Isoquinoline derivatives and isoquinoline combinatorial libraries
US6893815B1 (en) * 1997-06-30 2005-05-17 Isis Pharmaceuticals, Inc. Nucleobase heterocyclic combinatorialization
US6080587A (en) * 1998-01-23 2000-06-27 Eli Lilly And Company Method for preparing and selecting pharmaceutically useful sulfur-bridged bi- and triaromatic ring compounds from a structurally diverse universal library
US6127381A (en) * 1998-04-28 2000-10-03 Basu; Amaresh Isoquinoline compound melanocortin receptor ligands and methods of using same
US6534503B1 (en) 1998-04-28 2003-03-18 Lion Bioscience Ag Melanocortin receptor-3 ligands to treat sexual dysfunction
US6284735B1 (en) 1998-04-28 2001-09-04 Lion Bioscience Ag HP-3228 and related peptides to treat sexual dysfunction
CA2319730A1 (en) * 1998-06-08 1999-12-16 Advanced Medicine, Inc. Bradykinin antagonists
US20040009535A1 (en) 1998-11-27 2004-01-15 Celltech R&D, Inc. Compositions and methods for increasing bone mineralization
CN101469329B (en) 1998-11-27 2012-10-24 达尔文发现有限公司 Compositions and methods for increasing bone mineralization
CA2368026A1 (en) * 1999-03-22 2000-09-28 Bi-Huang Hu Oxazole and thiazole combinatorial libraries
US6864235B1 (en) 1999-04-01 2005-03-08 Eva A. Turley Compositions and methods for treating cellular response to injury and other proliferating cell disorders regulated by hyaladherin and hyaluronans
US6911429B2 (en) 1999-04-01 2005-06-28 Transition Therapeutics Inc. Compositions and methods for treating cellular response to injury and other proliferating cell disorders regulated by hyaladherin and hyaluronans
US7507542B2 (en) 2001-05-08 2009-03-24 Ucb Sa Method for regulating immune function using the FOXP3 protein
WO2004009531A1 (en) * 2002-07-24 2004-01-29 Janssen Pharmaceutica N.V. Acetylenic compounds useful in treating inflammatory disorders
ATE481422T1 (en) 2002-11-21 2010-10-15 Celltech R & D Inc MODULATING IMMUNE RESPONSES
US7022703B2 (en) 2003-07-24 2006-04-04 Janssen Pharmaceutica, N.V. Acetylenic compound useful in treating inflammatory disorders
EP2257536A4 (en) 2008-02-14 2011-03-23 Amira Pharmaceuticals Inc Cyclic diaryl ether as antagonists of prostaglandin d2 receptors
JP2011518130A (en) 2008-04-02 2011-06-23 アミラ ファーマシューティカルズ,インク. Aminoalkylphenyl antagonist of prostaglandin D2 receptor
WO2010057118A2 (en) 2008-11-17 2010-05-20 Amira Pharmaceuticals, Inc. Heterocyclic antagonists of prostaglandin d2 receptors
GB0903482D0 (en) * 2009-02-27 2009-04-08 Ucl Business Plc New compounds
CA3217862A1 (en) 2021-05-05 2022-11-10 Radius Pharmaceuticals, Inc. Animal model having homologous recombination of mouse pth1 receptor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5218124A (en) * 1989-10-27 1993-06-08 American Home Products Corporation Substituted benzoylbenzene-, biphenyl- and 2-oxazole-alkanoic acid derivatives as inhibitors of pla2 and lipoxygenase
US5250548A (en) * 1990-09-10 1993-10-05 Abbott Laboratories Angiotensin II receptor antagonists

Also Published As

Publication number Publication date
CA2168886A1 (en) 1995-02-09
JPH09504511A (en) 1997-05-06
EP0712493A4 (en) 1997-01-15
WO1995004277A1 (en) 1995-02-09
EP0712493A1 (en) 1996-05-22
PE14895A1 (en) 1995-06-08

Similar Documents

Publication Publication Date Title
AU7329394A (en) A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library
AU5961794A (en) A rapid tree-based method for vector quantization
AU1426095A (en) New ginkgolide derivatives and a process for preparing them
AU7171894A (en) A process stabilizing process controller
AU7875494A (en) Method for inhibiting angiogenesis
AU9320898A (en) Methods for searching a knowledge base
AU4985193A (en) Method and system for assembling a wall
AU6406794A (en) System for positioning a workpoint
AU6518694A (en) A process for preparing halogenated isothiazoles
AU3214693A (en) Apparatus for partitioning a storage space
AU7122394A (en) A vibration-compensating apparatus for counteracting vibrations
AU5746694A (en) Mechanical lockout for a pneumatic tool
AU6847194A (en) Equipment for handling drill rods
AU6388094A (en) A method for cascading of microbases
AU3369093A (en) Locking apparatus for a string
AU7424594A (en) Method for preparing 3-aminopyridines from 3-nitropyridines
AU7122294A (en) A dual vibration-compensating apparatus
AU1384795A (en) Process for preparing carbamates
GB9317491D0 (en) New compound and a process for preparation thereof
AU7058498A (en) Method for the preparation of a chemical library
AU5096293A (en) A process for preparing dinitrotoluene
AU4815493A (en) A method for classifying a client
AU7723994A (en) Apparatus for remote implementation of a command
ZA945731B (en) Method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library
AU6414494A (en) Method for supporting a transportation surface