AU7073296A - 5,6,7,8-tetrahydropyrido{2,3-d}pyrimidines - Google Patents

5,6,7,8-tetrahydropyrido{2,3-d}pyrimidines

Info

Publication number
AU7073296A
AU7073296A AU70732/96A AU7073296A AU7073296A AU 7073296 A AU7073296 A AU 7073296A AU 70732/96 A AU70732/96 A AU 70732/96A AU 7073296 A AU7073296 A AU 7073296A AU 7073296 A AU7073296 A AU 7073296A
Authority
AU
Australia
Prior art keywords
tetrahydropyrido
pyrimidines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU70732/96A
Inventor
Lynn S. Gossett
Koo Lee
Chuan Shih
Edward C. Taylor
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Princeton University
Original Assignee
Eli Lilly and Co
Princeton University
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co, Princeton University filed Critical Eli Lilly and Co
Publication of AU7073296A publication Critical patent/AU7073296A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU70732/96A 1996-05-01 1996-09-17 5,6,7,8-tetrahydropyrido{2,3-d}pyrimidines Abandoned AU7073296A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US2117496P 1996-05-01 1996-05-01
US64066996A 1996-05-01 1996-05-01
US60021174 1996-05-01
US08640669 1996-05-01
PCT/US1996/014822 WO1997041115A1 (en) 1996-05-01 1996-09-17 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES

Publications (1)

Publication Number Publication Date
AU7073296A true AU7073296A (en) 1997-11-19

Family

ID=26694360

Family Applications (1)

Application Number Title Priority Date Filing Date
AU70732/96A Abandoned AU7073296A (en) 1996-05-01 1996-09-17 5,6,7,8-tetrahydropyrido{2,3-d}pyrimidines

Country Status (5)

Country Link
EP (1) EP0904271A4 (en)
JP (1) JP2001524927A (en)
AU (1) AU7073296A (en)
CA (1) CA2251813A1 (en)
WO (1) WO1997041115A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004113337A1 (en) * 2003-06-25 2004-12-29 Pfizer Inc. Convergent synthesis of a garft inhibitor containing a methyl substitute thiophene core and a tetrahydropyrido`2,3-d! pyrimidine ring system and intermediates therefor
US7488747B2 (en) * 2003-12-29 2009-02-10 Sepracor Inc. Pyrrole and pyrazole DAAO inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4895946A (en) * 1987-10-26 1990-01-23 The Trustees Of Princeton University Process for the preparation of fused pyridine compounds
DK172753B1 (en) * 1988-05-25 1999-06-28 Lilly Co Eli N- (5,6,7,8-tetrahydropyrido [2,3-d] pyrimidin-6-yl-alkanoyl) -glutamic acid derivatives, their use, pharmaceutical preparations
US5008391A (en) * 1989-07-07 1991-04-16 Eli Lilly And Company Enantioselective synthesis of antifolates
US5508281A (en) * 1991-04-08 1996-04-16 Duquesne University Of The Holy Ghost Derivatives of pyrido [2,3-d] and [3,2-d] pyrimidine and methods of using these derivatives
US5354751A (en) * 1992-03-03 1994-10-11 Sri International Heteroaroyl 10-deazaamino-pterine compounds and use for rheumatoid arthritis
US5536724A (en) * 1992-03-03 1996-07-16 Sri International Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins

Also Published As

Publication number Publication date
EP0904271A4 (en) 2002-01-23
JP2001524927A (en) 2001-12-04
WO1997041115A1 (en) 1997-11-06
CA2251813A1 (en) 1997-11-06
EP0904271A1 (en) 1999-03-31

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