AU6850787A - Process for acylating amines with 2-benzothiazolyl thioesters of carboxylic acids - Google Patents

Process for acylating amines with 2-benzothiazolyl thioesters of carboxylic acids

Info

Publication number
AU6850787A
AU6850787A AU68507/87A AU6850787A AU6850787A AU 6850787 A AU6850787 A AU 6850787A AU 68507/87 A AU68507/87 A AU 68507/87A AU 6850787 A AU6850787 A AU 6850787A AU 6850787 A AU6850787 A AU 6850787A
Authority
AU
Australia
Prior art keywords
carboxylic acids
thioesters
benzothiazolyl
acylating amines
acylating
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU68507/87A
Other versions
AU605754B2 (en
Inventor
Andre Furlenmeier
Urs Weiss
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of AU6850787A publication Critical patent/AU6850787A/en
Application granted granted Critical
Publication of AU605754B2 publication Critical patent/AU605754B2/en
Assigned to F. HOFFMANN-LA ROCHE AG reassignment F. HOFFMANN-LA ROCHE AG Alteration of Name(s) in Register under S187 Assignors: F. HOFFMANN-LA ROCHE AG
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/70—Sulfur atoms
    • C07D277/74—Sulfur atoms substituted by carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU68507/87A 1986-02-07 1987-02-04 Process for acylating amines with 2-benzothiazolyl thioesters of carboxylic acids Ceased AU605754B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH48786 1986-02-07
CH487/86 1986-02-07

Publications (2)

Publication Number Publication Date
AU6850787A true AU6850787A (en) 1987-08-13
AU605754B2 AU605754B2 (en) 1991-01-24

Family

ID=4188132

Family Applications (1)

Application Number Title Priority Date Filing Date
AU68507/87A Ceased AU605754B2 (en) 1986-02-07 1987-02-04 Process for acylating amines with 2-benzothiazolyl thioesters of carboxylic acids

Country Status (20)

Country Link
EP (1) EP0231845B1 (en)
JP (1) JPH0745411B2 (en)
KR (1) KR940009793B1 (en)
CN (1) CN1019300B (en)
AR (1) AR243529A1 (en)
AT (1) ATE77378T1 (en)
AU (1) AU605754B2 (en)
CA (1) CA1339312C (en)
DE (1) DE3779768D1 (en)
DK (1) DK53787A (en)
ES (1) ES2042507T3 (en)
FI (1) FI88391C (en)
GR (1) GR3005744T3 (en)
HU (1) HU201767B (en)
IE (1) IE59862B1 (en)
IL (1) IL81457A (en)
NO (1) NO169231C (en)
PH (1) PH24285A (en)
PT (1) PT84254B (en)
ZA (1) ZA87745B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT402928B (en) * 1994-12-23 1997-09-25 Biochemie Gmbh NEW METHOD FOR PRODUCING CEFOTAXIM
AT406773B (en) * 1998-04-02 2000-08-25 Biochemie Gmbh NEW SALT OF 7- (2- (AMINOTHIAZOL-4YL) -2-
KR100777450B1 (en) 2005-05-28 2007-11-21 삼성전자주식회사 Encoder Speed Correction Method and System thereof
WO2011042775A1 (en) * 2009-10-09 2011-04-14 Nectar Lifesciences Ltd. Process for preparation of cefotaxime acid
CN101792456A (en) * 2010-03-11 2010-08-04 池州东升药业有限公司 Preparation method of cefetamet pivoxil hydrochloride
CN102093151B (en) * 2011-01-13 2013-04-24 武汉大学 Method for synthesizing amide compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3165922D1 (en) * 1980-03-28 1984-10-18 Biochemie Gmbh New process for the production of cephalosporin antibiotics, and novel intermediates used in such process and their production
EP0075104A3 (en) * 1981-09-23 1984-11-28 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Cephalosporin derivatives, process for their preparation, pharmaceutical compositions containing them and intermediates
EP0115770B2 (en) * 1983-01-07 1996-06-19 Takeda Chemical Industries, Ltd. Thiazole Derivatives
WO1985004659A1 (en) * 1984-04-10 1985-10-24 Biochemie Gesellschaft M.B.H. Intermediary products of cephalosporine, preparation process thereof and utilization thereof
DE3585154D1 (en) * 1984-11-15 1992-02-20 Hoffmann La Roche METHOD FOR PRODUCING CEPHALOSPORINE ESTERS.
AT383810B (en) * 1985-11-20 1987-08-25 Biochemie Gmbh METHOD FOR PRODUCING CEPHALOSPORINE DERIVATIVES

Also Published As

Publication number Publication date
EP0231845B1 (en) 1992-06-17
NO169231B (en) 1992-02-17
DK53787D0 (en) 1987-02-02
FI870446A (en) 1987-08-08
PH24285A (en) 1990-05-29
ZA87745B (en) 1987-09-30
DK53787A (en) 1987-08-08
AU605754B2 (en) 1991-01-24
CN1019300B (en) 1992-12-02
ES2042507T3 (en) 1993-12-16
GR3005744T3 (en) 1993-06-07
CN87100860A (en) 1987-08-26
AR243529A1 (en) 1993-08-31
JPS6372692A (en) 1988-04-02
FI88391B (en) 1993-01-29
ATE77378T1 (en) 1992-07-15
IE870317L (en) 1987-08-07
NO870482L (en) 1987-08-10
KR940009793B1 (en) 1994-10-17
CA1339312C (en) 1997-08-19
KR870007939A (en) 1987-09-23
PT84254A (en) 1987-03-01
EP0231845A3 (en) 1989-03-15
IL81457A (en) 1992-03-29
NO870482D0 (en) 1987-02-06
HU201767B (en) 1990-12-28
IL81457A0 (en) 1987-09-16
FI88391C (en) 1993-05-10
IE59862B1 (en) 1994-04-20
HUT46328A (en) 1988-10-28
JPH0745411B2 (en) 1995-05-17
PT84254B (en) 1989-09-14
FI870446A0 (en) 1987-02-02
NO169231C (en) 1992-05-27
EP0231845A2 (en) 1987-08-12
DE3779768D1 (en) 1992-07-23

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired