AU6339599A - Quinoline derivatives and their use as antibacterial agents - Google Patents
Quinoline derivatives and their use as antibacterial agentsInfo
- Publication number
- AU6339599A AU6339599A AU63395/99A AU6339599A AU6339599A AU 6339599 A AU6339599 A AU 6339599A AU 63395/99 A AU63395/99 A AU 63395/99A AU 6339599 A AU6339599 A AU 6339599A AU 6339599 A AU6339599 A AU 6339599A
- Authority
- AU
- Australia
- Prior art keywords
- antibacterial agents
- quinoline derivatives
- derivatives
- quinoline
- mammals
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Abstract
Piperidine derivatives and pharmaceutical derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9822440.5A GB9822440D0 (en) | 1998-10-14 | 1998-10-14 | Medicaments |
GB9822440 | 1998-10-14 | ||
PCT/EP1999/007766 WO2000021952A1 (en) | 1998-10-14 | 1999-10-11 | Quinoline derivatives and their use as antibacterial agents |
Publications (1)
Publication Number | Publication Date |
---|---|
AU6339599A true AU6339599A (en) | 2000-05-01 |
Family
ID=10840577
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU63395/99A Abandoned AU6339599A (en) | 1998-10-14 | 1999-10-11 | Quinoline derivatives and their use as antibacterial agents |
Country Status (11)
Country | Link |
---|---|
US (1) | US6602882B1 (en) |
EP (1) | EP1121355B1 (en) |
JP (1) | JP2002527434A (en) |
AT (1) | ATE312831T1 (en) |
AU (1) | AU6339599A (en) |
DE (1) | DE69928952T2 (en) |
ES (1) | ES2255306T3 (en) |
GB (1) | GB9822440D0 (en) |
MA (1) | MA25009A1 (en) |
PE (1) | PE20001112A1 (en) |
WO (1) | WO2000021952A1 (en) |
Families Citing this family (47)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69840599D1 (en) | 1997-09-15 | 2009-04-09 | Procter & Gamble | ANTIMICROBIAL CHINOLONE, ITS COMPOSITIONS, AND ITS USES |
GB9822450D0 (en) * | 1998-10-14 | 1998-12-09 | Smithkline Beecham Plc | Medicaments |
GB9914486D0 (en) * | 1999-06-21 | 1999-08-18 | Smithkline Beecham Plc | Medicaments |
GB9917406D0 (en) * | 1999-07-23 | 1999-09-22 | Smithkline Beecham Plc | Compounds |
GB9917408D0 (en) * | 1999-07-23 | 1999-09-22 | Smithkline Beecham Plc | Compounds |
SE9902987D0 (en) | 1999-08-24 | 1999-08-24 | Astra Pharma Prod | Novel compounds |
US6803369B1 (en) | 2000-07-25 | 2004-10-12 | Smithkline Beecham Corporation | Compounds and methods for the treatment of neoplastic disease |
DE60125373T2 (en) | 2000-07-26 | 2007-10-18 | Smithkline Beecham P.L.C., Brentford | AMINOPIPERIDINE CHINOLINE AND ITS AZAISOSTERIC ANALOGUE WITH ANTIBACTERIAL EFFECT |
JP2004509885A (en) * | 2000-09-21 | 2004-04-02 | スミスクライン ビーチャム パブリック リミテッド カンパニー | Quinoline derivatives as antibacterial agents |
GB0031088D0 (en) * | 2000-12-20 | 2001-01-31 | Smithkline Beecham Plc | Medicaments |
GB0031086D0 (en) * | 2000-12-20 | 2001-01-31 | Smithkline Beecham Plc | Medicaments |
GB0101577D0 (en) * | 2001-01-22 | 2001-03-07 | Smithkline Beecham Plc | Compounds |
GB0104050D0 (en) | 2001-02-19 | 2001-04-04 | Astrazeneca Ab | Chemical compounds |
GB0107228D0 (en) | 2001-03-22 | 2001-05-16 | Astrazeneca Ab | Chemical compounds |
GB0112836D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
GB0112834D0 (en) * | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
GB0118238D0 (en) * | 2001-07-26 | 2001-09-19 | Smithkline Beecham Plc | Medicaments |
US20050119302A1 (en) * | 2001-10-30 | 2005-06-02 | Rahme Laurence G. | Methods for the prevention or treament of bacterial and fungal infections |
SE0103818D0 (en) | 2001-11-15 | 2001-11-15 | Astrazeneca Ab | Chemical compounds |
EP2181996A1 (en) | 2002-01-29 | 2010-05-05 | Glaxo Group Limited | Aminopiperidine derivatives |
WO2003064431A2 (en) * | 2002-01-29 | 2003-08-07 | Glaxo Group Limited | Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them |
AR040335A1 (en) * | 2002-06-26 | 2005-03-30 | Glaxo Group Ltd | CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND |
AR040336A1 (en) | 2002-06-26 | 2005-03-30 | Glaxo Group Ltd | PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND |
US6900224B2 (en) | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
JP4704755B2 (en) | 2002-11-05 | 2011-06-22 | グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー | Antibacterial agent |
DE60334016D1 (en) | 2002-11-05 | 2010-10-14 | Glaxo Group Ltd | ANTIBACTERIAL AGENTS |
EP1567520B1 (en) | 2002-12-04 | 2008-10-15 | Glaxo Group Limited | Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents |
AR042486A1 (en) * | 2002-12-18 | 2005-06-22 | Glaxo Group Ltd | QUINOLINE AND NAFTIRIDINE COMPOSITE HALOSUSTITUDED IN POSITION 3, PROCEDURE TO PREPARE THE COMPOUND, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND ITS USE TO PREPARE SUCH COMPOSITION. |
ATE440835T1 (en) * | 2003-03-06 | 2009-09-15 | Glaxo Group Ltd | HETEROCYCLIC UREA DERIVATIVES FOR THE TREATMENT OF PAIN. |
US7514562B2 (en) * | 2003-03-07 | 2009-04-07 | Glaxo Group Limited | Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain |
GB0305426D0 (en) * | 2003-03-08 | 2003-04-16 | Glaxo Group Ltd | Novel compounds |
FR2867472B1 (en) * | 2004-03-12 | 2008-07-18 | Aventis Pharma Sa | QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
US20070254872A1 (en) * | 2004-07-08 | 2007-11-01 | Glaxo Group Limited | Antibacterial Agents |
EP1846418A4 (en) | 2005-01-25 | 2009-12-23 | Glaxo Group Ltd | Antibacterial agents |
WO2006081178A2 (en) * | 2005-01-25 | 2006-08-03 | Glaxo Group Limited | Antibacterial agents |
JP2008528604A (en) | 2005-01-25 | 2008-07-31 | グラクソ グループ リミテッド | Antibacterial agent |
JP2008528587A (en) | 2005-01-25 | 2008-07-31 | グラクソ グループ リミテッド | Antibacterial agent |
US7605169B2 (en) | 2005-01-25 | 2009-10-20 | Glaxo Group Limited | Antibacterial agents |
MX2007012234A (en) | 2005-03-31 | 2008-03-18 | Johnson & Johnson | Bicyclic pyrazole compounds as antibacterial agents. |
MY150958A (en) | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
CA2635126A1 (en) | 2006-01-26 | 2007-08-02 | Actelion Pharmaceuticals Ltd | Tetrahydropyrane antibiotics |
AU2007230630B2 (en) | 2006-03-28 | 2012-12-20 | Taigen Biotechnology Co., Ltd | Malate salts, and polymorphs of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid |
KR101084521B1 (en) | 2006-03-28 | 2011-11-18 | 워너 칠콧 컴퍼니 엘엘씨 | A coupling process for preparing quinolone intermediates |
WO2008139288A2 (en) * | 2007-05-09 | 2008-11-20 | Pfizer Inc. | Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials |
EP2332939A1 (en) | 2009-11-26 | 2011-06-15 | Æterna Zentaris GmbH | Novel Naphthyridine derivatives and the use thereof as kinase inhibitors |
EP3927703B1 (en) | 2019-02-19 | 2023-04-05 | Univerza V Ljubljani | Antibacterials based on monocyclic fragments coupled to aminopiperidine naphthyridine scaffold |
CN114793434A (en) | 2019-10-18 | 2022-07-26 | 加利福尼亚大学董事会 | 3-phenylsulfonyl-quinoline derivatives as agents for the treatment of pathogenic vascular disorders |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4418299Y1 (en) | 1965-01-16 | 1969-08-07 | ||
US4472404A (en) * | 1982-08-16 | 1984-09-18 | The Dow Chemical Company | 8-Quinolinyl carbamates and their use as urinary tract antimicrobials |
EP0387510A1 (en) * | 1989-02-10 | 1990-09-19 | Bayer Ag | Substituted 8-carbamoyloxy-quinoline derivatives, process for their preparation and their use as pesticides |
JPH0495071A (en) * | 1990-08-10 | 1992-03-27 | Kyorin Pharmaceut Co Ltd | Carbamic acid derivative |
JP3169188B2 (en) * | 1991-01-31 | 2001-05-21 | 杏林製薬株式会社 | Carbamic acid derivative and method for producing the same |
WO1994014801A1 (en) | 1992-12-29 | 1994-07-07 | Smithkline Beecham Plc | Heterocyclic urea derivatives as 5ht2c and 5ht2b antagonists |
ATE239720T1 (en) * | 1995-02-02 | 2003-05-15 | Daiichi Seiyaku Co | HETEROCYCLIC COMPOUNDS |
WO1997014681A1 (en) | 1995-10-16 | 1997-04-24 | Fujisawa Pharmaceutical Co., Ltd. | Heterocyclic compounds as h+-atpases |
JP3933244B2 (en) | 1997-04-04 | 2007-06-20 | 株式会社資生堂 | Alkylenediamine derivatives and anti-ulcer agents, antibacterial agents |
ES2201674T3 (en) | 1998-01-26 | 2004-03-16 | Smithkline Beecham Plc | DERIVATIVES OF QUINOLINA WITH ANTIBACTERIAL PROPERTIES. |
FR2798656B1 (en) | 1999-09-17 | 2004-12-17 | Aventis Pharma Sa | DERIVATIVES OF QUINOLYL PROPYL PIPERIDINE, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM |
-
1998
- 1998-10-14 GB GBGB9822440.5A patent/GB9822440D0/en not_active Ceased
-
1999
- 1999-10-11 WO PCT/EP1999/007766 patent/WO2000021952A1/en active IP Right Grant
- 1999-10-11 AT AT99950730T patent/ATE312831T1/en not_active IP Right Cessation
- 1999-10-11 DE DE69928952T patent/DE69928952T2/en not_active Expired - Fee Related
- 1999-10-11 EP EP99950730A patent/EP1121355B1/en not_active Expired - Lifetime
- 1999-10-11 ES ES99950730T patent/ES2255306T3/en not_active Expired - Lifetime
- 1999-10-11 AU AU63395/99A patent/AU6339599A/en not_active Abandoned
- 1999-10-11 US US09/807,341 patent/US6602882B1/en not_active Expired - Fee Related
- 1999-10-11 JP JP2000575858A patent/JP2002527434A/en active Pending
- 1999-10-12 PE PE1999001028A patent/PE20001112A1/en not_active Application Discontinuation
- 1999-10-12 MA MA25816A patent/MA25009A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
US6602882B1 (en) | 2003-08-05 |
JP2002527434A (en) | 2002-08-27 |
ES2255306T3 (en) | 2006-06-16 |
DE69928952T2 (en) | 2007-01-11 |
ATE312831T1 (en) | 2005-12-15 |
EP1121355A1 (en) | 2001-08-08 |
GB9822440D0 (en) | 1998-12-09 |
MA25009A1 (en) | 2000-07-01 |
PE20001112A1 (en) | 2000-10-14 |
DE69928952D1 (en) | 2006-01-19 |
WO2000021952A1 (en) | 2000-04-20 |
EP1121355B1 (en) | 2005-12-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |