AU5535080A - Preparation of 7-(sulphonomidoyl) xanthane-2 carboxylic acid derivatives - Google Patents

Preparation of 7-(sulphonomidoyl) xanthane-2 carboxylic acid derivatives

Info

Publication number
AU5535080A
AU5535080A AU55350/80A AU5535080A AU5535080A AU 5535080 A AU5535080 A AU 5535080A AU 55350/80 A AU55350/80 A AU 55350/80A AU 5535080 A AU5535080 A AU 5535080A AU 5535080 A AU5535080 A AU 5535080A
Authority
AU
Australia
Prior art keywords
preparation
sulphonomidoyl
xanthane
carboxylic acid
acid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU55350/80A
Other versions
AU531013B2 (en
Inventor
Alan Charles Barnes
Peter David Kennewell
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of AU5535080A publication Critical patent/AU5535080A/en
Application granted granted Critical
Publication of AU531013B2 publication Critical patent/AU531013B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C07D311/82—Xanthenes
    • C07D311/84—Xanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D311/86—Oxygen atoms, e.g. xanthones

Abstract

A process for the preparation of compounds of general formula I, <IMAGE> (wherein R represents a hydrogen atom or an alkyl radical containing from 1 to 9 carbon atoms and R1 represents an alkyl radical containing from 1 to 5 carbon atoms) which comprises cyclising a compound of formula II, <IMAGE> (wherein R and R1 are as defined above, Ar represents an aryl group and R2 and R3, which may be the same or different, each represents an esterifying group) followed if required, by hydrolysis to the free acid of formula I. The compounds of general formula I possess interesting anti-allergic activity.
AU55350/80A 1979-02-09 1980-02-08 Preparation of 7-(sulphonomidoyl) xanthane-2 carboxylic acid derivatives Ceased AU531013B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7904649 1979-02-09
GB7904649 1979-02-09

Publications (2)

Publication Number Publication Date
AU5535080A true AU5535080A (en) 1980-08-14
AU531013B2 AU531013B2 (en) 1983-08-04

Family

ID=10503083

Family Applications (1)

Application Number Title Priority Date Filing Date
AU55350/80A Ceased AU531013B2 (en) 1979-02-09 1980-02-08 Preparation of 7-(sulphonomidoyl) xanthane-2 carboxylic acid derivatives

Country Status (15)

Country Link
EP (1) EP0016665B1 (en)
JP (1) JPS55108867A (en)
AT (1) ATE967T1 (en)
AU (1) AU531013B2 (en)
CA (1) CA1146571A (en)
DE (1) DE3060348D1 (en)
DK (1) DK145948C (en)
ES (1) ES8102115A1 (en)
FI (1) FI800392A (en)
GB (1) GB2042540B (en)
HU (1) HU180552B (en)
IE (1) IE49389B1 (en)
IL (1) IL59046A (en)
PT (1) PT70795B (en)
ZA (1) ZA80141B (en)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL47519A (en) * 1974-07-09 1979-03-12 Roussel Uclaf 7-sulphinimidoyl(sulphimidoyl)-xanthone-2-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
JPS5850225B2 (en) * 1976-01-01 1983-11-09 ルセル・ユクラフ Novel xanthones, their salts and esters, and pharmaceuticals comprising these compounds
SE445346B (en) * 1978-03-03 1986-06-16 Roussel Uclaf SET TO PREPARE 7-SULPHONIMIDOYL-XANTON-2-CARBOXYLIC ACID DERIVATIVE

Also Published As

Publication number Publication date
AU531013B2 (en) 1983-08-04
DK54180A (en) 1980-08-10
IE49389B1 (en) 1985-10-02
FI800392A (en) 1980-08-10
EP0016665B1 (en) 1982-05-05
ES488385A0 (en) 1980-12-16
GB2042540B (en) 1982-11-24
DK145948C (en) 1983-09-26
ZA80141B (en) 1981-02-25
DE3060348D1 (en) 1982-06-24
ES8102115A1 (en) 1980-12-16
PT70795A (en) 1980-03-01
JPH0144710B2 (en) 1989-09-29
HU180552B (en) 1983-03-28
IE800250L (en) 1980-08-09
DK145948B (en) 1983-04-25
GB2042540A (en) 1980-09-24
ATE967T1 (en) 1982-05-15
EP0016665A1 (en) 1980-10-01
IL59046A0 (en) 1980-03-31
IL59046A (en) 1985-03-31
JPS55108867A (en) 1980-08-21
PT70795B (en) 1981-06-11
CA1146571A (en) 1983-05-17

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