AU3573793A - 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof - Google Patents

3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof

Info

Publication number
AU3573793A
AU3573793A AU35737/93A AU3573793A AU3573793A AU 3573793 A AU3573793 A AU 3573793A AU 35737/93 A AU35737/93 A AU 35737/93A AU 3573793 A AU3573793 A AU 3573793A AU 3573793 A AU3573793 A AU 3573793A
Authority
AU
Australia
Prior art keywords
tetrazol
pyrido
pyrimidine
preparation
same
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
AU35737/93A
Inventor
Maria Balogh
Kinga Boer
Istvan Hermecz
Agnes Horvath
Zoltan Kapui
Geza Kereszturi
Aniko Pajor
Judit Sipos
Lelle Vasvary
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chinoin Private Co Ltd
Original Assignee
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Publication of AU3573793A publication Critical patent/AU3573793A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU35737/93A 1992-02-13 1993-02-12 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof Withdrawn AU3573793A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU9200432A HUT64064A (en) 1992-02-13 1992-02-13 Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient
HU9200432 1992-02-13

Publications (1)

Publication Number Publication Date
AU3573793A true AU3573793A (en) 1993-09-03

Family

ID=10981335

Family Applications (1)

Application Number Title Priority Date Filing Date
AU35737/93A Withdrawn AU3573793A (en) 1992-02-13 1993-02-12 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof

Country Status (7)

Country Link
CN (1) CN1080289A (en)
AU (1) AU3573793A (en)
HU (1) HUT64064A (en)
IL (1) IL104706A0 (en)
MX (1) MX9300779A (en)
SI (1) SI9300075A (en)
WO (1) WO1993016076A1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU663886B2 (en) * 1990-09-25 1995-10-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara New 3-(substituted tetrazolyl)-4-oxo-4H-pyrido-{1,2-a}pyrimidines, salts thereof, pharmaceutical compositions containing them and process for preparing same

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20011764A1 (en) * 2001-08-10 2003-02-10 Dinamite Dipharma Spa HIGH PURITY PEMIROLAST METHOD
KR101122782B1 (en) * 2002-10-04 2012-04-12 프라나 바이오테크놀로지 리미티드 Neurologically-active compounds
EP1818058A3 (en) * 2006-02-13 2007-11-07 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
WO2007093184A2 (en) * 2006-02-13 2007-08-23 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
MY162507A (en) 2009-06-29 2017-06-15 Incyte Holdings Corp Pyrimidinones as pi3k inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
CA2796311A1 (en) 2010-04-14 2011-10-20 Incyte Corporation Fused derivatives as pi3k.delta. inhibitors
WO2011163195A1 (en) 2010-06-21 2011-12-29 Incyte Corporation Fused pyrrole derivatives as pi3k inhibitors
WO2012087881A1 (en) 2010-12-20 2012-06-28 Incyte Corporation N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors
US9108984B2 (en) 2011-03-14 2015-08-18 Incyte Corporation Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors
US9126948B2 (en) 2011-03-25 2015-09-08 Incyte Holdings Corporation Pyrimidine-4,6-diamine derivatives as PI3K inhibitors
RS55737B1 (en) 2011-09-02 2017-07-31 Incyte Holdings Corp Heterocyclylamines as pi3k inhibitors
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
CR20210055A (en) 2015-02-27 2021-04-27 Incyte Corp Salts of pi3k inhibitor and processes for their preparation
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2044796C (en) * 1990-06-21 2001-10-16 Atsunori Sano Process for producing pyrido[1,2-a] pyrimidine derivative

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU663886B2 (en) * 1990-09-25 1995-10-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara New 3-(substituted tetrazolyl)-4-oxo-4H-pyrido-{1,2-a}pyrimidines, salts thereof, pharmaceutical compositions containing them and process for preparing same

Also Published As

Publication number Publication date
HU9200432D0 (en) 1992-04-28
IL104706A0 (en) 1993-06-10
CN1080289A (en) 1994-01-05
HUT64064A (en) 1993-11-29
SI9300075A (en) 1993-09-30
MX9300779A (en) 1993-09-30
WO1993016076A1 (en) 1993-08-19

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