AU3014592A - Systemic control of parasites - Google Patents
Systemic control of parasitesInfo
- Publication number
- AU3014592A AU3014592A AU30145/92A AU3014592A AU3014592A AU 3014592 A AU3014592 A AU 3014592A AU 30145/92 A AU30145/92 A AU 30145/92A AU 3014592 A AU3014592 A AU 3014592A AU 3014592 A AU3014592 A AU 3014592A
- Authority
- AU
- Australia
- Prior art keywords
- group
- different
- integer
- hydrogen
- halogen atom
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/116—Heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Polymers & Plastics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Zoology (AREA)
- Animal Husbandry (AREA)
- Food Science & Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
The invention relates to a method for combating ectoparasites. More particularly, it relates to a treatment method in which the warm-blooded animal receives a dose of an effective amount, from the ovicidal viewpoint, of a heterocyclic compound containing nitrogen chosen from the group represented by the formula: <IMAGE> in which R1 is one of the following groups: <IMAGE> in which R7, R8, R9, R10, R11, R12, R13, R14, R15 , R16 and R17, which are identical or different, are each a hydrogen or halogen atom, a C1-4 alkoxy group, a C1-4 alkylthio group, a trifluoromethyl group or a nitro group; R18, R19, R20 and R21, which are identical or different, are each a hydrogen atom or a methyl group, k is an integer from 0 to 1 and l is an integer from 0 to 3; R2 and R3, which are identical or different, are each a hydrogen or halogen atom or a methyl group; R4 is a halogen atom or a methyl group; R5 and R6, which are identical or different, are each a hydrogen or halogen atom or a C1-4 haloalkyl or C1-4 haloalkoxy group; X, Y and Z, which are identical or different, are each an oxygen or sulphur atom or a methylene group, m is an integer from 0 to 4 and n is an integer from 0 to 2, which is transmitted to the ectoparasite via the blood of the animal. According to another aspect, a compound chosen from the group consisting of ivermectin, milbemycin, milbemycin oxime, moxidectin and avermectin and avermectin derivatives is also used.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81243091A | 1991-12-23 | 1991-12-23 | |
US812430 | 1991-12-23 |
Publications (2)
Publication Number | Publication Date |
---|---|
AU3014592A true AU3014592A (en) | 1993-06-24 |
AU660205B2 AU660205B2 (en) | 1995-06-15 |
Family
ID=25209544
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU30145/92A Ceased AU660205B2 (en) | 1991-12-23 | 1992-12-15 | Systemic control of parasites |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP0549441B1 (en) |
JP (1) | JP3170077B2 (en) |
AT (1) | ATE156357T1 (en) |
AU (1) | AU660205B2 (en) |
DE (1) | DE69221454T2 (en) |
ES (1) | ES2108099T3 (en) |
NZ (1) | NZ245548A (en) |
ZA (1) | ZA929950B (en) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5632999A (en) * | 1993-08-18 | 1997-05-27 | Virbac, Inc. | Sustained release pyriproxifen compositions for parasite control |
TW328044B (en) * | 1994-12-01 | 1998-03-11 | Mitsui Toatsu Chemicals | An insecticidal and acaricidal composition |
IE80657B1 (en) * | 1996-03-29 | 1998-11-04 | Merial Sas | Insecticidal combination to control mammal fleas in particular fleas on cats and dogs |
CA2378409A1 (en) * | 1999-07-23 | 2001-02-01 | Bioparken As | Control of crustacean infestation of aquatic animals |
EP1204320A2 (en) * | 1999-07-23 | 2002-05-15 | Bioparken AS | Novel juvenile hormone analogues and their use as antifouling agents |
JP4288794B2 (en) | 1999-10-26 | 2009-07-01 | 住友化学株式会社 | Insecticide and acaricide composition |
JP4701538B2 (en) * | 2001-05-21 | 2011-06-15 | 住友化学株式会社 | Agricultural pest control composition |
ES2717621T3 (en) * | 2010-07-30 | 2019-06-24 | Ceva Sante Animale Sa | Compositions to treat infestation by the heart worm |
JP6033610B2 (en) * | 2012-08-31 | 2016-11-30 | 日本ケーブル株式会社 | Evacuation support device |
WO2019005700A1 (en) * | 2017-06-26 | 2019-01-03 | Merial, Inc. | Dual active parasiticidal granule compositions, methods and uses thereof |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3950360A (en) | 1972-06-08 | 1976-04-13 | Sankyo Company Limited | Antibiotic substances |
US4031239A (en) | 1975-02-13 | 1977-06-21 | American Cyanamid Company | Cyclopropanecarboxylates for systemic control of ectoparasites |
US3962458A (en) | 1975-02-13 | 1976-06-08 | American Cyanamid Company | Systemic control of ectoparasites with pyrethroids |
US4006236A (en) | 1975-08-04 | 1977-02-01 | American Cyanamid Company | Substituted octahydrophenanthridine pesticides |
US4053631A (en) | 1976-04-02 | 1977-10-11 | American Cyanamid Company | Systemic control of ectoparasites with α-cyano-m-phenoxybenzyl α1 -C4 alkyl-2-naphthaleneacetates |
US4089975A (en) | 1977-05-13 | 1978-05-16 | The Dow Chemical Company | Method of controlling manure-breeding insects |
US4092421A (en) | 1977-05-13 | 1978-05-30 | The Dow Chemical Company | Method of controlling manure-breeding insects |
US4199569A (en) | 1977-10-03 | 1980-04-22 | Merck & Co., Inc. | Selective hydrogenation products of C-076 compounds and derivatives thereof |
US4166107A (en) | 1978-07-25 | 1979-08-28 | The United States Of America As Represented By The Secretary Of Agriculture | Sustained release bolus formulations containing insect growth regulators for control of livestock pests |
JPS5632481A (en) | 1979-08-23 | 1981-04-01 | Sankyo Co Ltd | Antibiotic b-41d, its preparation, and acaricide and anthelminthic agent and repellent containing the same as active constituent |
FR2470104A1 (en) | 1979-11-19 | 1981-05-29 | Carbonisation Entr Ceram | PULVERULENT COMPOSITION AND REFRACTORY PART OBTAINED FROM THE COMPOSITION |
US4251223A (en) | 1979-12-17 | 1981-02-17 | Miles Laboratories, Inc. | Sensitizers for peroxidative activity tests |
US4323582A (en) | 1980-07-21 | 1982-04-06 | Siegel Norman H | Method of treating animals and humans for internal and external parasites |
JPS59108785A (en) | 1982-11-25 | 1984-06-23 | Sankyo Co Ltd | 5-oxime derivative of milbemycins |
JPS59199673A (en) * | 1983-04-25 | 1984-11-12 | Sumitomo Chem Co Ltd | Nitrogen-containing heterocyclic compound, its preparation and pesticide containing the same |
US4694974A (en) | 1985-06-14 | 1987-09-22 | Michael Heck | Escapement apparatus for an automatic screw feeding machine |
ES8800986A1 (en) * | 1985-07-27 | 1987-12-01 | Pfizer | Antiparasitic avermectin and milbemycin derivatives and process for their preparation. |
NZ221262A (en) * | 1986-08-06 | 1990-08-28 | Ciba Geigy Ag | Preventing the reinfestation of dogs and cats by fleas by administering to the host a flea growth inhibiting substance orally, parenterally or by implant |
US4751223A (en) | 1986-10-14 | 1988-06-14 | Hoechst-Roussel Pharmaceuticals, Inc. | Antiinflammatory and analgesic aminoalkyl tetracyclic benzodiazepines |
DE3805235A1 (en) | 1988-02-19 | 1989-08-31 | Shell Int Research | METHOD FOR PRODUCING 3,3-DIARYLACRYLIC ACID AMIDES |
US4988824A (en) | 1989-09-11 | 1991-01-29 | Maulding Donald R | Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds |
-
1992
- 1992-12-15 AU AU30145/92A patent/AU660205B2/en not_active Ceased
- 1992-12-21 NZ NZ245548A patent/NZ245548A/en unknown
- 1992-12-21 EP EP92403478A patent/EP0549441B1/en not_active Expired - Lifetime
- 1992-12-21 ES ES92403478T patent/ES2108099T3/en not_active Expired - Lifetime
- 1992-12-21 DE DE69221454T patent/DE69221454T2/en not_active Expired - Lifetime
- 1992-12-21 AT AT92403478T patent/ATE156357T1/en not_active IP Right Cessation
- 1992-12-22 ZA ZA929950A patent/ZA929950B/en unknown
- 1992-12-22 JP JP34277492A patent/JP3170077B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
DE69221454T2 (en) | 1997-12-11 |
JPH06211792A (en) | 1994-08-02 |
NZ245548A (en) | 1996-04-26 |
EP0549441B1 (en) | 1997-08-06 |
JP3170077B2 (en) | 2001-05-28 |
EP0549441A1 (en) | 1993-06-30 |
ES2108099T3 (en) | 1997-12-16 |
ATE156357T1 (en) | 1997-08-15 |
AU660205B2 (en) | 1995-06-15 |
ZA929950B (en) | 1993-11-03 |
DE69221454D1 (en) | 1997-09-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |