AU2017341825B2 - Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders - Google Patents

Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders Download PDF

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Publication number: AU2017341825B2
Authority: AU; Australia
Prior art keywords: pharmaceutical composition; subject; compound; use according; day
Prior art date: 2016-10-13
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

AU2017341825A

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English (en)

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AU2017341825A1 (en

Inventor

Radko KOMERS

Alvin SHIH

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Travere Therapeutics Inc

Original Assignee

Travere Therapeutics Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2016-10-13

Filing date

2017-10-13

Publication date

2023-06-01

2017-10-13 Application filed by Travere Therapeutics Inc filed Critical Travere Therapeutics Inc

2019-04-11 Publication of AU2017341825A1 publication Critical patent/AU2017341825A1/en

2021-03-18 Assigned to Travere Therapeutics, Inc. reassignment Travere Therapeutics, Inc. Amend patent request/document other than specification (104) Assignors: Retrophin, Inc.

2023-06-01 Application granted granted Critical

2023-06-01 Publication of AU2017341825B2 publication Critical patent/AU2017341825B2/en

2023-08-22 Priority to AU2023219839A priority Critical patent/AU2023219839A1/en

Status Active legal-status Critical Current

2037-10-13 Anticipated expiration legal-status Critical

Links

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NHDIQVFFNDKAQU-UHFFFAOYSA-N tripropan-2-yl borate Chemical compound CC(C)OB(OC(C)C)OC(C)C NHDIQVFFNDKAQU-UHFFFAOYSA-N 0.000 description 1
230000002485 urinary effect Effects 0.000 description 1
230000006442 vascular tone Effects 0.000 description 1
230000002227 vasoactive effect Effects 0.000 description 1
235000015112 vegetable and seed oil Nutrition 0.000 description 1
239000008158 vegetable oil Substances 0.000 description 1
229920002554 vinyl polymer Polymers 0.000 description 1
238000005550 wet granulation Methods 0.000 description 1
238000009736 wetting Methods 0.000 description 1
229940100445 wheat starch Drugs 0.000 description 1
235000010447 xylitol Nutrition 0.000 description 1
239000000811 xylitol Substances 0.000 description 1
HEBKCHPVOIAQTA-SCDXWVJYSA-N xylitol Chemical compound OC[C@H](O)[C@@H](O)[C@H](O)CO HEBKCHPVOIAQTA-SCDXWVJYSA-N 0.000 description 1
229960002675 xylitol Drugs 0.000 description 1
239000011592 zinc chloride Substances 0.000 description 1
235000005074 zinc chloride Nutrition 0.000 description 1
239000002888 zwitterionic surfactant Substances 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

AU2017341825A 2016-10-13 2017-10-13 Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders Active AU2017341825B2 (en)

Priority Applications (1)

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AU2023219839A AU2023219839A1 (en)	2016-10-13	2023-08-22	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US201662407860P	2016-10-13	2016-10-13
US62/407,860		2016-10-13
US201662423079P	2016-11-16	2016-11-16
US62/423,079		2016-11-16
PCT/US2017/056538 WO2018071784A1 (en)	2016-10-13	2017-10-13	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders

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AU2023219839A Division AU2023219839A1 (en)	2016-10-13	2023-08-22	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders

Publications (2)

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AU2017341825A1 AU2017341825A1 (en)	2019-04-11
AU2017341825B2 true AU2017341825B2 (en)	2023-06-01

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AU2017341825A Active AU2017341825B2 (en)	2016-10-13	2017-10-13	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders
AU2023219839A Pending AU2023219839A1 (en)	2016-10-13	2023-08-22	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders

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AU2023219839A Pending AU2023219839A1 (en)	2016-10-13	2023-08-22	Biphenyl sulfonamide compounds for the treatment of kidney diseases or disorders

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US (3)	US20190262317A1 (zh)
EP (1)	EP3525784A1 (zh)
JP (3)	JP2019530713A (zh)
KR (3)	KR102528435B1 (zh)
CN (5)	CN110049764A (zh)
AU (2)	AU2017341825B2 (zh)
BR (1)	BR112019007576A2 (zh)
CA (1)	CA3039819A1 (zh)
MA (1)	MA46524A (zh)
WO (1)	WO2018071784A1 (zh)

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EP3860594A1 (en)	2018-10-04	2021-08-11	Travere Therapeutics, Inc.	Biphenyl sulfonamide compounds for the treatment of type iv collagen diseases
WO2020132594A1 (en)	2018-12-21	2020-06-25	Retrophin, Inc.	Amorphous sparsentan compositions
US20220304979A1 (en) *	2019-12-17	2022-09-29	Chinook Therapeutics, Inc.	Methods of reducing disease flares
JP2023507739A (ja) *	2019-12-17	2023-02-27	チヌークセラピューティクス，インコーポレイテッド	アトラセンタンによるｉｇａ腎症を治療する方法
CN115768421A (zh) *	2020-04-10	2023-03-07	切诺克治疗公司	治疗糖尿病肾病的方法
WO2022246200A1 (en)	2021-05-21	2022-11-24	Travere Therapeutics, Inc.	Methods of treating kidney diseases or disorders
KR20240051999A (ko)	2021-08-26	2024-04-22	상하이 한서 바이오메디컬 컴퍼니 리미티드	방향족 고리 함유 생물학적 길항제, 이의 제조 방법 및 용도
WO2024073672A1 (en)	2022-09-30	2024-04-04	Travere Therapeutics, Inc.	Combination therapy with sparsentan and a sglt2 inhibitor for treating kidney diseases or disorders

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2017
- 2017-10-13 CN CN201780076280.6A patent/CN110049764A/zh active Pending
- 2017-10-13 CN CN202311092711.1A patent/CN116983302A/zh active Pending
- 2017-10-13 WO PCT/US2017/056538 patent/WO2018071784A1/en unknown
- 2017-10-13 AU AU2017341825A patent/AU2017341825B2/en active Active
- 2017-10-13 EP EP17791821.6A patent/EP3525784A1/en active Pending
- 2017-10-13 KR KR1020227032048A patent/KR102528435B1/ko active IP Right Grant
- 2017-10-13 US US16/340,848 patent/US20190262317A1/en not_active Abandoned
- 2017-10-13 CN CN202311093985.2A patent/CN117085013A/zh active Pending
- 2017-10-13 BR BR112019007576A patent/BR112019007576A2/pt unknown
- 2017-10-13 CN CN202311094233.8A patent/CN117017985A/zh active Pending
- 2017-10-13 KR KR1020197011413A patent/KR20190077348A/ko not_active Application Discontinuation
- 2017-10-13 CA CA3039819A patent/CA3039819A1/en active Pending
- 2017-10-13 CN CN202210441043.8A patent/CN114788823A/zh active Pending
- 2017-10-13 JP JP2019519669A patent/JP2019530713A/ja not_active Withdrawn
- 2017-10-13 MA MA046524A patent/MA46524A/fr unknown
- 2017-10-13 KR KR1020237014470A patent/KR20230066644A/ko not_active Application Discontinuation
2020
- 2020-05-22 US US16/882,206 patent/US10864197B2/en active Active
- 2020-11-12 US US17/096,637 patent/US20210196688A1/en not_active Abandoned
2022
- 2022-07-15 JP JP2022113880A patent/JP2022141802A/ja active Pending
- 2022-07-15 JP JP2022113881A patent/JP2022137245A/ja active Pending
2023
- 2023-08-22 AU AU2023219839A patent/AU2023219839A1/en active Pending

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Also Published As

Publication number	Publication date
EP3525784A1 (en)	2019-08-21
BR112019007576A2 (pt)	2019-07-02
CN110049764A (zh)	2019-07-23
KR20190077348A (ko)	2019-07-03
CN117085013A (zh)	2023-11-21
US20210196688A1 (en)	2021-07-01
JP2022141802A (ja)	2022-09-29
JP2022137245A (ja)	2022-09-21
CN114788823A (zh)	2022-07-26
US10864197B2 (en)	2020-12-15
CA3039819A1 (en)	2018-04-19
US20190262317A1 (en)	2019-08-29
KR20220132030A (ko)	2022-09-29
AU2023219839A1 (en)	2023-09-07
JP2019530713A (ja)	2019-10-24
AU2017341825A1 (en)	2019-04-11
KR20230066644A (ko)	2023-05-16
US20200281901A1 (en)	2020-09-10
KR102528435B1 (ko)	2023-05-03
CN116983302A (zh)	2023-11-03
CN117017985A (zh)	2023-11-10
MA46524A (fr)	2019-08-21
WO2018071784A1 (en)	2018-04-19

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2023-09-28

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