AU2017262960A1 - Substituted 5,6,7,8-tetrahydro(1,2,4)triazolo(4,3-a)pyridine-3(2H)-ones and 2,5,6,7-tetrahydro-3H-pyrrolo(2,1-c)(1,2,4)triazol-3-ones, and use thereof - Google Patents
Substituted 5,6,7,8-tetrahydro(1,2,4)triazolo(4,3-a)pyridine-3(2H)-ones and 2,5,6,7-tetrahydro-3H-pyrrolo(2,1-c)(1,2,4)triazol-3-ones, and use thereofInfo
- Publication number
- AU2017262960A1 AU2017262960A1 AU2017262960A AU2017262960A AU2017262960A1 AU 2017262960 A1 AU2017262960 A1 AU 2017262960A1 AU 2017262960 A AU2017262960 A AU 2017262960A AU 2017262960 A AU2017262960 A AU 2017262960A AU 2017262960 A1 AU2017262960 A1 AU 2017262960A1
- Authority
- AU
- Australia
- Prior art keywords
- tetrahydro
- ones
- triazolo
- pyrrolo
- triazol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- WTMDBOJIFXBWBL-UHFFFAOYSA-N 2,5,6,7-tetrahydropyrrolo[2,1-c][1,2,4]triazol-3-one Chemical class C1CCN2C(=O)NN=C21 WTMDBOJIFXBWBL-UHFFFAOYSA-N 0.000 title 1
- VNJXPEWQUVGHKM-UHFFFAOYSA-N 5,6,7,8-tetrahydro-2H-[1,2,4]triazolo[4,3-a]pyridin-3-one Chemical class C1CCCN2C(=O)NN=C21 VNJXPEWQUVGHKM-UHFFFAOYSA-N 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP16168809 | 2016-05-09 | ||
EPEP16168809.8 | 2016-05-09 | ||
PCT/EP2017/060900 WO2017194459A1 (en) | 2016-05-09 | 2017-05-08 | Substituted 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine-3(2h)-ones and 2,5,6,7-tetrahydro-3h-pyrrolo[2,1-c][1,2,4]triazol-3-ones, and use thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2017262960A1 true AU2017262960A1 (en) | 2018-11-15 |
AU2017262960B2 AU2017262960B2 (en) | 2021-11-11 |
Family
ID=55919764
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2017262960A Active AU2017262960B2 (en) | 2016-05-09 | 2017-05-08 | Substituted 5,6,7,8-tetrahydro(1,2,4)triazolo(4,3-a)pyridine-3(2H)-ones and 2,5,6,7-tetrahydro-3H-pyrrolo(2,1-c)(1,2,4)triazol-3-ones, and use thereof |
Country Status (30)
Country | Link |
---|---|
US (1) | US10722501B2 (en) |
JP (1) | JP6987784B2 (en) |
KR (1) | KR102438965B1 (en) |
CN (1) | CN109476658B (en) |
AR (1) | AR110600A1 (en) |
AU (1) | AU2017262960B2 (en) |
BR (1) | BR112018073061A2 (en) |
CA (1) | CA3023383A1 (en) |
CL (1) | CL2018003194A1 (en) |
CO (1) | CO2018012136A2 (en) |
CR (1) | CR20180540A (en) |
CU (1) | CU24536B1 (en) |
DO (1) | DOP2018000246A (en) |
EA (1) | EA037531B1 (en) |
EC (1) | ECSP18083950A (en) |
GE (1) | GEP20227365B (en) |
IL (1) | IL262548B (en) |
JO (1) | JOP20170113B1 (en) |
MX (1) | MX2018013797A (en) |
NI (1) | NI201800118A (en) |
PE (1) | PE20190325A1 (en) |
PH (1) | PH12018502359A1 (en) |
SA (1) | SA518400397B1 (en) |
SG (1) | SG11201809724PA (en) |
SV (1) | SV2018005783A (en) |
TN (1) | TN2018000376A1 (en) |
TW (1) | TWI758291B (en) |
UA (1) | UA125644C2 (en) |
UY (1) | UY37234A (en) |
WO (1) | WO2017194459A1 (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2007009796A (en) | 2007-08-14 | 2009-02-25 | Cell Therapy And Technology S | Gel containing pirfenidone. |
MX346763B (en) | 2012-03-28 | 2017-03-31 | Cell Therapy And Tech S A De C V | Semi-solid topical composition which contains pirfenidone and modified diallyl disulphide oxide (m-ddo) for eliminating or preventing acne. |
US11337973B2 (en) | 2017-11-07 | 2022-05-24 | Bayer Aktiengesellschaft | Substituted [1,2,4]triazolo[4,3-A]pyrazines as prolyl endopeptidase inhibitors |
CN110950797A (en) * | 2019-12-06 | 2020-04-03 | 丽水绿氟科技有限公司 | Preparation method of 2-trifluoromethyl-3-fluoro-4-picolinic acid and derivatives thereof |
CN115466212B (en) * | 2022-10-26 | 2023-09-22 | 河南农业大学 | 2-trifluoromethyl quinoline compound and synthetic method and application thereof |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3966781A (en) | 1970-12-17 | 1976-06-29 | Merck Sharp & Dohme (I.A.) Corporation | Deuteration of functional group-containing hydrocarbons |
HUT76640A (en) * | 1995-08-17 | 1997-10-28 | Chinoin Gyogyszer Es Vegyeszet | Compounds of pharmaceutical activity cyclic amide derivatives, pharmaceutical compositions containing them, process for producing them and their use |
DE19834044A1 (en) | 1998-07-29 | 2000-02-03 | Bayer Ag | New substituted pyrazole derivatives |
DE19834047A1 (en) | 1998-07-29 | 2000-02-03 | Bayer Ag | Substituted pyrazole derivatives |
DE19943639A1 (en) | 1999-09-13 | 2001-03-15 | Bayer Ag | Dicarboxylic acid derivatives with novel pharmaceutical properties |
DE19943634A1 (en) | 1999-09-13 | 2001-04-12 | Bayer Ag | Novel dicarboxylic acid derivatives with pharmaceutical properties |
DE19943636A1 (en) | 1999-09-13 | 2001-03-15 | Bayer Ag | Novel dicarboxylic acid derivatives with pharmaceutical properties |
DE19943635A1 (en) | 1999-09-13 | 2001-03-15 | Bayer Ag | Novel aminodicarboxylic acid derivatives with pharmaceutical properties |
AR031176A1 (en) | 2000-11-22 | 2003-09-10 | Bayer Ag | NEW DERIVATIVES OF PIRAZOLPIRIDINA SUBSTITUTED WITH PIRIDINE |
DE10110750A1 (en) | 2001-03-07 | 2002-09-12 | Bayer Ag | Novel aminodicarboxylic acid derivatives with pharmaceutical properties |
DE10110749A1 (en) | 2001-03-07 | 2002-09-12 | Bayer Ag | Substituted aminodicarboxylic acid derivatives |
DE10220570A1 (en) | 2002-05-08 | 2003-11-20 | Bayer Ag | Carbamate-substituted pyrazolopyridines |
US7618983B2 (en) | 2004-11-10 | 2009-11-17 | Janssen Pharmaceutica, N.V. | Bicyclic triazole α4 integrin inhibitors |
US8524654B2 (en) * | 2007-05-21 | 2013-09-03 | The Uab Research Foundation | Prolyl endopeptidase inhibitors for reducing or preventing neutrophilic inflammation |
WO2011062864A2 (en) | 2009-11-17 | 2011-05-26 | Emory University | Inhibitors of nox enzymes and methods of use thereof |
DE102010021637A1 (en) | 2010-05-26 | 2011-12-01 | Bayer Schering Pharma Aktiengesellschaft | Substituted 5-fluoro-1H-pyrazolopyridines and their use |
EP2708539A1 (en) | 2010-07-09 | 2014-03-19 | Bayer Intellectual Property GmbH | Annulated pyrimidines and triazines and their use |
DE102010040233A1 (en) | 2010-09-03 | 2012-03-08 | Bayer Schering Pharma Aktiengesellschaft | Bicyclic aza heterocycles and their use |
DE102010043379A1 (en) | 2010-11-04 | 2012-05-10 | Bayer Schering Pharma Aktiengesellschaft | Substituted 6-fluoro-1H-pyrazolo [4,3-b] pyridines and their use |
EP2675440B1 (en) | 2011-02-14 | 2020-03-25 | Merck Sharp & Dohme Corp. | Cathepsin cysteine protease inhibitors |
KR20130091464A (en) * | 2012-02-08 | 2013-08-19 | 한미약품 주식회사 | Triazolopyridine derivatives as a tyrosine kinase inhibitor |
US9624214B2 (en) | 2012-11-05 | 2017-04-18 | Bayer Pharma Aktiengesellschaft | Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
-
2017
- 2017-05-04 JO JOP/2017/0113A patent/JOP20170113B1/en active
- 2017-05-08 TW TW106115093A patent/TWI758291B/en active
- 2017-05-08 JP JP2018558379A patent/JP6987784B2/en active Active
- 2017-05-08 UY UY0001037234A patent/UY37234A/en not_active Application Discontinuation
- 2017-05-08 BR BR112018073061-0A patent/BR112018073061A2/en active Search and Examination
- 2017-05-08 TN TNP/2018/000376A patent/TN2018000376A1/en unknown
- 2017-05-08 PE PE2018002337A patent/PE20190325A1/en unknown
- 2017-05-08 KR KR1020187032180A patent/KR102438965B1/en active IP Right Grant
- 2017-05-08 WO PCT/EP2017/060900 patent/WO2017194459A1/en unknown
- 2017-05-08 US US16/300,480 patent/US10722501B2/en active Active
- 2017-05-08 CU CU2018000139A patent/CU24536B1/en unknown
- 2017-05-08 EA EA201892518A patent/EA037531B1/en not_active IP Right Cessation
- 2017-05-08 GE GEAP201714952A patent/GEP20227365B/en unknown
- 2017-05-08 AU AU2017262960A patent/AU2017262960B2/en active Active
- 2017-05-08 AR ARP170101192A patent/AR110600A1/en unknown
- 2017-05-08 SG SG11201809724PA patent/SG11201809724PA/en unknown
- 2017-05-08 CA CA3023383A patent/CA3023383A1/en active Pending
- 2017-05-08 CN CN201780042622.2A patent/CN109476658B/en active Active
- 2017-05-08 UA UAA201811797A patent/UA125644C2/en unknown
- 2017-05-08 CR CR20180540A patent/CR20180540A/en unknown
- 2017-05-08 MX MX2018013797A patent/MX2018013797A/en unknown
-
2018
- 2018-10-24 IL IL262548A patent/IL262548B/en unknown
- 2018-11-08 SA SA518400397A patent/SA518400397B1/en unknown
- 2018-11-08 PH PH12018502359A patent/PH12018502359A1/en unknown
- 2018-11-09 DO DO2018000246A patent/DOP2018000246A/en unknown
- 2018-11-09 NI NI201800118A patent/NI201800118A/en unknown
- 2018-11-09 CL CL2018003194A patent/CL2018003194A1/en unknown
- 2018-11-09 CO CONC2018/0012136A patent/CO2018012136A2/en unknown
- 2018-11-09 EC ECSENADI201883950A patent/ECSP18083950A/en unknown
- 2018-11-09 SV SV2018005783A patent/SV2018005783A/en unknown
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