AU2002257497A1 - Derivatives of exendin - Google Patents

Derivatives of exendin

Info

Publication number: AU2002257497A1
Authority: AU; Australia
Prior art keywords: exendin; derivatives
Prior art date: 2001-05-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2002257497A

Other versions

AU2002257497B2 (en

Inventor

Chunjuan Shen

Yukun Sun

Dengxi Wu

Gang Yu

Shaoling Zhao

Jiaxiang Zhou

Zhiyong Zhu

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Shanghai Benemae Pharmaceutical Corp

Original Assignee

Shanghai Benemae Pharmaceutical Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-10

Filing date

2002-05-08

Publication date

2003-05-01

2001-05-10 Priority claimed from CNB011128569A external-priority patent/CN1162446C/en

2002-05-08 Application filed by Shanghai Benemae Pharmaceutical Corp filed Critical Shanghai Benemae Pharmaceutical Corp

2003-05-01 Publication of AU2002257497A1 publication Critical patent/AU2002257497A1/en

2007-10-11 Application granted granted Critical

2007-10-11 Publication of AU2002257497B2 publication Critical patent/AU2002257497B2/en

2015-07-23 Assigned to SHANGHAI BENEMAE PHARMACEUTICAL CORPORATION reassignment SHANGHAI BENEMAE PHARMACEUTICAL CORPORATION Request to Amend Deed and Register Assignors: SHANGHAI HUAYI BIO LAB

2022-05-08 Anticipated expiration legal-status Critical

Status Expired legal-status Critical Current

Links

AU2002257497A 2001-05-10 2002-05-08 Derivatives of exendin Expired AU2002257497B2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
CNB011128569A CN1162446C (en)	2001-05-10	2001-05-10	Insulinotropic hormone secretion peptide derivative
CN01112856.9		2001-05-10
PCT/CN2002/000316 WO2002090388A1 (en)	2001-05-10	2002-05-08	Derivatives of exendin

Publications (2)

Publication Number	Publication Date
AU2002257497A1 true AU2002257497A1 (en)	2003-05-01
AU2002257497B2 AU2002257497B2 (en)	2007-10-11

Family

ID=4659603

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2002257497A Expired AU2002257497B2 (en)	2001-05-10	2002-05-08	Derivatives of exendin

Country Status (9)

Country	Link
US (1)	US7329646B2 (en)
EP (2)	EP1386930A4 (en)
JP (1)	JP4287153B2 (en)
KR (1)	KR100902208B1 (en)
CN (1)	CN1162446C (en)
AU (1)	AU2002257497B2 (en)
BR (1)	BRPI0209685B8 (en)
CA (1)	CA2446394C (en)
WO (1)	WO2002090388A1 (en)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6924264B1 (en) *	1999-04-30	2005-08-02	Amylin Pharmaceuticals, Inc.	Modified exendins and exendin agonists
CN1162446C (en) *	2001-05-10	2004-08-18	上海华谊生物技术有限公司	Insulinotropic hormone secretion peptide derivative
JP2008515856A (en)	2004-10-07	2008-05-15	ノボノルディスクアクティーゼルスカブ	Delayed GLP-1 compound
JP5107713B2 (en)	2004-10-07	2012-12-26	ノヴォノルディスクアー／エス	Delayed exendin-4 compound
CN100429227C (en) *	2005-06-29	2008-10-29	常州制药厂有限公司	Exendin 4 polypeptide segment
CN100374462C (en) *	2005-11-21	2008-03-12	大连帝恩生物工程有限公司	Gerobriecin pancrease glucagon peptidel (SGLP-1), its preparation and use
BRPI0712559A2 (en) *	2006-05-26	2012-11-20	Amylin Pharmaceuticals Inc	compositions and methods for the treatment of congestive heart failure
CN101125207B (en) *	2006-11-14	2012-09-05	上海华谊生物技术有限公司	Exendin or its analogs with polyethylene group and its preparation and application
EP3456340B1 (en) *	2007-01-08	2022-02-16	The Trustees of the University of Pennsylvania	Glp-1 receptor antagonist for use in the treatment of congenital hyperinsulinism
RU2413528C2 (en)	2007-01-18	2011-03-10	Открытое Акционерное Общество "Валента Фармацевтика"	Exenatide and dalargin drug for treating diabetes, adminisration and therapy
CN101040936B (en) *	2007-04-28	2011-10-19	大连水产学院	Compound Chinese traditional medicine agent for preventing fish verminosis
CN101215324B (en) *	2007-12-26	2010-11-24	吉林大学	Exenatide short peptide simulation peptide and application thereof in preparing medicament for curing diabetes
KR100864584B1 (en) *	2008-02-25	2008-10-24	성균관대학교산학협력단	Exendin derivative linked biotin, method for the preparation thereof and pharmaceutical composition comprising the same
CN101463078B (en) *	2009-01-12	2011-07-27	华东师范大学	Exendin-4 derivative and solid phase chemical synthesis thereof
CN101665799A (en) *	2009-06-29	2010-03-10	华东师范大学	Recombination preparation method and application of Exendin-4 derivative
WO2011063549A1 (en) *	2009-11-26	2011-06-03	Wu Xiaoyan	Long-acting exendin 4 analogues
CN102397558B (en) *	2010-09-09	2013-08-14	中国人民解放军军事医学科学院毒物药物研究所	Positioning pegylation modified compound of Exendin-4 analog and application thereof
CN102532301B (en) *	2010-12-31	2014-09-03	上海医药工业研究院	Novel Exendin-4 analogues and preparation method thereof
CN106928341B (en) *	2011-03-30	2021-06-01	上海仁会生物制药股份有限公司	Fixed-point mono-substituted pegylated Exendin analogue and preparation method thereof
UA116217C2 (en)	2012-10-09	2018-02-26	Санофі	Exendin-4 derivatives as dual glp1/glucagon agonists
ES2688367T3 (en)	2012-12-21	2018-11-02	Sanofi	Derivatives of exendin-4 as dual agonists of GLP1 / GIP or trigonal of GLP1 / GIP / glucagon
AU2014234314B2 (en)	2013-03-21	2018-02-15	Sanofi-Aventis Deutschland Gmbh	Synthesis of cyclic imide containing peptide products
US10087221B2 (en)	2013-03-21	2018-10-02	Sanofi-Aventis Deutschland Gmbh	Synthesis of hydantoin containing peptide products
TW201609795A (en)	2013-12-13	2016-03-16	賽諾菲公司	EXENDIN-4 peptide analogues as dual GLP-1/GIP receptor agonists
EP3080152A1 (en)	2013-12-13	2016-10-19	Sanofi	Non-acylated exendin-4 peptide analogues
EP3080154B1 (en)	2013-12-13	2018-02-07	Sanofi	Dual glp-1/gip receptor agonists
WO2015086733A1 (en)	2013-12-13	2015-06-18	Sanofi	Dual glp-1/glucagon receptor agonists
TW201625669A (en)	2014-04-07	2016-07-16	賽諾菲公司	Peptidic dual GLP-1/glucagon receptor agonists derived from Exendin-4
TW201625670A (en)	2014-04-07	2016-07-16	賽諾菲公司	Dual GLP-1/glucagon receptor agonists derived from EXENDIN-4
TW201625668A (en)	2014-04-07	2016-07-16	賽諾菲公司	Exendin-4 derivatives as peptidic dual GLP-1/glucagon receptor agonists
US9932381B2 (en)	2014-06-18	2018-04-03	Sanofi	Exendin-4 derivatives as selective glucagon receptor agonists
AR105319A1 (en)	2015-06-05	2017-09-27	Sanofi Sa	PROPHARMS THAT INCLUDE A DUAL AGONIST GLU-1 / GLUCAGON CONJUGATE HIALURONIC ACID CONNECTOR
TW201706291A (en)	2015-07-10	2017-02-16	賽諾菲公司	New EXENDIN-4 derivatives as selective peptidic dual GLP-1/glucagon receptor agonists

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE69129226T2 (en)	1990-01-24	1998-07-30	Douglas I Buckley	GLP-1 ANALOG USES IN DIABETE TREATMENT
US5424286A (en)	1993-05-24	1995-06-13	Eng; John	Exendin-3 and exendin-4 polypeptides, and pharmaceutical compositions comprising same
DK144093D0 (en) *	1993-12-23	1993-12-23	Novo Nordisk As
US6265204B1 (en) *	1997-01-17	2001-07-24	Genencor International, Inc.	DNA sequences, vectors, and fusion polypeptides for secretion of polypeptides in filamentous fungi
DK1032587T4 (en) *	1997-11-14	2013-04-08	Amylin Pharmaceuticals Llc	New exendin agonist compounds
BR9815670A (en) *	1997-11-14	2000-10-17	Amylin Pharmaceuticals Inc	Exendin agonist compounds
US6329336B1 (en) *	1999-05-17	2001-12-11	Conjuchem, Inc.	Long lasting insulinotropic peptides
US6514500B1 (en)	1999-10-15	2003-02-04	Conjuchem, Inc.	Long lasting synthetic glucagon like peptide {GLP-!}
US6506724B1 (en)	1999-06-01	2003-01-14	Amylin Pharmaceuticals, Inc.	Use of exendins and agonists thereof for the treatment of gestational diabetes mellitus
EP1076066A1 (en) *	1999-07-12	2001-02-14	Zealand Pharmaceuticals A/S	Peptides for lowering blood glucose levels
US6528486B1 (en)	1999-07-12	2003-03-04	Zealand Pharma A/S	Peptide agonists of GLP-1 activity
WO2001041561A1 (en) *	1999-12-07	2001-06-14	Lee Yong Hwa	A bathtub for a pet dog
CN1162446C (en) *	2001-05-10	2004-08-18	上海华谊生物技术有限公司	Insulinotropic hormone secretion peptide derivative
CN1363654A (en)	2001-07-19	2002-08-14	上海华谊生物技术有限公司	Genetically engineered bacteria and process for preparing insulinotropic hormone secretion peptide GLP-1 (7-36)

2001
- 2001-05-10 CN CNB011128569A patent/CN1162446C/en not_active Expired - Lifetime
2002
- 2002-05-08 EP EP02727167A patent/EP1386930A4/en not_active Withdrawn
- 2002-05-08 CA CA2446394A patent/CA2446394C/en not_active Expired - Lifetime
- 2002-05-08 WO PCT/CN2002/000316 patent/WO2002090388A1/en active Application Filing
- 2002-05-08 EP EP10001237.6A patent/EP2223938B1/en not_active Expired - Lifetime
- 2002-05-08 AU AU2002257497A patent/AU2002257497B2/en not_active Expired
- 2002-05-08 BR BRPI0209685A patent/BRPI0209685B8/en not_active IP Right Cessation
- 2002-05-08 JP JP2002587464A patent/JP4287153B2/en not_active Expired - Lifetime
- 2002-05-08 KR KR1020037014451A patent/KR100902208B1/en active IP Right Grant
2003
- 2003-11-07 US US10/704,409 patent/US7329646B2/en not_active Expired - Lifetime

Publication	Publication Date	Title
AU2002257497A1 (en)	2003-05-01	Derivatives of exendin
AU2002363005A1 (en)	2003-05-06	Derivatives of uk-2a
EP1386930A4 (en)	2005-09-07	Derivatives of exendin
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