AU2002255077A1 - Derivatives of N-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same - Google Patents
Derivatives of N-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing sameInfo
- Publication number
- AU2002255077A1 AU2002255077A1 AU2002255077A AU2002255077A AU2002255077A1 AU 2002255077 A1 AU2002255077 A1 AU 2002255077A1 AU 2002255077 A AU2002255077 A AU 2002255077A AU 2002255077 A AU2002255077 A AU 2002255077A AU 2002255077 A1 AU2002255077 A1 AU 2002255077A1
- Authority
- AU
- Australia
- Prior art keywords
- aminoacids
- arylsulfonyl
- beta
- derivatives
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000004202 aminomethyl group Chemical group [H]N([H])C([H])([H])* 0.000 title 1
- 150000001576 beta-amino acids Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR01/04315 | 2001-03-28 | ||
FR0104315A FR2822827B1 (en) | 2001-03-28 | 2001-03-28 | NOVEL N- (ARYLSULFONYL) BETA-AMINOACIDS DERIVATIVES COMPRISING A SUBSTITUTED AMINOMETHYL GROUP, THEIR PREPARATION METHOD AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
PCT/FR2002/001059 WO2002076964A1 (en) | 2001-03-28 | 2002-03-27 | Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002255077A1 true AU2002255077A1 (en) | 2003-03-27 |
AU2002255077B2 AU2002255077B2 (en) | 2007-08-16 |
Family
ID=8861734
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002255077A Ceased AU2002255077B2 (en) | 2001-03-28 | 2002-03-27 | Derivatives of N-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same |
Country Status (38)
Country | Link |
---|---|
US (1) | US7157454B2 (en) |
EP (1) | EP1373233B1 (en) |
JP (1) | JP4188695B2 (en) |
KR (1) | KR100887038B1 (en) |
CN (1) | CN1297546C (en) |
AR (1) | AR033686A1 (en) |
AT (1) | ATE372329T1 (en) |
AU (1) | AU2002255077B2 (en) |
BG (1) | BG108201A (en) |
BR (1) | BR0208489A (en) |
CA (1) | CA2436225C (en) |
CY (1) | CY1106980T1 (en) |
CZ (1) | CZ301337B6 (en) |
DE (1) | DE60222248T2 (en) |
DK (1) | DK1373233T3 (en) |
EA (1) | EA006430B1 (en) |
EE (1) | EE05198B1 (en) |
ES (1) | ES2291464T3 (en) |
FR (1) | FR2822827B1 (en) |
HK (1) | HK1059931A1 (en) |
HR (1) | HRP20030748B1 (en) |
HU (1) | HUP0401538A3 (en) |
IL (3) | IL157215A0 (en) |
IS (1) | IS2582B (en) |
MA (1) | MA26995A1 (en) |
ME (1) | MEP25408A (en) |
MX (1) | MXPA03008756A (en) |
NO (1) | NO326519B1 (en) |
NZ (1) | NZ527429A (en) |
PL (1) | PL207553B1 (en) |
PT (1) | PT1373233E (en) |
RS (1) | RS52138B (en) |
SK (1) | SK286753B6 (en) |
TN (1) | TNSN03058A1 (en) |
TW (1) | TWI233923B (en) |
UA (1) | UA75906C2 (en) |
WO (1) | WO2002076964A1 (en) |
ZA (1) | ZA200306037B (en) |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HUP0303644A3 (en) * | 2001-03-30 | 2008-06-30 | Pfizer Prod Inc | Pyridazinone-derivatives aldose reductase inhibitors, their use and pharmaceutical compositions containing them |
FR2840897B1 (en) | 2002-06-14 | 2004-09-10 | Fournier Lab Sa | NOVEL ARYLSULFONAMIDE DERIVATIVES AND THEIR USE IN THERAPEUTICS |
US7425631B2 (en) | 2003-04-10 | 2008-09-16 | Amgen Inc. | Compounds and methods of use |
US20050038099A1 (en) * | 2003-05-02 | 2005-02-17 | Tung Jay S. | Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists |
DE602004021933D1 (en) * | 2003-05-02 | 2009-08-20 | Elan Pharm Inc | 4-BROM-5- (2-CHLORO-BENZOYLAMINO) -1H-PYRAZOLE-3-CARBOXYLIC ACID (PHENYL) AMID DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B1 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES |
ES2314418T3 (en) * | 2003-05-02 | 2009-03-16 | Elan Pharmaceuticals, Inc. | DERIVATIVES OF AMIDAS OF THE ACID 4-BROMO-5- (2-CHLOROBENZOYLAMINE) -1H-PIRAZOL-3-CARBOXYCLIC AND RELATED COMPOUNDS AS ANTIGONISTS OF THE B1 BRADIQUININE RECEPTOR FOR THE TREATMENT OF INFLAMMATORY DISEASES. |
CA2534188A1 (en) * | 2003-08-07 | 2005-02-24 | Merck & Co., Inc. | Sulfonyl substituted n-(biarylmethyl) aminocyclopropanecarboxamides |
DE602004027301D1 (en) * | 2003-12-22 | 2010-07-01 | Merck Sharp & Dohme | ALPHA-HYDROXYAMIDES AS BRADYKININANTAGONISTS OR INVERSE AGONISTS |
WO2006036664A1 (en) * | 2004-09-23 | 2006-04-06 | Amgen Inc. | Substituted sulfonamidopropionamides and methods of use |
CA2582459A1 (en) * | 2004-10-06 | 2006-04-20 | Amgen Inc. | Substituted sulfones and methods of use |
AU2005295818A1 (en) | 2004-10-12 | 2006-04-27 | Amgen Inc. | Novel B1 bradykinin receptor antagonists |
US7612060B2 (en) | 2004-10-13 | 2009-11-03 | Amgen Inc. | Triazoles and methods of use |
US20060217362A1 (en) * | 2004-12-29 | 2006-09-28 | Tung Jay S | Novel compounds useful for bradykinin B1 receptor antagonism |
EP1741444A1 (en) * | 2005-07-05 | 2007-01-10 | Jerini AG | Kinin antagonists for treating bladder dysfunction |
ATE428702T1 (en) * | 2005-09-21 | 2009-05-15 | Reddy S Lab Eu Ltd Dr | METHOD FOR PRODUCING AMINO ACID DERIVATIVES |
HU230518B1 (en) | 2005-12-20 | 2016-10-28 | Richter Gedeon Nyrt. | New phenantridine derivatives as selective bradykinin b1 receptor antagonists, process for their preparation and pharmaceutical compositions containing them |
WO2008046573A1 (en) | 2006-10-16 | 2008-04-24 | Grünenthal GmbH | Substituted sulfonamide derivatives for use as bradykinin 1 receptor modulators |
HUP0600810A3 (en) * | 2006-10-27 | 2008-09-29 | Richter Gedeon Nyrt | New sulfonamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them |
HUP0600808A3 (en) | 2006-10-27 | 2008-09-29 | Richter Gedeon Nyrt | New benzamide derivatives as bradykinin antagonists, process for their preparation and pharmaceutical compositions containing them |
HUP0600809A3 (en) * | 2006-10-27 | 2008-09-29 | Richter Gedeon Nyrt | New phenylsulfamoyl-benzamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them |
FR2916352B1 (en) * | 2007-05-23 | 2009-07-31 | Sanofi Aventis Sa | USE OF A NON-PEPTIDE ANTAGONIST OF BRADYKININ B1 RECEPTOR FOR THE PREPARATION OF MEDICAMENTS USEFUL IN THE PREVENTION OR TREATMENT OF ARTERIAL HYPERTENSION. |
WO2008153967A1 (en) * | 2007-06-08 | 2008-12-18 | Contec Therapeutics, Inc. | Bk1 antagonist conjugates |
FR2919803B1 (en) * | 2007-08-07 | 2011-07-22 | Sanofi Aventis | USE OF A NON-PEPTIDE RECEPTOR B1 ANTAGONIST FOR THE PREPARATION OF MEDICAMENTS USEFUL IN THE TREATMENT OF OBESITY AND OBESITY OR DIABETES PATHOLOGIES |
AU2007360523A1 (en) * | 2007-10-27 | 2009-04-30 | Richter Gedeon Nyrt. | New non-peptide derivatives as bradykinin B1 antagonists |
PE20091782A1 (en) * | 2008-04-08 | 2009-11-15 | Gruenenthal Chemie | SUBSTITUTE SULFONAMIDE DERIVATIVES |
CN102159210A (en) * | 2008-08-21 | 2011-08-17 | 吉瑞工厂 | Methods for treating cns disorders |
EP2330899A1 (en) * | 2008-08-21 | 2011-06-15 | Richter Gedeon Nyrt. | Methods for treating neuropathic pain |
HUP1000598A2 (en) | 2010-11-05 | 2012-09-28 | Richter Gedeon Nyrt | Indole derivatives |
AR097279A1 (en) | 2013-08-09 | 2016-03-02 | Actelion Pharmaceuticals Ltd | DERIVATIVES OF BENZIMIDAZOLIL-METIL UREA AS ALX RECEIVER AGONISTS |
JP6448498B2 (en) * | 2015-08-04 | 2019-01-09 | 日本ゴア株式会社 | Precision filter for circuit board manufacturing process liquid |
EP3672938B1 (en) | 2017-08-25 | 2023-11-01 | The Board of Supervisors of Louisiana State University and Agricultural and Mechanical College | Compounds for ameliorating pain |
NZ762985A (en) | 2017-09-22 | 2024-03-22 | Jubilant Epipad LLC | Heterocyclic compounds as pad inhibitors |
HUE061607T2 (en) | 2017-10-18 | 2023-07-28 | Jubilant Epipad LLC | Imidazo-pyridine compounds as pad inhibitors |
CN111386265A (en) | 2017-11-06 | 2020-07-07 | 朱比连特普罗德尔有限责任公司 | Pyrimidine derivatives as inhibitors of PD1/PD-L1 activation |
EP3704120B1 (en) | 2017-11-24 | 2024-03-06 | Jubilant Episcribe LLC | Heterocyclic compounds as prmt5 inhibitors |
BR112020018610A2 (en) | 2018-03-13 | 2020-12-29 | Jubilant Prodel LLC | COMPOUNDS OF FORMULA I, FORMULA II, FORMULA III, FORMULA IV, FORMULA V, FORMULA VI, OR ITS POLYMORPHOS, STEREOISOMERS, TAUTOMERS, PROPHARMACES, SOLVATES AND PHARMACEUTICAL MALES OF THE MESOUSLY MESOUS MOSES; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND METHOD FOR THE TREATMENT AND / OR PREVENTION OF VARIOUS DISEASES, INCLUDING CANCER AND INFECTIOUS DISEASES |
CN114075274B (en) * | 2022-01-18 | 2022-04-12 | 浙江湃肽生物有限公司深圳分公司 | Somarunotide analog and preparation method and application thereof |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5714497A (en) * | 1993-02-15 | 1998-02-03 | Sanofi | Compounds bearing sulphamoyl and amidino radicals, their preparation process and pharmaceutical compositions containing them |
FR2701480B1 (en) * | 1993-02-15 | 1995-05-24 | Sanofi Elf | Compounds with a sulfamoyl and amidino group, process for their preparation and pharmaceutical compositions containing them. |
FR2735128B1 (en) * | 1995-06-07 | 1997-07-25 | Fournier Ind & Sante | NOVEL BENZENESULFONAMIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USE. |
DE19548709A1 (en) * | 1995-12-23 | 1997-07-03 | Merck Patent Gmbh | Tyrosine derivatives |
FR2743562B1 (en) * | 1996-01-11 | 1998-04-03 | Sanofi Sa | N- (ARYLSULFONYL) AMINO ACID DERIVATIVES, THEIR PREPARATION, THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
ATE359264T1 (en) * | 1996-01-23 | 2007-05-15 | Shionogi & Co | SULFONATED AMINO ACID DERIVATIVES AND METALLOPROTEINASE INHIBITORS CONTAINING SAME |
-
2001
- 2001-03-28 FR FR0104315A patent/FR2822827B1/en not_active Expired - Fee Related
-
2002
- 2002-03-26 AR ARP020101096A patent/AR033686A1/en active IP Right Grant
- 2002-03-27 CA CA2436225A patent/CA2436225C/en not_active Expired - Fee Related
- 2002-03-27 ZA ZA200306037A patent/ZA200306037B/en unknown
- 2002-03-27 EA EA200300942A patent/EA006430B1/en not_active IP Right Cessation
- 2002-03-27 BR BR0208489-9A patent/BR0208489A/en not_active Application Discontinuation
- 2002-03-27 PT PT02724383T patent/PT1373233E/en unknown
- 2002-03-27 AU AU2002255077A patent/AU2002255077B2/en not_active Ceased
- 2002-03-27 UA UA2003087628A patent/UA75906C2/en unknown
- 2002-03-27 CN CNB028075390A patent/CN1297546C/en not_active Expired - Fee Related
- 2002-03-27 EE EEP200300417A patent/EE05198B1/en not_active IP Right Cessation
- 2002-03-27 TN TNPCT/FR2002/001059A patent/TNSN03058A1/en unknown
- 2002-03-27 ES ES02724383T patent/ES2291464T3/en not_active Expired - Lifetime
- 2002-03-27 US US10/472,674 patent/US7157454B2/en not_active Expired - Lifetime
- 2002-03-27 AT AT02724383T patent/ATE372329T1/en active
- 2002-03-27 KR KR1020037012554A patent/KR100887038B1/en not_active IP Right Cessation
- 2002-03-27 TW TW091106017A patent/TWI233923B/en not_active IP Right Cessation
- 2002-03-27 RS YU74403A patent/RS52138B/en unknown
- 2002-03-27 CZ CZ20032588A patent/CZ301337B6/en not_active IP Right Cessation
- 2002-03-27 DK DK02724383T patent/DK1373233T3/en active
- 2002-03-27 HU HU0401538A patent/HUP0401538A3/en not_active Application Discontinuation
- 2002-03-27 NZ NZ527429A patent/NZ527429A/en not_active IP Right Cessation
- 2002-03-27 JP JP2002576224A patent/JP4188695B2/en not_active Expired - Fee Related
- 2002-03-27 MX MXPA03008756A patent/MXPA03008756A/en active IP Right Grant
- 2002-03-27 PL PL367242A patent/PL207553B1/en unknown
- 2002-03-27 ME MEP-254/08A patent/MEP25408A/en unknown
- 2002-03-27 IL IL15721502A patent/IL157215A0/en unknown
- 2002-03-27 SK SK1204-2003A patent/SK286753B6/en not_active IP Right Cessation
- 2002-03-27 EP EP02724383A patent/EP1373233B1/en not_active Expired - Lifetime
- 2002-03-27 WO PCT/FR2002/001059 patent/WO2002076964A1/en active IP Right Grant
- 2002-03-27 DE DE60222248T patent/DE60222248T2/en not_active Expired - Lifetime
-
2003
- 2003-08-03 IL IL157215A patent/IL157215A/en not_active IP Right Cessation
- 2003-08-07 IS IS6906A patent/IS2582B/en unknown
- 2003-08-13 MA MA27279A patent/MA26995A1/en unknown
- 2003-09-17 HR HR20030748A patent/HRP20030748B1/en not_active IP Right Cessation
- 2003-09-24 NO NO20034267A patent/NO326519B1/en not_active IP Right Cessation
- 2003-09-25 BG BG108201A patent/BG108201A/en unknown
-
2004
- 2004-04-19 HK HK04102735A patent/HK1059931A1/en not_active IP Right Cessation
-
2007
- 2007-11-07 CY CY20071101426T patent/CY1106980T1/en unknown
-
2008
- 2008-06-16 IL IL192233A patent/IL192233A/en not_active IP Right Cessation
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU2002255077A1 (en) | Derivatives of N-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same | |
PL367242A1 (en) | Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same | |
AU2001237526A1 (en) | Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof | |
AU2002363236A1 (en) | Compounds, pharmaceutical compositions and methods of use therefor | |
HK1067626A1 (en) | Novel 2h-pyridazine-3-one derivatives, pharmaceutical compositions containing the same and a process for the preparation of the active ingredient | |
AU2002365516A1 (en) | Benzamide derivatives, processes for their preparation, and their pharmaceutical use | |
HK1043365B (en) | N-(iminomethyl)amine derivatives, their preparation, their use as medicines and compositions containing them | |
AU2002233463A1 (en) | Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use | |
IL162185A0 (en) | Phenylpropionate derivatives, methods for the preparation thereof and pharmaceutical compositions containing the same | |
AU2001235737A1 (en) | Novel 1,3-dihydro-2h-indol-2-one, preparation method and pharmaceutical compositions containing same | |
AU2003251695A1 (en) | Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same | |
AU2001292331A2 (en) | 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation | |
AU2001292331A1 (en) | 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation | |
AU2002360117A1 (en) | Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same | |
AU2002313065A1 (en) | Novel piperidinecarboxamide derivatives, method for preparing same and pharmaceutical compositions containing same | |
AU2002306687A1 (en) | Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them | |
SI1245565T1 (en) | Indenoindolone derivatives, process for their preparation and pharmaceutical compositions containing them | |
AU2002300093A1 (en) | New benzenesulphonamide compounds, a process for their preparation and pharmaceutical compositions containing them | |
HUP0304065A2 (en) | Novel 5-thio-betha-d-xylopyranoside derivatives, preparation method thereof, pharmaceutical compositions containing same and use thereof | |
AU2001269190A1 (en) | Carbamate and thiocarbamate podophyllotoxin derivatives, preparation method and pharmaceutical compositions containing them | |
AU2001274000A1 (en) | Optically active 2-aminotetralin derivatives, the processes for the preparation thereof and the therapeutical use of pharmaceutical compositions containing them | |
AU2002300092A1 (en) | New benzenesulphonamide compounds, a process for their preparation and pharmaceutical compositions containing them | |
SI1266887T1 (en) | Indenoindoline derivatives, their process of preparation and pharmaceutical compositions containing them | |
AU2002349008A1 (en) | Derivatives of etoposide and analogs, and pharmaceutical compositions containing them | |
AU2002313036A1 (en) | Novel 5-thio-B-D-xylopyranoside Derivatives, Preparation Method Thereof, Pharmaceutical Compositions Containing Same and the Therapeutic Use Thereof |