AU2001289937A1 - Substituted 1-aminobutan-3-ol derivatives - Google Patents

Substituted 1-aminobutan-3-ol derivatives

Info

Publication number: AU2001289937A1
Authority: AU; Australia
Prior art keywords: aminobutan; derivatives; substituted
Prior art date: 2000-09-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001289937A

Other versions

AU2001289937B2 (en

Inventor

Helmut Buschmann

Boris Chizh

Michael Haurand

Utz-Peter Jagusch

Corinna Maul

Bernd Sundermann

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Gruenenthal GmbH

Original Assignee

Gruenenthal GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-09-29

Filing date

2001-09-28

Publication date

2002-06-27

2000-09-29 Priority claimed from DE10049483A external-priority patent/DE10049483A1/en

2001-09-28 Application filed by Gruenenthal GmbH filed Critical Gruenenthal GmbH

2002-06-27 Publication of AU2001289937A1 publication Critical patent/AU2001289937A1/en

2007-01-18 Application granted granted Critical

2007-01-18 Publication of AU2001289937B2 publication Critical patent/AU2001289937B2/en

2021-09-28 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Links

NAXUFNXWXFZVSI-UHFFFAOYSA-N 4-aminobutan-2-ol Chemical class CC(O)CCN NAXUFNXWXFZVSI-UHFFFAOYSA-N 0.000 title 1

AU2001289937A 2000-09-29 2001-09-28 Substituted 1-aminobutan-3-ol derivatives Ceased AU2001289937B2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10049483.8		2000-09-29
DE10049483A DE10049483A1 (en)	2000-09-29	2000-09-29	Substituted 1-aminobutan-3-ol derivatives
PCT/EP2001/011231 WO2002028817A1 (en)	2000-09-29	2001-09-28	Substituted 1-aminobutan-3-ol derivatives

Publications (2)

Publication Number	Publication Date
AU2001289937A1 true AU2001289937A1 (en)	2002-06-27
AU2001289937B2 AU2001289937B2 (en)	2007-01-18

Family

ID=7658871

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
AU2002220578A Ceased AU2002220578B2 (en)	2000-09-29	2001-09-28	O-substituted 6-methyl-tramadol derivatives
AU2057802A Pending AU2057802A (en)	2000-09-29	2001-09-28	O-substituted 6-methyl-tramadol derivatives
AU8993701A Pending AU8993701A (en)	2000-09-29	2001-09-28	Substituted 1-aminobutan-3-ol derivatives
AU2001289937A Ceased AU2001289937B2 (en)	2000-09-29	2001-09-28	Substituted 1-aminobutan-3-ol derivatives

Family Applications Before (3)

Application Number	Title	Priority Date	Filing Date
AU2002220578A Ceased AU2002220578B2 (en)	2000-09-29	2001-09-28	O-substituted 6-methyl-tramadol derivatives
AU2057802A Pending AU2057802A (en)	2000-09-29	2001-09-28	O-substituted 6-methyl-tramadol derivatives
AU8993701A Pending AU8993701A (en)	2000-09-29	2001-09-28	Substituted 1-aminobutan-3-ol derivatives

Country Status (29)

Country	Link
US (2)	US7022739B2 (en)
EP (2)	EP1322592B2 (en)
JP (2)	JP2004509939A (en)
KR (2)	KR100835549B1 (en)
CN (2)	CN1478067A (en)
AR (1)	AR034158A1 (en)
AT (2)	ATE272046T1 (en)
AU (4)	AU2002220578B2 (en)
BR (2)	BR0114380A (en)
CA (2)	CA2423860A1 (en)
DE (3)	DE10049483A1 (en)
DK (2)	DK1322593T3 (en)
EC (2)	ECSP034532A (en)
ES (2)	ES2225605T5 (en)
HK (2)	HK1052924B (en)
HU (2)	HUP0303361A3 (en)
IL (2)	IL155106A0 (en)
MX (2)	MXPA03002738A (en)
NO (2)	NO20031387L (en)
NZ (2)	NZ525171A (en)
PE (1)	PE20020413A1 (en)
PL (2)	PL361382A1 (en)
PT (2)	PT1322592E (en)
RU (2)	RU2286334C2 (en)
SI (2)	SI1322592T1 (en)
SK (2)	SK3382003A3 (en)
TR (2)	TR200402230T4 (en)
WO (2)	WO2002028817A1 (en)
ZA (2)	ZA200303220B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE10049483A1 (en) *	2000-09-29	2002-05-02	Gruenenthal Gmbh	Substituted 1-aminobutan-3-ol derivatives
CN1599607A (en)	2001-10-16	2005-03-23	恩都制药公司	Carbinols for the treatment of neuropathic dysfunction
BR0306811A (en) *	2002-01-11	2004-10-26	Sankyo Co	Compound, pharmacologically acceptable ester thereof, pharmaceutical composition and methods for the prevention or treatment of autoimmune diseases, rheumatoid arthritis and rejection caused by the transplantation of various organs in a mammal
US8128957B1 (en)	2002-02-21	2012-03-06	Valeant International (Barbados) Srl	Modified release compositions of at least one form of tramadol
US20050182056A9 (en) *	2002-02-21	2005-08-18	Seth Pawan	Modified release formulations of at least one form of tramadol
PT1562567T (en) *	2002-11-22	2017-08-24	Gruenenthal Gmbh	Combination of selected analgesics and cox-ii inhibitors
KR20110136901A (en)	2004-02-24	2011-12-21	상꾜 가부시키가이샤	Amino alcohol compound
NZ580429A (en) *	2007-05-31	2012-04-27	Sepracor Inc	Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors
KR20110100241A (en) *	2008-12-05	2011-09-09	아르퀼 인코포레이티드	Raf inhibitors and their uses
ES2343050B1 (en) *	2008-12-16	2011-06-14	Chemo Iberica, S.A.	PROCEDURE FOR THE PREPARATION OF DEVENLAFAXINE AND ITS PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS.
WO2012100423A1 (en) *	2011-01-27	2012-08-02	Eli Lilly And Company	Analgesic compounds, methods, and formulations
JP2019502761A (en) *	2016-01-21	2019-01-31	ラボラトリオスレヴィエセエレ	Method of making ((R) -3-[(-1-methylpyrrolidin-2-yl) methyl] -5- (2-phenylsulfonylethyl) -1H-indole

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3652589A (en) *	1967-07-27	1972-03-28	Gruenenthal Chemie	1-(m-substituted phenyl)-2-aminomethyl cyclohexanols
ZA732238B (en) *	1972-04-06	1974-01-30	American Home Prod	Benzylamine analgesics
US4155935A (en)	1973-03-26	1979-05-22	American Home Products Corporation	Benzylamine analgesics
DE19525137C2 (en) *	1995-07-11	2003-02-27	Gruenenthal Gmbh	6-Dimethylaminomethyl-1-phenyl-cyclohexane compounds as intermediates for the preparation of pharmaceutical agents
US6017963A (en) *	1995-11-14	2000-01-25	Euro-Celtique, S.A.	Formulation for intranasal administration
DE19547766A1 (en) *	1995-12-20	1997-06-26	Gruenenthal Gmbh	1-phenyl-2-dimethylaminomethyl-cyclohexan-1-ol compounds as active pharmaceutical ingredients
DE19601744C2 (en) *	1996-01-19	1998-04-16	Gruenenthal Gmbh	Process for the preparation of the enantiomers of O-demethyltramadol
DE19609847A1 (en) *	1996-03-13	1997-09-18	Gruenenthal Gmbh	Dimethyl- (3-aryl-but-3-enyl) amine compounds as active pharmaceutical ingredients
US5919826A (en) *	1996-10-24	1999-07-06	Algos Pharmaceutical Corporation	Method of alleviating pain
US6245804B1 (en) *	1997-05-30	2001-06-12	Schering Aktiengesellschaft	Nonsteroidal gestagens
EP0996613B1 (en) *	1997-07-15	2002-10-30	Russinsky Limited	Pure cis-tramadol hydrochloride production
ATE257147T1 (en) *	1998-05-22	2004-01-15	Mallinckrodt Inc	AN IMPROVED SYNTHESIS AND PURIFICATION PROCESS FOR (R,R)-2-((DIMETHYLAMINO)METHYL)-1-(3-METHOXYPHENYL) CYCLOHEXANOL HYDROCHLORIDE
ES2141688B1 (en) *	1998-11-06	2001-02-01	Vita Invest Sa	NEW ESTERS DERIVED FROM SUBSTITUTED FENIL-CICLOHEXIL COMPOUNDS.
DE19915601A1 (en) *	1999-04-07	2000-10-19	Gruenenthal Gmbh	3-Amino-3-arylpropan-1-ol derivatives, their preparation and use
CZ2002524A3 (en) *	1999-08-20	2002-11-13	Ortho-Mcneil Pharmaceutical, Inc.	Composition containing tramadol and anticonvulsants
PE20010623A1 (en) *	1999-10-05	2001-07-07	Gruenenthal Chemie	USE OF (+) - TRAMADOL AND / OR O-DEMETILTRAMADOL FOR TREATMENT OF INCREASED URINARY URGENCY AND / OR URINARY INCONTINENCE
US6339105B1 (en) *	1999-10-12	2002-01-15	Ortho-Mcneil Pharmaceutical, Inc.	Analgesic regimen
DE10000312A1 (en) *	2000-01-05	2001-07-12	Gruenenthal Gmbh	Substituted aminomethyl phenyl cyclohexane derivatives
DE10049483A1 (en) *	2000-09-29	2002-05-02	Gruenenthal Gmbh	Substituted 1-aminobutan-3-ol derivatives
DE10048714A1 (en) *	2000-09-30	2002-04-11	Gruenenthal Gmbh	5-amino-1-penlen-3-ol derivatives
US6649783B2 (en) *	2001-10-03	2003-11-18	Euro-Celtique, S.A.	Synthesis of (+/-)-2-((dimethylamino)methyl)-1-(aryl)cyclohexanols
AU2002364517A1 (en) *	2001-11-30	2003-06-17	Sepracor Inc.	Tramadol analogs and uses thereof

2000
- 2000-09-29 DE DE10049483A patent/DE10049483A1/en not_active Withdrawn
2001
- 2001-09-28 TR TR2004/02230T patent/TR200402230T4/en unknown
- 2001-09-28 WO PCT/EP2001/011231 patent/WO2002028817A1/en active IP Right Grant
- 2001-09-28 BR BR0114380-8A patent/BR0114380A/en not_active IP Right Cessation
- 2001-09-28 SK SK338-2003A patent/SK3382003A3/en not_active Application Discontinuation
- 2001-09-28 PE PE2001000968A patent/PE20020413A1/en not_active Application Discontinuation
- 2001-09-28 ES ES01969791T patent/ES2225605T5/en not_active Expired - Lifetime
- 2001-09-28 SI SI200130184T patent/SI1322592T1/en unknown
- 2001-09-28 SI SI200130189T patent/SI1322593T1/en unknown
- 2001-09-28 PL PL01361382A patent/PL361382A1/en unknown
- 2001-09-28 PT PT01969791T patent/PT1322592E/en unknown
- 2001-09-28 KR KR1020037004490A patent/KR100835549B1/en not_active IP Right Cessation
- 2001-09-28 AU AU2002220578A patent/AU2002220578B2/en not_active Ceased
- 2001-09-28 AU AU2057802A patent/AU2057802A/en active Pending
- 2001-09-28 AR ARP010104583A patent/AR034158A1/en unknown
- 2001-09-28 CN CNA018196454A patent/CN1478067A/en active Pending
- 2001-09-28 NZ NZ525171A patent/NZ525171A/en unknown
- 2001-09-28 AU AU8993701A patent/AU8993701A/en active Pending
- 2001-09-28 MX MXPA03002738A patent/MXPA03002738A/en active IP Right Grant
- 2001-09-28 TR TR2004/02030T patent/TR200402030T4/en unknown
- 2001-09-28 NZ NZ524976A patent/NZ524976A/en unknown
- 2001-09-28 DK DK01985699T patent/DK1322593T3/en active
- 2001-09-28 HU HU0303361A patent/HUP0303361A3/en unknown
- 2001-09-28 JP JP2002531080A patent/JP2004509939A/en active Pending
- 2001-09-28 PL PL01361632A patent/PL361632A1/en not_active Application Discontinuation
- 2001-09-28 KR KR1020037004521A patent/KR100864796B1/en not_active IP Right Cessation
- 2001-09-28 IL IL15510601A patent/IL155106A0/en unknown
- 2001-09-28 JP JP2002532404A patent/JP2004510755A/en active Pending
- 2001-09-28 EP EP01969791A patent/EP1322592B2/en not_active Expired - Lifetime
- 2001-09-28 PT PT01985699T patent/PT1322593E/en unknown
- 2001-09-28 DK DK01969791T patent/DK1322592T4/en active
- 2001-09-28 CN CNB018166067A patent/CN100391933C/en not_active Expired - Fee Related
- 2001-09-28 AT AT01985699T patent/ATE272046T1/en not_active IP Right Cessation
- 2001-09-28 IL IL15510501A patent/IL155105A0/en unknown
- 2001-09-28 EP EP01985699A patent/EP1322593B1/en not_active Expired - Lifetime
- 2001-09-28 MX MXPA03002737A patent/MXPA03002737A/en active IP Right Grant
- 2001-09-28 DE DE50103036T patent/DE50103036D1/en not_active Expired - Lifetime
- 2001-09-28 CA CA002423860A patent/CA2423860A1/en not_active Abandoned
- 2001-09-28 HU HU0303195A patent/HUP0303195A3/en unknown
- 2001-09-28 ES ES01985699T patent/ES2225628T3/en not_active Expired - Lifetime
- 2001-09-28 RU RU2003111756/04A patent/RU2286334C2/en not_active IP Right Cessation
- 2001-09-28 CA CA002423903A patent/CA2423903A1/en not_active Abandoned
- 2001-09-28 RU RU2003111753/04A patent/RU2288219C2/en not_active IP Right Cessation
- 2001-09-28 WO PCT/EP2001/011276 patent/WO2002026694A1/en active IP Right Grant
- 2001-09-28 AU AU2001289937A patent/AU2001289937B2/en not_active Ceased
- 2001-09-28 SK SK340-2003A patent/SK286727B6/en not_active IP Right Cessation
- 2001-09-28 DE DE50103035T patent/DE50103035D1/en not_active Expired - Lifetime
- 2001-09-28 BR BR0114381-6A patent/BR0114381A/en not_active IP Right Cessation
- 2001-09-28 AT AT01969791T patent/ATE272045T1/en active
2003
- 2003-03-26 NO NO20031387A patent/NO20031387L/en not_active Application Discontinuation
- 2003-03-26 NO NO20031382A patent/NO20031382L/en not_active Application Discontinuation
- 2003-03-28 EC EC2003004532A patent/ECSP034532A/en unknown
- 2003-03-28 US US10/401,020 patent/US7022739B2/en not_active Expired - Fee Related
- 2003-03-28 EC EC2003004530A patent/ECSP034530A/en unknown
- 2003-03-31 US US10/402,147 patent/US6828345B2/en not_active Expired - Fee Related
- 2003-04-24 ZA ZA200303220A patent/ZA200303220B/en unknown
- 2003-04-24 ZA ZA200303214A patent/ZA200303214B/en unknown
- 2003-07-16 HK HK03105140.5A patent/HK1052924B/en not_active IP Right Cessation
- 2003-07-17 HK HK03105163.7A patent/HK1052925B/en not_active IP Right Cessation

Publication	Publication Date	Title
AU2001280099A1 (en)	2002-04-02	4-acylaminopyrazole derivatives
AU2001230584A1 (en)	2001-08-20	1h-imidazopyridine derivatives
AU2001230537A1 (en)	2001-08-14	Pyridoxazine derivatives
AU2002349676A1 (en)	2003-06-10	4-oxoquinoline derivatives
AU2000267458A1 (en)	2001-10-15	Hypercomputer
AU2001281802A1 (en)	2001-12-17	6-phenylpyrrolopyrimidinedione derivatives
AU2001278790A1 (en)	2002-03-04	1h-imidazopyridine derivatives
AU2002213978A1 (en)	2002-06-27	Substituted C-cyclohexylmethylamine derivatives
AU2002212301A1 (en)	2002-04-15	Diazacycloalkanedione derivatives
AU5256301A (en)	2001-11-12	Froindazole derivative
AU2002212959A1 (en)	2002-04-29	Cycloalkylfluorosulfonamide derivatives
AU2001265871A1 (en)	2001-11-07	Substituted sulfonylaminopyrimidines
AU2001254731A1 (en)	2001-10-23	Substituted phenyluracils
AU2001289937A1 (en)	2002-06-27	Substituted 1-aminobutan-3-ol derivatives
AU2002215212A1 (en)	2002-08-01	1-methylcarbapenem derivatives
AU2001258255A1 (en)	2001-11-29	Substituted benzoylcyclohexenones
AU2001254661A1 (en)	2001-09-03	Aminosulfonylbiphenyl derivatives
AU2001230565A1 (en)	2001-08-14	Perfluoroisopropylbenzene derivatives
AU2001234313A1 (en)	2001-09-03	Novel phenylheteroalkylamine derivatives
AU2001242772A1 (en)	2001-10-03	3-substituted-4-pyrimidone derivatives
AU2002212263A1 (en)	2002-04-15	Substituted 5-amino-1-pentene-3-ol derivatives
AU2002221632A1 (en)	2002-06-27	5-amino-1-pentene-3-ol substituted derivatives
AU2001288484A1 (en)	2002-03-13	Novel metallotexaphyrin derivatives
AU2002223604A1 (en)	2002-07-11	Substituted phenyluracils
AU2002358715A1 (en)	2003-07-09	Tetrahydrobenzfluorene derivatives