AU2001248849A1 - Estra-1,3,5(10)-triene derivatives - Google Patents

Estra-1,3,5(10)-triene derivatives

Info

Publication number: AU2001248849A1
Authority: AU; Australia
Prior art keywords: estra; triene derivatives; triene; derivatives
Prior art date: 2000-04-24
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2001248849A

Inventor

Tsutomu Agatsuma

Shiro Akinaga

Nobuyoshi Amishiro

Kozue Hayashi

Yoji Ino

Mayumi Miyata

Chikara Murakata

Takeshi Takahashi

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

KH Neochem Co Ltd

Original Assignee

Kyowa Hakko Kogyo Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-24

Filing date

2001-04-24

Publication date

2001-11-07

2001-04-24 Application filed by Kyowa Hakko Kogyo Co Ltd filed Critical Kyowa Hakko Kogyo Co Ltd

2001-11-07 Publication of AU2001248849A1 publication Critical patent/AU2001248849A1/en

Status Abandoned legal-status Critical Current

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring

AU2001248849A 2000-04-24 2001-04-24 Estra-1,3,5(10)-triene derivatives Abandoned AU2001248849A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2000121960		2000-04-24
JP2000-121960		2000-04-24
PCT/JP2001/003505 WO2001081364A1 (en)	2000-04-24	2001-04-24	Estra-1,3,5(10)-triene derivatives

Publications (1)

Publication Number	Publication Date
AU2001248849A1 true AU2001248849A1 (en)	2001-11-07

Family

ID=18632506

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2001248849A Abandoned AU2001248849A1 (en)	2000-04-24	2001-04-24	Estra-1,3,5(10)-triene derivatives

Country Status (5)

Country	Link
US (1)	US6953785B2 (en)
EP (1)	EP1284272A4 (en)
JP (1)	JPWO2001081364A1 (en)
AU (1)	AU2001248849A1 (en)
WO (1)	WO2001081364A1 (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20040214807A1 (en) *	1993-08-06	2004-10-28	D'amato Robert J.	Estrogenic compounds as anti-mitotic agents
US6995278B2 (en) *	2000-08-18	2006-02-07	Entre Med, Inc.	Antiangiogenic agents
US20050192258A1 (en) *	2000-08-18	2005-09-01	Agoston Gregory E.	Antiangiogenic agents
EP1446388B1 (en) *	2001-11-21	2013-01-09	Sterix Limited	1,2,4-triazole derivatives containing a sulphamate group as aromatase inhibitors
EP1568381A1 (en) *	2002-10-09	2005-08-31	Kyowa Hakko Kogyo Co., Ltd.	Remedy for hormone-dependent cancer
BRPI0408703A (en)	2003-03-24	2006-03-07	Sterix Ltd	estrogen derivatives as steroid sulfatase inhibitors
GB0306717D0 (en) *	2003-03-24	2003-04-30	Sterix Ltd	Compound
JP2006526025A (en) *	2003-05-28	2006-11-16	エントレメッドインコーポレイテッド	Anti-angiogenic agent
JP2007529426A (en)	2004-03-12	2007-10-25	エントレメッドインコーポレイテッド	Anti-angiogenic drugs
US20070004689A1 (en) *	2004-03-12	2007-01-04	Agoston Gregory E	Antiangiogenic agents
DE102004025985A1 (en) *	2004-05-21	2005-12-15	Schering Ag	Estriol and estetrol prodrugs
DE102004025966A1 (en) *	2004-05-21	2005-12-15	Schering Ag	Estradiol prodrugs
GB0421106D0 (en) *	2004-09-22	2004-10-27	Sterix Ltd	Compound
CA2587448A1 (en) *	2004-11-29	2006-06-01	Entremed, Inc.	A method of administering anti-angiogenic agents and a method of treating disease using same
WO2007109312A2 (en)	2006-03-20	2007-09-27	Entremed, Inc.	Disease modifying anti-arthritic activity of 2-methoxyestradiol
US20080051380A1 (en)	2006-08-25	2008-02-28	Auerbach Alan H	Methods and compositions for treating cancer
MX2015000347A (en) *	2012-07-10	2015-04-14	Bayer Pharma AG	3-substituted estra-1,3,5(10),16-tetraene derivatives, methods for the production thereof, pharmaceutical preparations containing same, and use thereof for the production of medicaments.

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9118478D0 (en) *	1991-08-29	1991-10-16	Imperial College	Steroid sulphatase inhibitors
GB9625334D0 (en)	1996-12-05	1997-01-22	Imperial College	Compound
GB9118465D0 (en) *	1991-08-29	1991-10-16	Imperial College	Steroid sulphatase inhibitors
US5556847A (en) *	1994-10-27	1996-09-17	Duquesne University Of The Holy Ghost	Methods of effecting memory enhancement mediated by steroid sulfatase inhibitors
US5571933A (en) *	1994-11-17	1996-11-05	Duquesne University Of The Holy Ghost	Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use
AU713341B2 (en) *	1996-09-12	1999-12-02	Teikoku Hormone Mfg. Co., Ltd.	3-substituted-d-homo-1,3,5,(10)-estratriene derivatives
US5763492A (en) *	1996-10-01	1998-06-09	Duguesne University Of The Holy Ghost	Methods for effecting memory enhancement mediated by non-steroidal sulfatase inhibitors
US5763432A (en) *	1997-01-29	1998-06-09	Sri International	Steriod inhibitors of estrone sulfatase and associated pharmaceutical compositions and methods of use
DE19712488A1 (en) *	1997-03-25	1998-10-01	Knoell Hans Forschung Ev	Steroid sulfamates, processes for their preparation and use thereof
US6288050B1 (en)	1997-07-18	2001-09-11	Duquesne University Of The Holy Ghost	Steroid sulfatase inhibitors and methods for making and using the same
US5880115A (en) *	1997-07-18	1999-03-09	Duquesne University Of The Holy Ghost	Steroid sulfatase inhibitors and methods for making and using the same
GB2331988B (en)	1997-12-04	2003-04-16	Imperial College	Polycyclic sulphamate inhibitors or oestrone sulphatase
GB2331987B (en)	1997-12-04	2002-11-27	Imperial College	Polycyclic sulphamate inhibitors of oestrone sulphatase
US6046186A (en) *	1997-12-24	2000-04-04	Sri International	Estrone sulfamate inhibitors of estrone sulfatase, and associated pharmaceutical compositions and methods of use
US6054446A (en)	1997-12-24	2000-04-25	Sri International	Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
WO2000053620A1 (en)	1999-03-10	2000-09-14	Nippon Organon K. K.	Novel estradiol derivatives
DE19943708B4 (en)	1999-09-08	2007-12-20	Bayer Schering Pharma Ag	New C13-substituted Estra-1,3,5 (10) -trien-3-yl-sulfamates, processes for their preparation and pharmaceutical compositions containing them

2001
- 2001-04-24 EP EP01922046A patent/EP1284272A4/en not_active Withdrawn
- 2001-04-24 WO PCT/JP2001/003505 patent/WO2001081364A1/en not_active Application Discontinuation
- 2001-04-24 AU AU2001248849A patent/AU2001248849A1/en not_active Abandoned
- 2001-04-24 US US10/258,454 patent/US6953785B2/en not_active Expired - Fee Related
- 2001-04-24 JP JP2001578452A patent/JPWO2001081364A1/en not_active Withdrawn

Also Published As

Publication number	Publication date
US6953785B2 (en)	2005-10-11
JPWO2001081364A1 (en)	2004-01-08
US20030216362A1 (en)	2003-11-20
EP1284272A4 (en)	2003-09-10
WO2001081364A1 (en)	2001-11-01
EP1284272A1 (en)	2003-02-19

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AU2001230026A1 (en)	2001-08-14	2,4-diaminothiazole derivatives
MXPA01011070A (en)	2003-06-30	Steroid derivatives.
AU2001260939A1 (en)	2001-12-03	Single seed sortation
AU2001243462A1 (en)	2001-09-17	Improved thoraco-lumbo-sacral orthosis
AU2001280099A1 (en)	2002-04-02	4-acylaminopyrazole derivatives
IL152448A0 (en)	2003-05-29	3-nitrogen-6, 7-dioxygen steroid derivatives and pharmaceutical compositions containing the same
AU2001230584A1 (en)	2001-08-20	1h-imidazopyridine derivatives
AU2001258341A1 (en)	2002-01-10	8beta-hydrocarbyl-substituted estratrienes for use as selective estrogens
AU2001284934A1 (en)	2002-02-25	Steroid derived antibiotics
AU2001230537A1 (en)	2001-08-14	Pyridoxazine derivatives
AU2001248849A1 (en)	2001-11-07	Estra-1,3,5(10)-triene derivatives
AU1405101A (en)	2001-05-30	Masks
AU2001281802A1 (en)	2001-12-17	6-phenylpyrrolopyrimidinedione derivatives
AU2001278790A1 (en)	2002-03-04	1h-imidazopyridine derivatives
AU9750398A (en)	1999-05-10	D-homo-9,10-secocholesta-23-yne-3,25-diol derivatives
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AU2001242772A1 (en)	2001-10-03	3-substituted-4-pyrimidone derivatives
AU2001262489A1 (en)	2001-12-03	Triterpenoid derivatives
AU2002218400A1 (en)	2002-06-03	3-substituted 2,7-naphthyridin-1-yl derivatives
AU2002224133A1 (en)	2002-06-24	Remedies for dermatophytosis