AU1123088A - Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy - Google Patents

Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy

Info

Publication number: AU1123088A
Authority: AU; Australia
Prior art keywords: aminoquinuclidine; enantiomers; therapy; preparing; application
Prior art date: 1987-02-04
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU11230/88A

Other versions

AU619731B2 (en

Inventor

Nicole Dorme

Michel Langlois

Alain Renaud

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Synthelabo SA

Original Assignee

Delalande SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-02-04

Filing date

1988-02-03

Publication date

1988-08-11

1988-02-03 Application filed by Delalande SA filed Critical Delalande SA

1988-08-11 Publication of AU1123088A publication Critical patent/AU1123088A/en

1992-02-06 Application granted granted Critical

1992-02-06 Publication of AU619731B2 publication Critical patent/AU619731B2/en

2008-02-03 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Links

HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 title 1
-1 amide derivatives of 3-aminoquinuclidine Chemical class 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
238000002560 therapeutic procedure Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

AU11230/88A 1987-02-04 1988-02-03 Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy Ceased AU619731B2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8701355A FR2610323B1 (en)	1987-02-04	1987-02-04	ENANTIOMERS OF ABSOLUTE CONFIGURATION OF AMINO-3 QUINUCLIDINE AMIDE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION
FR8701355		1987-02-04

Publications (2)

Publication Number	Publication Date
AU1123088A true AU1123088A (en)	1988-08-11
AU619731B2 AU619731B2 (en)	1992-02-06

Family

ID=9347585

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU11230/88A Ceased AU619731B2 (en)	1987-02-04	1988-02-03	Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy

Country Status (7)

Country	Link
EP (1)	EP0280603A1 (en)
JP (1)	JPH0681754B2 (en)
AU (1)	AU619731B2 (en)
DE (1)	DE280603T1 (en)
ES (1)	ES2009718A4 (en)
FR (1)	FR2610323B1 (en)
ZA (1)	ZA88723B (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU618027B2 (en) *	1987-10-16	1991-12-12	A.H. Robins Company, Incorporated	Anxiolytic-r-n-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides
US5360820A (en) *	1991-09-20	1994-11-01	Glaxo Group Limited	Medical use for tachykinin antagonists
US5547964A (en) *	1993-03-19	1996-08-20	Glaxo Group Limited	Medical use for tachykinin antagonists
US7043496B2 (en)	2000-11-10	2006-05-09	Masae Yanagi	Data managing method, data managing system, data managing apparatus, data handling apparatus, computer program, and recording medium

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5126343A (en) *	1989-09-11	1992-06-30	G. D. Searle & Co.	N-azabicyclo [3.3.0]octane amides of aromatic acids
US5290938A (en) *	1989-09-15	1994-03-01	Chiron Laboratories A.S.	Preparation of S-(-)- and R-(+)-N-(quinuclidinyl-3)-amide
NO168529C (en) *	1989-09-15	1992-03-04	Chiron Lab As	PROCEDURE FOR THE PREPARATION OF S - (-) AND R - (+) - N- (QUINUCLIDINYL-3) AMIDES.
IN187238B (en) *	1995-06-30	2002-03-09	Astra Ab

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2529548A1 (en) *	1982-07-02	1984-01-06	Delalande Sa	NOVEL DERIVATIVES OF AMINO-3 QUINUCLIDINE, THEIR PROCESS AND THEIR THERAPEUTIC APPLICATION
US4593034A (en) *	1984-04-06	1986-06-03	A. H. Robins Company, Inc.	2-alkoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamides and thiobenzamides
US4870181A (en) *	1985-02-04	1989-09-26	A. H. Robins Company, Incorporated	Process for the preparation of 2-alkoxy-N-(1-azabicyclo[2.2.2])octan-3-yl)aminobenzamides
JPS63146850A (en) *	1986-11-12	1988-06-18	メルク　エンド　カムパニー　インコーポレーテツド	Renin inhibitor having phenylalanyl-histidine substitute component
GB8629962D0 (en) *	1986-12-16	1987-01-28	Naylor R J	Benzamides & thiobenzamides

1987
- 1987-02-04 FR FR8701355A patent/FR2610323B1/en not_active Expired
1988
- 1988-02-02 ZA ZA88723A patent/ZA88723B/en unknown
- 1988-02-03 EP EP88400253A patent/EP0280603A1/en not_active Withdrawn
- 1988-02-03 AU AU11230/88A patent/AU619731B2/en not_active Ceased
- 1988-02-03 ES ES88400253T patent/ES2009718A4/en active Pending
- 1988-02-03 DE DE198888400253T patent/DE280603T1/en active Pending
- 1988-02-04 JP JP63022969A patent/JPH0681754B2/en not_active Expired - Lifetime

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU618027B2 (en) *	1987-10-16	1991-12-12	A.H. Robins Company, Incorporated	Anxiolytic-r-n-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides
US5360820A (en) *	1991-09-20	1994-11-01	Glaxo Group Limited	Medical use for tachykinin antagonists
US5538982A (en) *	1991-09-20	1996-07-23	Glaxo Group Limited	Medical use for tachykinin antagonists
US5798363A (en) *	1991-09-20	1998-08-25	Glaxo Group Limited	Use for tachykinin antagonists to treat emesis
US7214692B2 (en)	1991-09-20	2007-05-08	Glaxo Group Limited	Medical use for tachykinin antagonists
US7342028B2 (en)	1991-09-20	2008-03-11	Glaxo Group Limited	Medical use for tachykinin antagonists
US5547964A (en) *	1993-03-19	1996-08-20	Glaxo Group Limited	Medical use for tachykinin antagonists
US6329394B1 (en)	1993-03-19	2001-12-11	Glaxo Group Limited	Medical use for tachykinin antagonists
US7043496B2 (en)	2000-11-10	2006-05-09	Masae Yanagi	Data managing method, data managing system, data managing apparatus, data handling apparatus, computer program, and recording medium

Also Published As

Publication number	Publication date
JPS63196583A (en)	1988-08-15
JPH0681754B2 (en)	1994-10-19
FR2610323A1 (en)	1988-08-05
ZA88723B (en)	1988-10-26
AU619731B2 (en)	1992-02-06
EP0280603A1 (en)	1988-08-31
DE280603T1 (en)	1989-10-05
ES2009718A4 (en)	1989-10-16
FR2610323B1 (en)	1989-06-23

Similar Documents

Publication	Publication Date	Title
AU3347389A (en)	1989-10-16	Medical material and process for their production
AU2454788A (en)	1989-05-04	N-substituted derivatives of 1-desoxynojirimycin 1- desoxymannojirimycin, processes for their preparation and their use in medicaments
HUT44779A (en)	1988-04-28	Process for producing imidazole derivatives and pharmaceutical preparations comprising the same
AU6112790A (en)	1991-02-28	N-(substituted benzyloxy)imine derivatives, process for the production thereof, use thereof, and method of use thereof
MY116593A (en)	2004-02-28	Process for the preparation of o-demethyltramadol enantiomers
HU912013D0 (en)	1991-12-30	Process for the production of benzopyrane derivatives and their heterocyclic analogues, antiyschemic medical preparations
HU910929D0 (en)	1991-10-28	Process for the production of 2,8-dioxa-bicyclo/3,2,1/octane derivatives and medical preparations containing them
AU591719B2 (en)	1989-12-14	Benzylamine derivatives, process for production thereof, and use thereof
AU2597688A (en)	1989-06-29	2,2-difluorocyclopropylethane derivatives, process for their preparation and their use as pesticides
HU9101576D0 (en)	1991-11-28	Process for the production of medical preparations for decreasing heart-fibrillation
AU2988789A (en)	1989-08-17	Process for the preparation of activated carbon
AU3968889A (en)	1990-02-05	Process and apparatus for the preparation of balloons
AU1123088A (en)	1988-08-11	Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy
HU911811D0 (en)	1991-12-30	Process for the production of acylized alpha, omega-amino-alcoholic derivatives and for using them in pesticide substances
AU2593188A (en)	1989-06-01	Iminophenylthiazolidines, process of preparation and method of use
HUT46644A (en)	1988-11-28	Process for producing propylophenone derivatives and pharmaceutical compositions comprising the same
AU1136088A (en)	1988-08-11	Substituted amine derivatives, their production and use
AU1313488A (en)	1988-10-06	Process for the preparation of nitroethene derivatives
AU2501288A (en)	1989-05-11	Sialocylglycerolipids and method for preparing the same
AU4178189A (en)	1990-05-17	Therapeutic agent for aids and process for preparing it
HU912213D0 (en)	1991-12-30	Process for the production of amino-diol derivatives and medical preparations containing them
AU2886089A (en)	1989-08-10	Process for preparing n-phosphono-methyl-imino-diacetic acid and acid chloride
IL86416A (en)	1993-07-08	Process for the preparation of 2-quinoxalinol derivatives
AU1289388A (en)	1988-09-29	Process for the preparation of polyamines and their use for production of polyurethanes
AU4827690A (en)	1990-08-01	Apparatus and method for the production of molded articles