ATE438656T1 - AN DER 4ß- BZW. 4'-STELLUNG SUBSTITUIERTES AVERMECTIN UND AVERMECTIN-MONOSACCHARID - Google Patents

AN DER 4ß- BZW. 4'-STELLUNG SUBSTITUIERTES AVERMECTIN UND AVERMECTIN-MONOSACCHARID

Info

Publication number: ATE438656T1
Authority: AT; Austria
Prior art keywords: avermectin; monosaccharide; position substituted; substituted; avermectin monosaccharide
Prior art date: 2004-04-07

Application number

AT05715877T

Other languages

English (en)

Inventor

Pierre Joseph Marcel Jung

Thomas Pitterna

Laura Quaranta

Ottmar Franz Hueter

Fiona Murphy-Kessabi

Original Assignee

Syngenta Participations Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-04-07

Filing date

2005-03-09

Publication date

2009-08-15

2005-03-09 Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag

2009-08-15 Application granted granted Critical

2009-08-15 Publication of ATE438656T1 publication Critical patent/ATE438656T1/de

Links

239000005660 Abamectin Substances 0.000 title 2
-1 AVERMECTIN MONOSACCHARIDE Chemical class 0.000 title 1
RRZXIRBKKLTSOM-XPNPUAGNSA-N avermectin B1a Chemical class C1=C[C@H](C)[C@@H]([C@@H](C)CC)O[C@]11O[C@H](C\C=C(C)\[C@@H](O[C@@H]2O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C2)[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 RRZXIRBKKLTSOM-XPNPUAGNSA-N 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

Life Sciences & Earth Sciences (AREA)
Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Biotechnology (AREA)
Environmental Sciences (AREA)
Zoology (AREA)
Wood Science & Technology (AREA)
Dentistry (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Veterinary Medicine (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Medicinal Chemistry (AREA)
Tropical Medicine & Parasitology (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Plural Heterocyclic Compounds (AREA)

AT05715877T 2004-04-07 2005-03-09 AN DER 4ß- BZW. 4'-STELLUNG SUBSTITUIERTES AVERMECTIN UND AVERMECTIN-MONOSACCHARID ATE438656T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP04008413		2004-04-07
PCT/EP2005/002489 WO2005097816A1 (en)	2004-04-07	2005-03-09	Avermectin and avermectin monosaccharide substituted in the 4”- and 4’- position respectively

Publications (1)

Publication Number	Publication Date
ATE438656T1 true ATE438656T1 (de)	2009-08-15

Family

ID=34924568

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT05715877T ATE438656T1 (de)	2004-04-07	2005-03-09	AN DER 4ß- BZW. 4'-STELLUNG SUBSTITUIERTES AVERMECTIN UND AVERMECTIN-MONOSACCHARID

Country Status (9)

Country	Link
US (1)	US7687470B2 (de)
EP (1)	EP1737876B1 (de)
JP (1)	JP5046116B2 (de)
AR (1)	AR049489A1 (de)
AT (1)	ATE438656T1 (de)
DE (1)	DE602005015835D1 (de)
ES (1)	ES2331421T3 (de)
TW (1)	TW200538461A (de)
WO (1)	WO2005097816A1 (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CR6574A (es) *	2001-02-27	2004-10-28	Syngenta Participations Ag	Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) *	2001-02-27	2004-04-28	Syngenta Participations Ag	Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) *	2001-08-28	2004-09-15	Syngenta Participations Ag	Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
TW200407330A (en) *	2002-05-07	2004-05-16	Syngenta Participations Ag	4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0302310D0 (en) *	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) *	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) *	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302547D0 (en) *	2003-02-04	2003-03-12	Syngenta Participations Ag	Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0320176D0 (en)	2003-08-28	2003-10-01	Syngenta Participations Ag	Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
CN103459370A (zh) *	2011-01-25	2013-12-18	拜耳知识产权有限责任公司	制备1-h-吡咯烷-2,4-二酮衍生物的方法
CN103396465B (zh) *	2013-07-19	2016-01-20	中国农业科学院植物保护研究所	一种阿维菌素烟碱二效价化合物及其制备和应用
US10118890B2 (en)	2014-10-10	2018-11-06	The Research Foundation For The State University Of New York	Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
CN104402954A (zh) *	2014-11-28	2015-03-11	大庆志飞生物化工有限公司	甲胺基阿维菌素单糖化合物及其制备方法和用途
CN105037467A (zh) *	2015-05-29	2015-11-11	河北威远生化农药有限公司	4”-脱氧-4”烷基化或酰基化胺基阿维菌素B2a/2b衍生物及其制备方法和用途
CN106995476B (zh) *	2017-05-16	2018-03-13	河北美荷药业有限公司	一种甲氨基阿维菌素b2苯甲酸盐的制备方法
CN109485683A (zh) *	2018-11-27	2019-03-19	齐鲁晟华制药有限公司	一种含氟系列阿维菌素衍生物及其制备方法
CN113150053A (zh) *	2020-01-22	2021-07-23	华东理工大学	偶氮苯类阿维菌素衍生物及其制备方法和应用
CN115403644B (zh) *	2022-09-01	2024-04-05	石家庄学院	一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4873224A (en) *	1988-05-23	1989-10-10	Merck & Co., Inc.	Avermectin derivatives
NZ231773A (en) *	1988-12-23	1992-09-25	Merck & Co Inc	Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
GB9201505D0 (en) *	1992-01-24	1992-03-11	Pfizer Ltd	Antiparasitic agents
CN100436589C (zh) *	2001-06-22	2008-11-26	印度技术研究院	一种通过共培养制备五倍子酸的方法
GB0302308D0 (en) *	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) *	2003-01-31	2003-03-05	Syngenta Participations Ag	Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302548D0 (en) *	2003-02-04	2003-03-12	Syngenta Participations Ag	Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
GB0302547D0 (en) *	2003-02-04	2003-03-12	Syngenta Participations Ag	Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0313937D0 (en) *	2003-06-16	2003-07-23	Syngenta Participations Ag	Avermectin B1 monosaccharide derivatives having an aminosulfonyloxy substituentin the 4'-position

2005
- 2005-03-07 TW TW094106807A patent/TW200538461A/zh unknown
- 2005-03-09 WO PCT/EP2005/002489 patent/WO2005097816A1/en active Application Filing
- 2005-03-09 EP EP05715877A patent/EP1737876B1/de active Active
- 2005-03-09 US US10/599,671 patent/US7687470B2/en active Active
- 2005-03-09 ES ES05715877T patent/ES2331421T3/es active Active
- 2005-03-09 JP JP2007506677A patent/JP5046116B2/ja active Active
- 2005-03-09 AT AT05715877T patent/ATE438656T1/de not_active IP Right Cessation
- 2005-03-09 DE DE602005015835T patent/DE602005015835D1/de active Active
- 2005-04-04 AR ARP050101317A patent/AR049489A1/es not_active Application Discontinuation

Also Published As

Publication number	Publication date
JP2007532497A (ja)	2007-11-15
AR049489A1 (es)	2006-08-09
ES2331421T3 (es)	2010-01-04
EP1737876B1 (de)	2009-08-05
DE602005015835D1 (de)	2009-09-17
EP1737876A1 (de)	2007-01-03
US7687470B2 (en)	2010-03-30
JP5046116B2 (ja)	2012-10-10
WO2005097816A1 (en)	2005-10-20
US20080051353A1 (en)	2008-02-28
TW200538461A (en)	2005-12-01

Legal Events

Date	Code	Title	Description
2010-02-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
ATE438656T1 (de)	2009-08-15	AN DER 4ß- BZW. 4'-STELLUNG SUBSTITUIERTES AVERMECTIN UND AVERMECTIN-MONOSACCHARID
ATE506362T1 (de)	2011-05-15	1-aza-bicycloä3.3.1ünonane
ATE349457T1 (de)	2007-01-15	Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen
DK1592700T3 (da)	2008-08-04	Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber
ATE391133T1 (de)	2008-04-15	Avermectine und avermectinmonosaccharide substituiert in der 4'- und 4''-stellung mit pestiziden eigenschaften
ES1048464Y (es)	2001-12-16	Mariposa de somier perfeccionada.
ES1050481Y (es)	2002-11-16	Pieza de construccion.
ES1050026Y (es)	2002-06-16	Disposicion de puerta ignifuga perfeccionada.
ES1050301Y (es)	2002-07-01	Ambientador perfeccionado.
김대원	2004	On the class of generalized paranormal operators
ES1048567Y (es)	2001-12-16	Curvatubos de carraca perfeccionado.
FR2810360B1 (fr)	2002-12-27	Cremone, cremone-serrure ou similaire
ES1050018Y (es)	2002-06-16	Macetero perfeccionado.
ES1048873Y (es)	2002-02-16	Descapsulador perfeccionado.
ES1049872Y (es)	2002-06-01	Azada perfeccionada.
ITSV20030024A1 (it)	2004-11-23	Porta, portone sezionale o simili.
ES1049899Y (es)	2002-06-01	Cenicero perfeccionado.
ITPG20050016A1 (it)	2006-09-16	Cosmeticus bibbia n.2
ES1055975Y (es)	2004-06-01	Ambientador perfeccionado.
ES1048804Y (es)	2002-02-16	Pliego autocopiativo perfeccionado.
ES1049516Y (es)	2002-08-01	Pupitre universitario perfeccionado.
ES1053939Y (es)	2003-09-16	Vitrina frigorifica perfeccionada.
ES1048763Y (es)	2002-02-01	Cortadora-ingletadora perfeccionada.
ES1049809Y (es)	2002-05-16	Humidificador-fitosanitario perfeccionado.
ES1048870Y (es)	2002-02-16	Capirote perfeccionado.