ATE291016T1 - Amidinophenylalaninderivate als thrombininhibitoren - Google Patents
Amidinophenylalaninderivate als thrombininhibitorenInfo
- Publication number
- ATE291016T1 ATE291016T1 AT01272199T AT01272199T ATE291016T1 AT E291016 T1 ATE291016 T1 AT E291016T1 AT 01272199 T AT01272199 T AT 01272199T AT 01272199 T AT01272199 T AT 01272199T AT E291016 T1 ATE291016 T1 AT E291016T1
- Authority
- AT
- Austria
- Prior art keywords
- thrombin inhibitors
- amidinophenylalanine derivatives
- amidinophenylalanine
- derivatives
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/48—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom
- C07C311/49—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom to nitrogen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200000326A SI20743A (sl) | 2000-12-22 | 2000-12-22 | Novi trombinski inhibitorji |
PCT/IB2001/002600 WO2002051824A1 (en) | 2000-12-22 | 2001-12-20 | Amidinophenylalanine derivatives as thrombin inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE291016T1 true ATE291016T1 (de) | 2005-04-15 |
Family
ID=20432799
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT01272199T ATE291016T1 (de) | 2000-12-22 | 2001-12-20 | Amidinophenylalaninderivate als thrombininhibitoren |
Country Status (10)
Country | Link |
---|---|
US (2) | US7285547B2 (de) |
EP (1) | EP1355894B1 (de) |
JP (1) | JP4390453B2 (de) |
AT (1) | ATE291016T1 (de) |
DE (1) | DE60109498T2 (de) |
DK (1) | DK1355894T3 (de) |
ES (1) | ES2240345T3 (de) |
PT (1) | PT1355894E (de) |
SI (1) | SI20743A (de) |
WO (1) | WO2002051824A1 (de) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0507577D0 (en) | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
GB0523539D0 (en) * | 2005-11-18 | 2005-12-28 | Lek Tovarna Farmacevtskih | New use of organic compounds |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9322976D0 (en) | 1993-11-08 | 1994-01-05 | Pfizer Ltd | Therapeutic agents |
-
2000
- 2000-12-22 SI SI200000326A patent/SI20743A/sl not_active IP Right Cessation
-
2001
- 2001-12-20 DE DE60109498T patent/DE60109498T2/de not_active Expired - Lifetime
- 2001-12-20 EP EP01272199A patent/EP1355894B1/de not_active Expired - Lifetime
- 2001-12-20 PT PT01272199T patent/PT1355894E/pt unknown
- 2001-12-20 ES ES01272199T patent/ES2240345T3/es not_active Expired - Lifetime
- 2001-12-20 WO PCT/IB2001/002600 patent/WO2002051824A1/en active IP Right Grant
- 2001-12-20 AT AT01272199T patent/ATE291016T1/de active
- 2001-12-20 US US10/433,358 patent/US7285547B2/en not_active Expired - Fee Related
- 2001-12-20 DK DK01272199T patent/DK1355894T3/da active
- 2001-12-20 JP JP2002552919A patent/JP4390453B2/ja not_active Expired - Fee Related
-
2007
- 2007-09-12 US US11/854,532 patent/US20080004256A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1355894A1 (de) | 2003-10-29 |
JP4390453B2 (ja) | 2009-12-24 |
SI20743A (sl) | 2002-06-30 |
JP2004516317A (ja) | 2004-06-03 |
US7285547B2 (en) | 2007-10-23 |
US20040048851A1 (en) | 2004-03-11 |
DK1355894T3 (da) | 2005-07-11 |
DE60109498D1 (en) | 2005-04-21 |
US20080004256A1 (en) | 2008-01-03 |
ES2240345T3 (es) | 2005-10-16 |
WO2002051824A1 (en) | 2002-07-04 |
PT1355894E (pt) | 2005-08-31 |
DE60109498T2 (de) | 2006-04-13 |
EP1355894B1 (de) | 2005-03-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification |
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