AR231533A1 - Un procedimiento para preparar derivados de 3-amino-alquel-1h-indol-5-il metano-sulfonamida - Google Patents

Un procedimiento para preparar derivados de 3-amino-alquel-1h-indol-5-il metano-sulfonamida

Info

Publication number
AR231533A1
AR231533A1 AR290026A AR29002682A AR231533A1 AR 231533 A1 AR231533 A1 AR 231533A1 AR 290026 A AR290026 A AR 290026A AR 29002682 A AR29002682 A AR 29002682A AR 231533 A1 AR231533 A1 AR 231533A1
Authority
AR
Argentina
Prior art keywords
alquel
indol
methane
amino
preparing
Prior art date
Application number
AR290026A
Other languages
English (en)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of AR231533A1 publication Critical patent/AR231533A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
AR290026A 1980-08-12 1982-07-20 Un procedimiento para preparar derivados de 3-amino-alquel-1h-indol-5-il metano-sulfonamida AR231533A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8026288 1980-08-12

Publications (1)

Publication Number Publication Date
AR231533A1 true AR231533A1 (es) 1984-12-28

Family

ID=10515412

Family Applications (1)

Application Number Title Priority Date Filing Date
AR290026A AR231533A1 (es) 1980-08-12 1982-07-20 Un procedimiento para preparar derivados de 3-amino-alquel-1h-indol-5-il metano-sulfonamida

Country Status (28)

Country Link
US (2) US4672067A (es)
JP (1) JPS5759864A (es)
AR (1) AR231533A1 (es)
AT (1) AT381304B (es)
AU (1) AU548270B2 (es)
BE (1) BE889930A (es)
CA (2) CA1169429A (es)
CH (1) CH651550A5 (es)
DE (1) DE3131748A1 (es)
DK (1) DK157680C (es)
ES (2) ES8300700A1 (es)
FI (1) FI812475L (es)
FR (1) FR2488605A1 (es)
GB (1) GB2081717B (es)
GR (1) GR74536B (es)
IE (1) IE51492B1 (es)
IL (1) IL63541A (es)
IT (1) IT1171451B (es)
LU (1) LU83546A1 (es)
MY (1) MY8600577A (es)
NL (1) NL8103768A (es)
NO (1) NO812722L (es)
NZ (1) NZ197997A (es)
PH (1) PH17428A (es)
PT (1) PT73503B (es)
SE (1) SE454881B (es)
ZA (1) ZA815539B (es)
ZW (1) ZW19381A1 (es)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
GB8332434D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Production of chemical compounds
HU196752B (en) * 1983-12-06 1989-01-30 Glaxo Group Ltd Process for production of medical compositions containing indole-derivatives and these compounds
GB8332437D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
GB8600398D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
US5270333A (en) * 1986-01-28 1993-12-14 Glaxo Group Limited Indole derivatives
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
DE3613623A1 (de) * 1986-04-23 1987-10-29 Bayer Ag N-dihydroindolylethyl-sulfonamide
GB8615599D0 (en) * 1986-06-26 1986-07-30 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
GB8819024D0 (en) * 1988-08-10 1988-09-14 Glaxo Group Ltd Chemical compounds
CA2042295A1 (fr) * 1990-05-15 1991-11-16 Jacques Chauveau Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant
ATE156823T1 (de) * 1990-06-07 1997-08-15 Zeneca Ltd Therapeutische heterocyclische verbindungen
GB9022250D0 (en) * 1990-10-12 1990-11-28 Glaxo Group Ltd Medicaments
US5578612A (en) * 1990-10-15 1996-11-26 Pfizer Inc. Indole derivatives
US5607951A (en) * 1990-10-15 1997-03-04 Pfizer Inc Indole derivatives
US5545644A (en) * 1990-10-15 1996-08-13 Pfizer Inc. Indole derivatives
DE9190141U1 (es) * 1990-10-15 1993-07-15 Pfizer, Inc., New York, N.Y., Us
US5559129A (en) * 1990-10-15 1996-09-24 Pfizer Inc Indole derivatives
US5559246A (en) * 1990-10-15 1996-09-24 Pfizer Inc. Indole derivatives
SK278998B6 (sk) * 1991-02-01 1998-05-06 Merck Sharp & Dohme Limited Deriváty imidazolu, triazolu a tetrazolu, spôsob i
GB9103770D0 (en) * 1991-02-22 1991-04-10 Glaxo Group Ltd Chemical compounds
ES2033578B1 (es) * 1991-06-06 1995-01-16 Quimica Sint S A Con El 50 Procedimiento para la obtencion de 3-(2-(dimetilamino)etil)-n-metil-1h-indol-5-metanosulfonamida.
ES2033577B1 (es) * 1991-06-06 1995-01-16 Quimica Sint S A Con El 50 Procedimiento para la obtencion de la 2-carboxi-3-(2-(dimetilamino)etil)-n-metil-1h-indol-5-metanosulfonamida y sus esteres alquilicos inferiores.
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
IL106445A (en) * 1992-07-30 1998-01-04 Merck Sharp & Dohme History of 1,2,4-Trans-Triazole 4-Transform, Preparation and Pharmaceutical Preparations Containing Them
AU686654B2 (en) * 1993-08-31 1998-02-12 Pfizer Inc. 5-arylindole derivatives
US5468768A (en) * 1994-01-06 1995-11-21 Bristol-Myers Squibb Company Antimigraine derivatives of indolylcycloalkanylamines
GB9417310D0 (en) * 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
WO1997013512A1 (en) * 1995-10-10 1997-04-17 Eli Lilly And Company N-[2-substituted-3-(2-aminoethyl)-1h-indol-5-yl]-amides: new 5-ht1f agonists
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
US5994352A (en) * 1998-11-13 1999-11-30 Pfizer Inc. 5-arylindole derivatives
WO2002079153A1 (en) * 2001-03-28 2002-10-10 Biocatalytics, Inc. Method for producing tryptamine derivatives
US7026364B2 (en) * 2001-04-13 2006-04-11 Organo Corporation Ion exchanger
ATE489138T1 (de) * 2005-04-13 2010-12-15 Neuraxon Inc Substituierte indolverbindungen mit nos-hemmender aktivität
CA2991108A1 (en) 2015-07-02 2017-01-05 Civitas Therapeutics, Inc. Triptan powders for pulmonary delivery

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2870162A (en) * 1954-04-28 1959-01-20 Upjohn Co Production of certain tryptamines and compounds produced in the process
BE632051A (fr) * 1963-05-08 1963-11-18 Sandoz Sa Nouveaux dérivés de l'indole et leur préparation.
CH442303A (de) * 1964-06-26 1967-08-31 Sandoz Ag Verfahren zur Herstellung von neuen Indol-Derivaten
US3472870A (en) * 1966-08-29 1969-10-14 Mead Johnson & Co Sulfonamidotryptamines
FR2334358A1 (fr) * 1975-12-12 1977-07-08 Sogeras Nouveaux medicaments derives de l'indole
US4180509A (en) * 1977-07-01 1979-12-25 Merrell Toraude Et Compagnie α-Ethynyl tryptophanes
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds

Also Published As

Publication number Publication date
GB2081717B (en) 1983-09-28
NZ197997A (en) 1985-08-16
ATA352881A (de) 1986-02-15
ES8404327A1 (es) 1984-04-16
PT73503B (en) 1983-09-14
FR2488605A1 (fr) 1982-02-19
ES504695A0 (es) 1982-11-01
IL63541A (en) 1985-08-30
JPS5759864A (en) 1982-04-10
BE889930A (fr) 1982-02-11
GB2081717A (en) 1982-02-24
JPH0148895B2 (es) 1989-10-20
GR74536B (es) 1984-06-29
PH17428A (en) 1984-08-20
ZW19381A1 (en) 1983-03-09
DK157680B (da) 1990-02-05
MY8600577A (en) 1986-12-31
DE3131748A1 (de) 1982-04-01
FR2488605B1 (es) 1984-11-16
FI812475L (fi) 1982-02-13
PT73503A (en) 1981-09-01
NO812722L (no) 1982-02-15
IE51492B1 (en) 1987-01-07
US4636521A (en) 1987-01-13
CA1169077A (en) 1984-06-12
DE3131748C2 (es) 1992-04-23
ZA815539B (en) 1983-03-30
LU83546A1 (fr) 1983-06-08
DK357181A (da) 1982-02-13
US4672067A (en) 1987-06-09
NL8103768A (nl) 1982-03-01
SE8104782L (sv) 1982-02-13
AT381304B (de) 1986-09-25
AU548270B2 (en) 1985-12-05
SE454881B (sv) 1988-06-06
DK157680C (da) 1990-07-09
AU7399681A (en) 1982-02-18
IE811831L (en) 1982-02-12
ES8300700A1 (es) 1982-11-01
IT8149086A0 (it) 1981-08-11
ES513935A0 (es) 1984-04-16
CA1169429A (en) 1984-06-19
CH651550A5 (fr) 1985-09-30
IT1171451B (it) 1987-06-10

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