AR217688A1 - PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL - Google Patents

PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL

Info

Publication number
AR217688A1
AR217688A1 AR271956A AR27195678A AR217688A1 AR 217688 A1 AR217688 A1 AR 217688A1 AR 271956 A AR271956 A AR 271956A AR 27195678 A AR27195678 A AR 27195678A AR 217688 A1 AR217688 A1 AR 217688A1
Authority
AR
Argentina
Prior art keywords
hexahidro
pirido
indol
trans
aryl
Prior art date
Application number
AR271956A
Other languages
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR217688A1 publication Critical patent/AR217688A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR271956A 1977-05-23 1978-04-28 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL AR217688A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US79939277A 1977-05-23 1977-05-23

Publications (1)

Publication Number Publication Date
AR217688A1 true AR217688A1 (en) 1980-04-15

Family

ID=25175793

Family Applications (2)

Application Number Title Priority Date Filing Date
AR271956A AR217688A1 (en) 1977-05-23 1978-04-28 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL
AR276191A AR221721A1 (en) 1977-05-23 1979-04-16 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR276191A AR221721A1 (en) 1977-05-23 1979-04-16 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4, A 5,9B-HEXAHIDRO-1H-PIRIDOL (4,3-B) -INDOL, INTERMEDIARIES USED THEREOF AND PROCEDURE FOR PREPARING SUCH INTERMEDIARIES

Country Status (31)

Country Link
JP (1) JPS53144600A (en)
AR (2) AR217688A1 (en)
AT (1) AT368995B (en)
AU (1) AU499618B1 (en)
BE (1) BE867249A (en)
CA (1) CA1094071A (en)
CH (1) CH634321A5 (en)
CS (1) CS207612B2 (en)
DD (4) DD146186A5 (en)
DE (1) DE2822465C2 (en)
DK (1) DK226678A (en)
EG (1) EG13590A (en)
FI (1) FI63402C (en)
FR (1) FR2392023A1 (en)
GB (1) GB1586655A (en)
GR (1) GR69985B (en)
HU (3) HU185009B (en)
IE (1) IE46975B1 (en)
IL (1) IL54755A (en)
IT (1) IT1096307B (en)
LU (1) LU79684A1 (en)
NL (1) NL7804210A (en)
NO (2) NO150204C (en)
NZ (1) NZ187333A (en)
PH (1) PH13756A (en)
PL (5) PL114547B1 (en)
PT (1) PT68058B (en)
SE (2) SE441448B (en)
SU (4) SU873883A3 (en)
YU (4) YU91478A (en)
ZA (1) ZA782918B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) * 1982-05-17 1984-05-29 Pfizer Inc. Process for preparing carboline derivatives and compounds used in their preparation
RU2106864C1 (en) * 1995-10-23 1998-03-20 Николай Серафимович Зефиров New approach to treatment of alzheimer's disease
SE9604786D0 (en) * 1996-12-20 1996-12-20 Astra Pharma Inc New compounds
US6974825B1 (en) 1996-12-20 2005-12-13 Astrazeneca Canada Inc. Compounds with analgesic effect
SE9904675D0 (en) 1999-12-20 1999-12-20 Astra Pharma Inc Novel compounds
SE0101773D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101770D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101769D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds
SE0101771D0 (en) 2001-05-18 2001-05-18 Astrazeneca Ab Novel compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR205452A1 (en) * 1973-12-06 1976-05-07 Endo Lab METHOD TO PREPARE NEW TRANS-2, 3, 4, 4A, 5, 9B-HEXAHYDRO-5-PHENYL-1H-PYRID (4,3-B) INDOLES
JPS50126699A (en) * 1974-03-20 1975-10-04
US4001263A (en) * 1974-04-01 1977-01-04 Pfizer Inc. 5-Aryl-1,2,3,4-tetrahydro-γ-carbolines

Also Published As

Publication number Publication date
SU818484A3 (en) 1981-03-30
DE2822465A1 (en) 1978-11-30
IL54755A0 (en) 1978-07-31
SE448459B (en) 1987-02-23
SE441448B (en) 1985-10-07
FI781612A (en) 1978-11-24
ZA782918B (en) 1979-06-27
PT68058B (en) 1979-10-24
NO150204B (en) 1984-05-28
HU185009B (en) 1984-11-28
DD145537A5 (en) 1980-12-17
DK226678A (en) 1978-11-24
CH634321A5 (en) 1983-01-31
SE8305917D0 (en) 1983-10-27
IE46975B1 (en) 1983-11-16
GB1586655A (en) 1981-03-25
BE867249A (en) 1978-11-20
PL116944B1 (en) 1981-07-31
DD146186A5 (en) 1981-01-28
AU499618B1 (en) 1979-04-26
YU221782A (en) 1983-01-21
EG13590A (en) 1982-03-31
FI63402C (en) 1983-06-10
PL114541B1 (en) 1981-02-28
SU843749A3 (en) 1981-06-30
DD138321A5 (en) 1979-10-24
PL117107B1 (en) 1981-07-31
ATA369678A (en) 1982-04-15
PL206903A1 (en) 1979-10-22
SE7803625L (en) 1978-11-24
NO151862B (en) 1985-03-11
JPS53144600A (en) 1978-12-15
NO150204C (en) 1984-09-05
NO831790L (en) 1978-11-24
HU188802B (en) 1986-05-28
IT7823673A0 (en) 1978-05-22
SU873883A3 (en) 1981-10-15
LU79684A1 (en) 1979-12-06
YU221682A (en) 1983-01-21
SU841589A3 (en) 1981-06-23
IT1096307B (en) 1985-08-26
IL54755A (en) 1981-02-27
PL114547B1 (en) 1981-02-28
NO151862C (en) 1985-06-19
CA1094071A (en) 1981-01-20
YU40796B (en) 1986-06-30
GR69985B (en) 1982-07-22
IE781013L (en) 1978-11-23
FR2392023B1 (en) 1980-11-07
JPS5711912B2 (en) 1982-03-08
AT368995B (en) 1982-11-25
SE8305917L (en) 1983-10-27
FI63402B (en) 1983-02-28
DD145536A5 (en) 1980-12-17
PT68058A (en) 1978-06-01
CS207612B2 (en) 1981-08-31
AR221721A1 (en) 1981-03-13
FR2392023A1 (en) 1978-12-22
NL7804210A (en) 1978-11-27
NZ187333A (en) 1984-05-31
NO781770L (en) 1978-11-24
HU187782B (en) 1986-02-28
YU91478A (en) 1983-01-21
PH13756A (en) 1980-09-17
YU221882A (en) 1983-01-21
DE2822465C2 (en) 1986-08-28

Similar Documents

Publication Publication Date Title
AR223958A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF (4-HYDROXYPROLROLIDIN-2-ON-1-IL) -ACILAMIDE
AR219560A1 (en) PROCEDURE FOR THE PREPARATION OF 5,5-DIMETHYL-HYDANTOINE DERIVATIVES
MX5527E (en) PROCEDURE FOR THE PREPARATION OF CARBOESTIRILE DERIVATIVES
AR219734A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF (4-HYDROXYPROLROLIDIN-2-ON-1-IL) -ACILAMIDE
AR221851A1 (en) PROCEDURE FOR THE PREPARATION OF 4-PIPERIDINE-6,7-DIALCOXY-QUINAZOLINE DERIVATIVES
AR216937A1 (en) PROCEDURE FOR THE PREPARATION OF 1,1,1,2-TETRAFLUORETHANE
AR224110A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 5 (6) -BENZIMIDAZOLES
AR220675A1 (en) PROCEDURE FOR THE PREPARATION OF SUBSTITUTED DERIVATIVES OF PIRIDO (1,2-A) PIRIMIDINAS
MX5479E (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 1-OXADETIACEFALOSPORINAS
MX5256E (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 20,21-DINOREBURNAMENINE
AR217688A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRANS-2-SUBSTITUTED-5-ARYL-2,3,4,4A, 5,9B-HEXAHIDRO-1H-PIRIDO (4,3-B) -INDOL
AR218296A1 (en) PROCEDURE FOR THE PREPARATION OF NEW DERIVATIVES OF 14-BETA-AMINO-MORPHINE
AR218498A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 1,3-DIFENOXIPROPAN-2-ONA
ES497530A0 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2,3-INDO- LEDIONA
MX5046E (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF (2,3-B) PIRIDO- (1,5) -BENZOTIAZEPINA, REPLACED IN POSITION 5
AR224501A1 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TIENO- (3,2-C) -PIRIDINE
ES499691A0 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 5,11-DIHI-DRO-6H-PIRIDO (2,3-B) (1,4) -BENZODIAZEPIN-6-ONA
ES493931A0 (en) PROCEDURE FOR THE PREPARATION OF NEW DERIVATIVES OF 3,4,5-TRIMETOXI-CINAMOIL-PIPERAZINE
AR221215A1 (en) PROCEDURE FOR THE PREPARATION OF SUBSTITUTED CHLOROACETHANILIDES
MX6009E (en) PROCEDURE FOR THE PREPARATION OF TETRAHIDRO-1,3,5-TIADIAZIN-4-ONAS
AR225415A1 (en) PROCEDURE FOR THE OBTAINING OF NEW DERIVATIVES OF PIRIDO (2,1-B) QUINAZOLINA
ES501213A0 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2,3,4,5- TETRAHIDRO-1-BENZOXEPIN-3,5-DIONA
MX5933E (en) PROCEDURE FOR THE PREPARATION OF 4,5-DICICLO-2- (TIOSUBSTITUIDOS) -IMIDAZOLES
AR230835A1 (en) PROCEDURE FOR THE OBTAINING OF DERIVATIVES OF 2,1,3-TIADIAZIN-4-ONA-2,2-DIOXIDO
ES494286A0 (en) PROCEDURE FOR THE PREPARATION OF NEW DERIVATIVES 1,1,2-TRI- FENILPROPANOS AND -PROPENOS