AR207799A1 - Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos - Google Patents

Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos

Info

Publication number
AR207799A1
AR207799A1 AR261449A AR26144975A AR207799A1 AR 207799 A1 AR207799 A1 AR 207799A1 AR 261449 A AR261449 A AR 261449A AR 26144975 A AR26144975 A AR 26144975A AR 207799 A1 AR207799 A1 AR 207799A1
Authority
AR
Argentina
Prior art keywords
azaciclo
phenylindoles
substitute
prepare
procedure
Prior art date
Application number
AR261449A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US456641A external-priority patent/US3925409A/en
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR207799A1 publication Critical patent/AR207799A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
AR261449A 1974-04-01 1975-01-01 Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos AR207799A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45664074A 1974-04-01 1974-04-01
US456641A US3925409A (en) 1974-04-01 1974-04-01 4-Aryl-1,2,3,4-tetrahydropyrrolo{8 3,4-b{9 indoles

Publications (1)

Publication Number Publication Date
AR207799A1 true AR207799A1 (es) 1976-10-29

Family

ID=27038317

Family Applications (2)

Application Number Title Priority Date Filing Date
AR258188A AR206812A1 (es) 1974-04-01 1975-01-01 Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica
AR261449A AR207799A1 (es) 1974-04-01 1975-01-01 Procedimiento para preparar azaciclo(3,4-a)-n-fenilindoles-2-substituidos

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR258188A AR206812A1 (es) 1974-04-01 1975-01-01 Compuestos intermediarios de azaciclo(3,4-a)indoles 4- y 5-fenil substituidos desprovistos de actividad terapeutica

Country Status (15)

Country Link
JP (1) JPS587635B2 (es)
AR (2) AR206812A1 (es)
AU (1) AU7955975A (es)
DD (1) DD118879A5 (es)
DE (1) DE2514084A1 (es)
DK (2) DK130575A (es)
ES (3) ES436157A1 (es)
FI (1) FI750940A (es)
FR (1) FR2265368A1 (es)
IL (1) IL46925A0 (es)
LU (1) LU72182A1 (es)
NL (1) NL7503700A (es)
NO (1) NO751055L (es)
RO (1) RO72884A (es)
SE (2) SE423630B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4224329A (en) * 1979-01-23 1980-09-23 Pfizer Inc. 2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4451655A (en) * 1982-05-17 1984-05-29 Pfizer Inc. Process for preparing carboline derivatives and compounds used in their preparation
CZ294532B6 (cs) * 1998-12-21 2005-01-12 Janssen Pharmaceutica N. V. Benzisoxazoly a fenony jako alfa2-antagonisté, způsob jejich přípravy a použití a farmaceutický prostředek
RU2320662C1 (ru) * 2006-08-24 2008-03-27 Андрей Александрович Иващенко ЗАМЕЩЕННЫЕ ПИРРОЛО[4,3-b]ИНДОЛЫ, КОМБИНАТОРНАЯ И ФОКУСИРОВАННАЯ БИБЛИОТЕКИ, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
KR101868165B1 (ko) * 2010-04-22 2018-07-19 인트라-셀룰라 써래피스, 인코퍼레이티드. 유기 화합물

Also Published As

Publication number Publication date
AU7955975A (en) 1976-09-30
ES453788A1 (es) 1978-01-01
SE423630B (sv) 1982-05-17
DK130575A (es) 1975-10-02
FI750940A (es) 1975-10-02
NO751055L (es) 1975-10-02
JPS587635B2 (ja) 1983-02-10
DD118879A5 (es) 1976-03-20
SE8200047L (sv) 1982-01-07
RO72884B (ro) 1983-07-30
JPS50140494A (es) 1975-11-11
NL7503700A (nl) 1975-10-03
AR206812A1 (es) 1976-08-23
ES453787A1 (es) 1978-01-01
SE7502927L (es) 1975-10-02
FR2265368A1 (en) 1975-10-24
IL46925A0 (en) 1975-05-22
ES436157A1 (es) 1977-04-16
LU72182A1 (es) 1976-03-02
RO72884A (ro) 1983-08-03
FR2265368B1 (es) 1978-07-28
DE2514084A1 (de) 1975-11-20
DK187878A (da) 1978-05-01

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