AR206306A1 - PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION - Google Patents

PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION

Info

Publication number
AR206306A1
AR206306A1 AR251422A AR25142273A AR206306A1 AR 206306 A1 AR206306 A1 AR 206306A1 AR 251422 A AR251422 A AR 251422A AR 25142273 A AR25142273 A AR 25142273A AR 206306 A1 AR206306 A1 AR 206306A1
Authority
AR
Argentina
Prior art keywords
methylamines
meta
dioxane
procedure
preparation
Prior art date
Application number
AR251422A
Other languages
Spanish (es)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of AR206306A1 publication Critical patent/AR206306A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55Acids; Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/041,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/061,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AR251422A 1972-12-08 1973-01-01 PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION AR206306A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31322172A 1972-12-08 1972-12-08

Publications (1)

Publication Number Publication Date
AR206306A1 true AR206306A1 (en) 1976-07-15

Family

ID=23214841

Family Applications (3)

Application Number Title Priority Date Filing Date
AR251422A AR206306A1 (en) 1972-12-08 1973-01-01 PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION
AR251423A AR212416A1 (en) 1972-12-08 1973-12-07 PROCEDURE FOR THE PREPARATION OF N-METHYL ALPHA-PHENYL-O 3-PYRIDYL-5-M-DIOXANE-METHYLAMINE COMPOUNDS AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS
AR258799A AR212012A1 (en) 1972-12-08 1975-05-14 PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE

Family Applications After (2)

Application Number Title Priority Date Filing Date
AR251423A AR212416A1 (en) 1972-12-08 1973-12-07 PROCEDURE FOR THE PREPARATION OF N-METHYL ALPHA-PHENYL-O 3-PYRIDYL-5-M-DIOXANE-METHYLAMINE COMPOUNDS AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS
AR258799A AR212012A1 (en) 1972-12-08 1975-05-14 PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE

Country Status (27)

Country Link
JP (2) JPS5742633B2 (en)
AR (3) AR206306A1 (en)
AT (2) AT330773B (en)
BE (1) BE808340A (en)
BG (4) BG21409A3 (en)
CA (2) CA1014560A (en)
CH (4) CH605903A5 (en)
CS (3) CS193480B2 (en)
CY (1) CY1017A (en)
DD (3) DD110864A5 (en)
DE (1) DE2361340C2 (en)
DK (1) DK134717B (en)
ES (4) ES421290A1 (en)
FR (1) FR2209578B1 (en)
GB (2) GB1455997A (en)
HK (1) HK60479A (en)
HU (2) HU168763B (en)
IE (1) IE40226B1 (en)
IL (1) IL43773A (en)
KE (1) KE2976A (en)
MY (1) MY8000064A (en)
NL (1) NL7316839A (en)
PH (2) PH15197A (en)
SE (3) SE403377B (en)
SU (4) SU578001A3 (en)
YU (3) YU35447B (en)
ZA (1) ZA739207B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6030752B2 (en) * 2012-05-09 2016-11-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Method for producing oxetane-3-ylmethanamine
LV14983B (en) * 2013-10-15 2015-06-20 Olainfarm, A/S Method for producing intermediates of phenibut

Also Published As

Publication number Publication date
CS193480B2 (en) 1979-10-31
BG21223A3 (en) 1976-03-20
MY8000064A (en) 1980-12-31
SU578001A3 (en) 1977-10-25
CS222209B2 (en) 1983-05-27
BG22386A3 (en) 1977-02-20
AU6321773A (en) 1975-06-05
BG21409A3 (en) 1976-05-20
CH605903A5 (en) 1978-10-13
CH619219A5 (en) 1980-09-15
SE428378B (en) 1983-06-27
ES444716A1 (en) 1977-05-16
AR212416A1 (en) 1978-07-14
YU318473A (en) 1980-09-25
ATA1026073A (en) 1975-10-15
SE7701795L (en) 1977-02-17
SE417196B (en) 1981-03-02
IE40226B1 (en) 1979-04-11
ES444911A1 (en) 1977-09-01
SU587861A3 (en) 1978-01-05
DD115653A5 (en) 1975-10-12
CS222208B2 (en) 1983-05-27
HK60479A (en) 1979-08-31
CA1014560A (en) 1977-07-26
YU36020B (en) 1981-11-13
DE2361340C2 (en) 1983-11-24
JPS5734835B2 (en) 1982-07-26
BG26205A4 (en) 1979-02-15
ES421290A1 (en) 1976-07-01
FR2209578B1 (en) 1977-09-02
DK134717B (en) 1977-01-03
SU663305A3 (en) 1979-05-15
IL43773A0 (en) 1974-03-14
CY1017A (en) 1979-11-23
JPS5742633B2 (en) 1982-09-09
ES421291A1 (en) 1976-07-01
DD109625A5 (en) 1974-11-12
CH630914A5 (en) 1982-07-15
CH614439A5 (en) 1979-11-30
YU109380A (en) 1981-04-30
KE2976A (en) 1979-07-20
AT332396B (en) 1976-09-27
CA1024150A (en) 1978-01-10
BE808340A (en) 1974-06-07
YU35447B (en) 1981-02-28
PH15197A (en) 1982-09-17
SU648081A3 (en) 1979-02-15
HU168763B (en) 1976-07-28
NL7316839A (en) 1974-06-11
AR212012A1 (en) 1978-04-28
DD110864A5 (en) 1975-01-12
JPS4987681A (en) 1974-08-22
IE40226L (en) 1974-06-08
SE7701796L (en) 1977-02-17
SE403377B (en) 1978-08-14
DK134717C (en) 1977-05-31
HU168620B (en) 1976-06-28
DE2361340A1 (en) 1974-06-12
JPS4987680A (en) 1974-08-22
GB1455997A (en) 1976-11-17
PH14923A (en) 1982-01-29
AT330773B (en) 1976-07-26
ATA1026173A (en) 1976-01-15
ZA739207B (en) 1975-07-30
IL43773A (en) 1979-05-31
YU318573A (en) 1981-06-30
GB1455998A (en) 1976-11-17
YU36171B (en) 1982-02-25
FR2209578A1 (en) 1974-07-05

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