AR204660A1 - PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID - Google Patents

PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID

Info

Publication number
AR204660A1
AR204660A1 AR258571A AR25857175A AR204660A1 AR 204660 A1 AR204660 A1 AR 204660A1 AR 258571 A AR258571 A AR 258571A AR 25857175 A AR25857175 A AR 25857175A AR 204660 A1 AR204660 A1 AR 204660A1
Authority
AR
Argentina
Prior art keywords
oxopyride
piperazinil
pyrimidine
procedure
preparing compounds
Prior art date
Application number
AR258571A
Other languages
Spanish (es)
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Application granted granted Critical
Publication of AR204660A1 publication Critical patent/AR204660A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR258571A 1973-04-03 1975-01-01 PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AR204660A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (en) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (en) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (en) 1973-06-07 1973-06-07

Publications (1)

Publication Number Publication Date
AR204660A1 true AR204660A1 (en) 1976-02-20

Family

ID=27289838

Family Applications (2)

Application Number Title Priority Date Filing Date
AR253060A AR204003A1 (en) 1973-04-03 1974-01-01 PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS
AR258571A AR204660A1 (en) 1973-04-03 1975-01-01 PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR253060A AR204003A1 (en) 1973-04-03 1974-01-01 PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS

Country Status (11)

Country Link
AR (2) AR204003A1 (en)
AT (1) AT340931B (en)
CA (1) CA1066701A (en)
CH (1) CH593281A5 (en)
ES (1) ES424851A1 (en)
FI (1) FI56011C (en)
IE (1) IE39102B1 (en)
NL (1) NL186087C (en)
NO (1) NO142221C (en)
PH (2) PH10529A (en)
SE (1) SE416051B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (en) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS.
NZ597050A (en) 2009-06-29 2014-02-28 Incyte Corp Pyrimidinones as pi3k inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
US8680108B2 (en) 2009-12-18 2014-03-25 Incyte Corporation Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
AR084366A1 (en) 2010-12-20 2013-05-08 Incyte Corp N- (1- (REPLACED PHENYL) ETIL) -9H-PURIN-6-AMINAS AS PI3K INHIBITORS
BR122019020716B1 (en) 2011-09-02 2021-02-17 Incyte Holdings Corporation heterocyclylamines as pi3k inhibitors and pharmaceutical composition comprising them
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
MD3262046T2 (en) 2015-02-27 2021-03-31 Incyte Corp Salts of pi3k inhibitor and processes for their preparation
US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor

Also Published As

Publication number Publication date
NL7401509A (en) 1974-10-07
CH593281A5 (en) 1977-11-30
NO740349L (en) 1974-10-04
NO142221C (en) 1980-07-16
IE39102B1 (en) 1978-08-02
FI56011B (en) 1979-07-31
ATA277774A (en) 1977-05-15
IE39102L (en) 1974-10-03
AR204003A1 (en) 1975-11-12
PH10529A (en) 1977-05-30
NL186087C (en) 1990-09-17
NO142221B (en) 1980-04-08
SE416051B (en) 1980-11-24
FI56011C (en) 1979-11-12
CA1066701A (en) 1979-11-20
PH10984A (en) 1977-10-18
AT340931B (en) 1978-01-10
ES424851A1 (en) 1976-06-01
NL186087B (en) 1990-04-17

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