AR119009A1 - Derivados de alcoxipiridina y alcoxipirimidina microbicidas - Google Patents

Derivados de alcoxipiridina y alcoxipirimidina microbicidas

Info

Publication number
AR119009A1
AR119009A1 ARP200101481A ARP200101481A AR119009A1 AR 119009 A1 AR119009 A1 AR 119009A1 AR P200101481 A ARP200101481 A AR P200101481A AR P200101481 A ARP200101481 A AR P200101481A AR 119009 A1 AR119009 A1 AR 119009A1
Authority
AR
Argentina
Prior art keywords
alkoxy
alkyl
cycloalkyl
heterocyclyl
haloalkyl
Prior art date
Application number
ARP200101481A
Other languages
English (en)
Inventor
Stefano Rendine
Hamdan Farhan Bou
Andrew Edmunds
Mathias Blum
David Burns
Daniel Stierli
Mattia Riccardo Monaco
Original Assignee
Syngenta Crop Protection Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Crop Protection Ag filed Critical Syngenta Crop Protection Ag
Publication of AR119009A1 publication Critical patent/AR119009A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/501,3-Diazoles; Hydrogenated 1,3-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647Triazoles; Hydrogenated triazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/761,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00Fungicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Abstract

Compuestos de fórmula (1) en donde los sustituyentes son como se definen en la reivindicación 1, útiles como pesticidas y, en especial, fungicidas. Reivindicación 1: Compuesto de fórmula (1) en la que A es N o CH; R¹ es hidrógeno, ciano, formilo, alquilcarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, alcoxi C₁₋₆-alquilcarbonilo C₁₋₆, cicloalquilcarbonilo C₃₋₆, alcoxi C₁₋₆-alcoxicarbonilo C₁₋₃, alcoxioxalilo C₁₋₆, alcoxicarbonilo C₁₋₆-alquil-C₁₋₄-alcoxicarbonilo C₁₋₆, alqueniloxicarbonilo C₂₋₆, o alquiniloxicarbonilo C₂₋₆; R² es hidrógeno, alquilo C₁₋₆, haloalquilo C₁₋₆, halógeno, hidroxilo, alcoxilo C₁₋₆, haloalcoxilo C₁₋₆, cicloalquiloxilo C₃₋₆, halocicloalquiloxilo C₃₋₆, alqueniloxilo C₂₋₆, haloalqueniloxilo C₂₋₆, alquiniloxilo C₂₋₆, haloalquiniloxilo C₂₋₆, cianoalquiloxilo C₁₋₆, alcoxi C₁₋₆-alcoxilo C₁₋₃, alcoxi C₁₋₆-alquilo C₁₋₂, alquinilo C₂₋₆, haloalquinilo C₂₋₆, o cicloalquil C₃₋₆-alcoxilo C₁₋₂; R³ es hidrógeno, alquilo C₁₋₆, haloalquilo C₁₋₆, halógeno, hidroxilo, alcoxilo C₁₋₆, haloalcoxilo C₁₋₆, cicloalquiloxilo C₃₋₆, halocicloalquiloxilo C₃₋₆, alqueniloxilo C₂₋₆, haloalqueniloxilo C₂₋₆, alquiniloxilo C₂₋₆, haloalquiniloxilo C₂₋₆, cianoalquiloxilo C₁₋₆, alcoxi C₁₋₆-alcoxilo C₁₋₃, alcoxi C₁₋₆-alquilo C₁₋₂, alcoxi C₁₋₆-alquilcarboniloxilo C₁₋₂, alquinilo C₂₋₆, haloalquinilo C₂₋₆, o cicloalquil C₃₋₆-alcoxilo C₁₋₂; R⁴ es alquilo C₁₋₈, haloalquilo C₁₋₈, alcoxilo C₁₋₈, alquinilo C₃₋₈, cicloalquilo C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₂, fenilo, fenilalquilo C₁₋₃, fenoxialquilo C₁₋₃, heteroarilo, heteroarilalquilo C₁₋₂, heteroarilalcoxiimino C₁₋₂-alquilo C₁₋₂, donde el heteroarilo es un anillo monocíclico aromático de 5 ó 6 miembros que comprende 1, 2, 3 ó 4 heteroátomos seleccionados individualmente de N, O y S, heterociclilo, heterociclilalquilo C₁₋₂, donde el heterociclilo es un anillo monocíclico no aromático de 4, 5 ó 6 miembros que comprende 1, 2 ó 3 heteroátomos seleccionados individualmente de N, O, y S, y donde los restos cicloalquilo, fenilo, heteroarilo o heterociclilo están cada uno sustituido opcionalmente con de 1 a 3 grupos representados por R⁶ o 1 grupo representado por R⁷; y donde cuando R⁴ es un heterociclilo sustituido, estos ciclos pueden contener un grupo sulfonilo (S(O)₂); o R⁴ es un sistema de anillos anulados de 6 a 10 miembros que comprende opcionalmente 1, 2, ó 3 heteroátomos seleccionados individualmente de N, O y S, opcionalmente sustituidos con 1 ó 2 grupos representados por R⁶, y opcionalmente unidos al resto de la molécula a través de un ligador alquileno C₁₋₂; o R⁴ es un sistema de anillos carbobi- o carbotri-ciclilo espirocíclico no aromático de 5 a 10 miembros que comprende opcionalmente 1, 2, 3, 4 ó 5 heteroátomos seleccionados individualmente de N, O y S, opcionalmente sustituidos con de 1 a 3 grupos representados por R⁶, y opcionalmente unidos al resto de la molécula a través de un ligador alquileno C₁₋₂; R⁵ es alquilo C₁₋₈, hidroxialquilo C₁₋₈, cicloalquilo C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₂, fenilo, heteroarilo, donde el heteroarilo es un anillo monocíclico aromático de 5 ó 6 miembros que comprende 1, 2 ó 3 heteroátomos seleccionados individualmente de N, O y S, heterociclilo, donde el heterociclilo es un anillo monocíclico no aromático de 4, 5 ó 6 miembros o un anillo bicíclico no aromático de 9 a 10 miembros que comprende 1, 2 ó 3 heteroátomos seleccionados individualmente de N, O y S, y donde los restos cicloalquilo, fenilo, heteroarilo y heterociclilo están cada uno opcionalmente sustituido por 1, 2 ó 3 sustituyentes, que pueden ser los mismos o diferentes, seleccionados de R⁹; R⁶ es halógeno, alquilo C₁₋₄, alcoxilo C₁₋₄, haloalquilo C₁₋₄, ciano, o haloalcoxilo C₁₋₄; R⁷ es alquilsulfonilo C₁₋₄, cicloalquilo C₃₋₈, fenilo, bencilo, fenoxilo, o piridilo, donde cada cicloalquilo, el grupo fenilo o piridilo está opcionalmente sustituido por 1 grupo representado por R⁸; R⁸ es halógeno o haloalquilo C₁₋₄; R⁹ es halógeno, ciano, bencilo, alquilo C₁₋₄, alcoxilo C₁₋₄, o haloalquilo C₁₋₄; o una sal o un N-óxido del mismo.
ARP200101481A 2019-05-29 2020-05-26 Derivados de alcoxipiridina y alcoxipirimidina microbicidas AR119009A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP19177418 2019-05-29

Publications (1)

Publication Number Publication Date
AR119009A1 true AR119009A1 (es) 2021-11-17

Family

ID=66676455

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP200101481A AR119009A1 (es) 2019-05-29 2020-05-26 Derivados de alcoxipiridina y alcoxipirimidina microbicidas

Country Status (9)

Country Link
US (1) US20220272976A1 (es)
EP (1) EP3976586A1 (es)
JP (1) JP2022534272A (es)
CN (1) CN113874353A (es)
AR (1) AR119009A1 (es)
BR (1) BR112021023888A2 (es)
TW (1) TW202110802A (es)
UY (1) UY38719A (es)
WO (1) WO2020239856A1 (es)

Family Cites Families (61)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61107392A (ja) 1984-10-31 1986-05-26 株式会社東芝 画像処理システム
BR8600161A (pt) 1985-01-18 1986-09-23 Plant Genetic Systems Nv Gene quimerico,vetores de plasmidio hibrido,intermediario,processo para controlar insetos em agricultura ou horticultura,composicao inseticida,processo para transformar celulas de plantas para expressar uma toxina de polipeptideo produzida por bacillus thuringiensis,planta,semente de planta,cultura de celulas e plasmidio
AU613521B2 (en) 1988-09-02 1991-08-01 Sankyo Company Limited 13-substituted milbemycin derivatives, their preparation and use
US5169629A (en) 1988-11-01 1992-12-08 Mycogen Corporation Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg
NZ231804A (en) 1988-12-19 1993-03-26 Ciba Geigy Ag Insecticidal toxin from leiurus quinquestriatus hebraeus
US5015630A (en) 1989-01-19 1991-05-14 Merck & Co., Inc. 5-oxime avermectin derivatives
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
GB8910624D0 (en) 1989-05-09 1989-06-21 Ici Plc Bacterial strains
CA2015951A1 (en) 1989-05-18 1990-11-18 Mycogen Corporation Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins
DE69018772T2 (de) 1989-11-07 1996-03-14 Pioneer Hi Bred Int Larven abtötende Lektine und darauf beruhende Pflanzenresistenz gegen Insekten.
JPH085894B2 (ja) 1990-03-01 1996-01-24 三共株式会社 ミルベマイシンエーテル誘導体
JPH0570366A (ja) 1991-03-08 1993-03-23 Meiji Seika Kaisha Ltd 薬用組成物
UA48104C2 (uk) 1991-10-04 2002-08-15 Новартіс Аг Фрагмент днк, який містить послідовність,що кодує інсектицидний протеїн, оптимізовану для кукурудзи,фрагмент днк, який забезпечує направлену бажану для серцевини стебла експресію зв'язаного з нею структурного гена в рослині, фрагмент днк, який забезпечує специфічну для пилку експресію зв`язаного з нею структурного гена в рослині, рекомбінантна молекула днк, спосіб одержання оптимізованої для кукурудзи кодуючої послідовності інсектицидного протеїну, спосіб захисту рослин кукурудзи щонайменше від однієї комахи-шкідника
EP0634408B1 (en) 1992-03-17 2002-01-02 Fujisawa Pharmaceutical Co., Ltd. Depsipeptide derivative, production thereof and use thereof
ES2118816T3 (es) 1992-04-28 1998-10-01 Yashima Kagaku Kogyo Kk 2-(2,6-difluorofenil)-4-(2-etoxi-4-terc-butilfenil)-2-oxazolina.
DE4317458A1 (de) 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
CA2105251C (en) 1992-09-01 2004-12-07 Mitsugi Shibano Novel processes for the production of 13-ether derivatives of milbemycins, and novel intermediates therefor
GB9300883D0 (en) 1993-01-18 1993-03-10 Pfizer Ltd Antiparasitic agents
CN1073560C (zh) 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
EP0739344B1 (en) 1994-01-14 1998-11-11 Pfizer Inc. Antiparasitic pyrrolobenzoxazine compounds
GB9402916D0 (en) 1994-02-16 1994-04-06 Pfizer Ltd Antiparasitic agents
US5530195A (en) 1994-06-10 1996-06-25 Ciba-Geigy Corporation Bacillus thuringiensis gene encoding a toxin active against insects
DE4437198A1 (de) 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
DE4440193A1 (de) 1994-11-10 1996-05-15 Bayer Ag Verwendung von Dioxomorpholinen zur Bekämpfung von Endoparasiten, neue Dioxomorpholine und Verfahren zur ihrer Herstellung
DE19520936A1 (de) 1995-06-08 1996-12-12 Bayer Ag Ektoparasitizide Mittel
GB9523675D0 (en) * 1995-11-20 1996-01-24 Celltech Therapeutics Ltd Chemical compounds
KR100482919B1 (ko) 1996-03-11 2005-10-12 신젠타 파티서페이션즈 아게 살충제로서의피리미딘-4-온유도체
WO2002015701A2 (en) 2000-08-25 2002-02-28 Syngenta Participations Ag Bacillus thuringiensis crystal protein hybrids
US7230167B2 (en) 2001-08-31 2007-06-12 Syngenta Participations Ag Modified Cry3A toxins and nucleic acid sequences coding therefor
WO2003052073A2 (en) 2001-12-17 2003-06-26 Syngenta Participations Ag Novel corn event
GB0303439D0 (en) 2003-02-14 2003-03-19 Pfizer Ltd Antiparasitic terpene alkaloids
US20090227612A1 (en) * 2005-12-22 2009-09-10 Boonsaeng Park Aminopyrimidine Derivatives Inhibiting Protein Kinase Activity, Method For The Preparation Thereof And Pharmaceutical Composition Containing Same
WO2010012793A1 (en) 2008-08-01 2010-02-04 Bayer Cropscience Sa Fungicide aminothiazole derivatives
CN103270041A (zh) 2010-05-06 2013-08-28 拜尔农作物科学股份公司 二噻英-四羧基-二酰亚胺的制备方法
GB201017345D0 (en) * 2010-10-14 2010-11-24 Proximagen Ltd Receptor antagonists
CN106478497B (zh) * 2010-10-18 2020-05-08 拉夸里亚创药株式会社 作为ttx-s阻滞剂的芳胺衍生物
MA37825B1 (fr) 2012-07-04 2016-06-30 Agro Kanesho Co Ltd Dérivé d'ester d'acide 2-aminonicotinique et bactéricide le contenant comme principe actif
EA027009B1 (ru) 2012-12-19 2017-06-30 Байер Кропсайенс Акциенгезельшафт Дифторметилникотиновые инданилкарбоксамиды
GB201316600D0 (en) * 2013-09-18 2013-10-30 Redx Pharma Ltd Agricultural chemicals
US10173983B2 (en) 2014-04-11 2019-01-08 Syngenta Participations Ag Fungicidal pyridylamidines
CN111892576A (zh) 2015-03-27 2020-11-06 先正达参股股份有限公司 杀微生物的杂二环衍生物
WO2016156290A1 (en) 2015-04-02 2016-10-06 Bayer Cropscience Aktiengesellschaft Novel 5-substituted imidazole derivatives
WO2016183741A1 (en) * 2015-05-15 2016-11-24 Merck Sharp & Dohme Corp. Pyrimidinone amide compounds as pde2 inhibitors
US10758522B2 (en) * 2015-06-01 2020-09-01 The Scripps Research Institute Small molecule analogs of the nemo binding peptide
JP2018522846A (ja) 2015-06-15 2018-08-16 バイエル・クロップサイエンス・アクチェンゲゼルシャフト ハロゲン置換フェノキシフェニルアミジン類及び殺菌剤としてのそれらの使用
AU2016305250B2 (en) 2015-08-12 2020-10-22 Syngenta Participations Ag Microbiocidal heterobicyclic derivatives
KR20180037267A (ko) 2015-08-14 2018-04-11 바이엘 크롭사이언스 악티엔게젤샤프트 트리아졸 유도체, 그의 중간체 및 살진균제로서의 그의 용도
WO2017055473A1 (en) 2015-10-02 2017-04-06 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
JP6864673B2 (ja) 2015-10-02 2021-04-28 シンジェンタ パーティシペーションズ アーゲー 殺微生物オキサジアゾール誘導体
US10640497B2 (en) 2015-12-02 2020-05-05 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
UY37062A (es) 2016-01-08 2017-08-31 Syngenta Participations Ag Derivados de aryl oxadiazol fungicidas
CR20180434A (es) 2016-03-10 2018-11-21 Syngenta Participations Ag Derivados microbiocidas de tipo (tio) carboxamida de la quinolina
CA3024528A1 (en) 2016-05-30 2017-12-07 Syngenta Participations Ag Microbiocidal thiazole derivatives
AR108745A1 (es) 2016-06-21 2018-09-19 Syngenta Participations Ag Derivados de oxadiazol microbiocidas
US10653146B2 (en) 2016-10-06 2020-05-19 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
WO2018153707A1 (en) 2017-02-22 2018-08-30 Basf Se Crystalline forms of a strobilurin type compound for combating phytopathogenic fungi
UY37623A (es) 2017-03-03 2018-09-28 Syngenta Participations Ag Derivados de oxadiazol tiofeno fungicidas
US20210084902A1 (en) 2017-05-02 2021-03-25 Basf Se Fungicidal mixture comprising substituted 3-phenyl-5-(trifluoromethyl)-1,2,4-oxadiazoles
US11154058B2 (en) 2017-06-14 2021-10-26 Syngenta Participations Ag Fungicidal compositions
EP3720846A1 (en) 2017-12-04 2020-10-14 Syngenta Participations AG Microbiocidal phenylamidine derivatives

Also Published As

Publication number Publication date
CN113874353A (zh) 2021-12-31
US20220272976A1 (en) 2022-09-01
JP2022534272A (ja) 2022-07-28
TW202110802A (zh) 2021-03-16
EP3976586A1 (en) 2022-04-06
UY38719A (es) 2020-12-31
WO2020239856A1 (en) 2020-12-03
BR112021023888A2 (pt) 2022-05-10

Similar Documents

Publication Publication Date Title
AR114254A1 (es) Moduladores del regulador de conductancia transmembrana de fibrosis quística, composiciones farmacéuticas, métodos de tratamiento y proceso de preparación de los moduladores
AR110922A1 (es) Compuestos inhibidores del vih
AR123926A2 (es) 4-amino-6-(heterocíclico)picolinatos y 6-amino-2-(heterocíclico)pirimidina-4-carboxilatos y su uso como herbicidas
AR111686A1 (es) 4-amino-6-(heterocíclico)picolinatos y 6-amino-2-(heterocíclico)pirimidina-4-carboxilatos y sus usos como herbicidas
AR110405A1 (es) Compuestos
AR100645A1 (es) Derivados de pirazolo-pirimidina
AR113929A1 (es) Compuestos heterocíclicos
AR100315A1 (es) Compuestos de piridina sustituida que tienen acción herbicida
AR117200A1 (es) Derivados de tiazol microbiocidas
AR117183A1 (es) Derivados de tiazol microbiocidas
AR113842A1 (es) Derivados de tiazol microbiocidas
AR108629A1 (es) Derivados de tiazol microbiocidas
AR107955A1 (es) Derivados de piridino- / pirimidino-piridina, con actividad herbicida
AR111808A1 (es) Derivados de pirimidina como moduladores del receptor de pge2
AR111941A1 (es) Derivados de pirimidina como moduladores del receptor de pge2
AR111807A1 (es) Derivados de benzofurano y benzotiofeno como moduladores del receptor pge2
AR111874A1 (es) Derivados de pirimidina
AR109964A1 (es) Derivados de aril-sulfonamidas como bloqueadores del canal de sodio
AR099789A1 (es) Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
AR111248A1 (es) Derivados de ciclopropilmetilamida activos como pesticida
AR109296A1 (es) Derivados de oxadiazolopiridina para el uso como inhibidores de ghrelin o-aciltransferasa (goat)
AR118015A1 (es) Compuestos herbicidas
AR114564A1 (es) DERIVADOS DE 2,4,6,7-TETRAHIDRO-PIRAZOLO[3,4-D]PIRIMIDIN-ONA COMO MODULADORES DEL RECEPTOR C5a Y COMPOSICIÓN FARMACÉUTICA QUE LOS COMPRENDE
AR120377A1 (es) Derivados heteroaromáticos de sulfiliminas o sulfoximinas con actividad fungicida
AR118154A1 (es) Compuestos herbicidas