AR103708A1 - BENZOXABOROL COMPOUNDS AND USES OF THE SAME - Google Patents

BENZOXABOROL COMPOUNDS AND USES OF THE SAME

Info

Publication number
AR103708A1
AR103708A1 ARP160100406A ARP160100406A AR103708A1 AR 103708 A1 AR103708 A1 AR 103708A1 AR P160100406 A ARP160100406 A AR P160100406A AR P160100406 A ARP160100406 A AR P160100406A AR 103708 A1 AR103708 A1 AR 103708A1
Authority
AR
Argentina
Prior art keywords
same
compounds
microbacterial
benzoxaborol compounds
benzoxaborol
Prior art date
Application number
ARP160100406A
Other languages
Spanish (es)
Original Assignee
Anacor Pharmaceuticals Inc
GLAXOSMITHKLINE INTELLECTUAL PROPERTY (Nº 2) LTD
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc, GLAXOSMITHKLINE INTELLECTUAL PROPERTY (Nº 2) LTD filed Critical Anacor Pharmaceuticals Inc
Publication of AR103708A1 publication Critical patent/AR103708A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composiciones que los contienen, su uso en terapia, incluyendo su uso como agentes anti-microbacterianos, por ejemplo, en el tratamiento de una infección microbacteriana en un mamífero, y los métodos para la preparación de estos compuestos. Reivindicación 1: Un compuesto que comprende la estructura de la fórmula (1), en donde X se selecciona a partir de flúor, cloro, bromo o yodo, y R¹ y R² se seleccionan cada uno independientemente a partir de H, -CH₃, -CH₂CH₃, -CH₂CH₂CH₃ y -CH(CH₃)₂; o una sal o hidrato del mismo.Compositions containing them, their use in therapy, including their use as anti-microbacterial agents, for example, in the treatment of a microbacterial infection in a mammal, and the methods for the preparation of these compounds. Claim 1: A compound comprising the structure of the formula (1), wherein X is selected from fluorine, chlorine, bromine or iodine, and R¹ and R² are each independently selected from H, -CH₃, - CH₂CH₃, -CH₂CH₂CH₃ and -CH (CH₃) ₂; or a salt or hydrate thereof.

ARP160100406A 2015-02-12 2016-02-15 BENZOXABOROL COMPOUNDS AND USES OF THE SAME AR103708A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP15382054 2015-02-12

Publications (1)

Publication Number Publication Date
AR103708A1 true AR103708A1 (en) 2017-05-31

Family

ID=52477755

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP160100406A AR103708A1 (en) 2015-02-12 2016-02-15 BENZOXABOROL COMPOUNDS AND USES OF THE SAME
ARP160100405A AR103707A1 (en) 2015-02-12 2016-02-15 BENZOXABOROL COMPOUNDS

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP160100405A AR103707A1 (en) 2015-02-12 2016-02-15 BENZOXABOROL COMPOUNDS

Country Status (1)

Country Link
AR (2) AR103708A1 (en)

Also Published As

Publication number Publication date
AR103707A1 (en) 2017-05-31

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