AR096626A1 - ANTIBODY-DRUG CONJUGATE COMPOUNDS 1- (CHLOROME) -2,3-DIHIDRO-1H-BENZO [E] INDOL, AND METHODS OF USE AND TREATMENT - Google Patents

ANTIBODY-DRUG CONJUGATE COMPOUNDS 1- (CHLOROME) -2,3-DIHIDRO-1H-BENZO [E] INDOL, AND METHODS OF USE AND TREATMENT

Info

Publication number
AR096626A1
AR096626A1 ARP140102283A ARP140102283A AR096626A1 AR 096626 A1 AR096626 A1 AR 096626A1 AR P140102283 A ARP140102283 A AR P140102283A AR P140102283 A ARP140102283 A AR P140102283A AR 096626 A1 AR096626 A1 AR 096626A1
Authority
AR
Argentina
Prior art keywords
antibody
benzo
chlorome
dihidro
indol
Prior art date
Application number
ARP140102283A
Other languages
Spanish (es)
Original Assignee
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of AR096626A1 publication Critical patent/AR096626A1/en

Links

Landscapes

  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)

Abstract

La solicitud proporciona conjugados anticuerpo-fármaco que comprenden un anticuerpo conjugado a un resto de fármaco dimérico de 1-(clorometil)-2,3-dihidro-1H-benzo[e]indol (CBI) mediante un ligante, y método para utilizar los conjugados anticuerpo-fármaco.The application provides antibody-drug conjugates comprising an antibody conjugated to a dimeric drug moiety of 1- (chloromethyl) -2,3-dihydro-1H-benzo [e] indole (CBI) by a binder, and method of using the antibody-drug conjugates.

ARP140102283A 2013-08-12 2014-06-16 ANTIBODY-DRUG CONJUGATE COMPOUNDS 1- (CHLOROME) -2,3-DIHIDRO-1H-BENZO [E] INDOL, AND METHODS OF USE AND TREATMENT AR096626A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361864889P 2013-08-12 2013-08-12

Publications (1)

Publication Number Publication Date
AR096626A1 true AR096626A1 (en) 2016-01-20

Family

ID=56125278

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140102283A AR096626A1 (en) 2013-08-12 2014-06-16 ANTIBODY-DRUG CONJUGATE COMPOUNDS 1- (CHLOROME) -2,3-DIHIDRO-1H-BENZO [E] INDOL, AND METHODS OF USE AND TREATMENT

Country Status (2)

Country Link
AR (1) AR096626A1 (en)
MA (1) MA38812B1 (en)

Also Published As

Publication number Publication date
MA38812B1 (en) 2018-11-30
MA38812A1 (en) 2018-05-31

Similar Documents

Publication Publication Date Title
CR20160125A (en) ANTIBODY-DRUG CONJUGATE COMPOUNDS 1- (CHLOROME) -2,3-DIHIDRO-1H-BENZO [E] INDOL, AND METHODS OF USE AND TREATMENT
BR112016013258A2 (en) antibody-drug conjugate, pharmaceutical composition, method for treating cancer and kit
CR20180243A (en) PIRROLOBENZODIAZEPIN ANTIBODY-DRUG CONJUGATES AND METHODS OF USE
CL2019000334A1 (en) New antibody conjugates and uses thereof (divisional application 201502357)
CO6771458A2 (en) Antibody-drug conjugates
PA8718601A1 (en) ANTI-5T4 ANTIBODIES AND THEIR USES
CL2015003280A1 (en) Benzimidazole derivatives as bromodomain inhibitors
CL2018003758A1 (en) Anti-dll3-antibody antibody conjugates and methods of use. (divisional application 201800458)
EA201791461A1 (en) BENZODIAZEPIN DYMERAS WITH BRIDGES HETEROARILENE, THEIR CONJUGATES, METHODS OF OBTAINING AND APPLICATION
BR112016010169A2 (en) anticlaudin antibodies and methods of use
PE20150891A1 (en) IL-13 ALPHA 2 ANTI-RECEPTOR ANTIBODIES AND DRUG ANTIBODY CONJUGATES
PE20150646A1 (en) METHODS OF TREATING A TAUOPATHY
CL2016002667A1 (en) Novel anti-rnf43 antibodies and methods for use
BR112013023015A2 (en) amatoxine conjugate and its use, pharmaceutical composition and its use, amatoxine conjugation molecule, method for the synthesis of an amatoxine conjugate.
EA201590171A1 (en) IMMUNOCONGATES CONTAINING ANTIBODIES TO CD79b
ECSP18049762A (en) NEW ANTI-CLAUDIN ANTIBODIES AND THEIR METHODS OF USE
UY35434A (en) ? 4-AMINO-6- (HETEROCYCLIC) PICOLINATES AND 6-AMINO-2- (HETEROCYCLIC) PYRIMIDIN-4-CARBOXYLATES AND ITS USE AS HERBICIDES ?.
CR20120522A (en) PIRROLOBENZODIACEPINAS AND CONJUGATES OF THE SAME
PE20170254A1 (en) ANTIBODIES AND ANTI-VISION FRAGMENTS
CU20190061A7 (en) ANTIBODY-DRUG CONJUGATES FOR ABLATION OF HEMATOPOIETIC STEM CELLS
CO2018005433A2 (en) Site-specific her2 antibody drug conjugates
CR20120221A (en) COMPOUNDS AND METHODS FOR THE MODULATION OF KINASES, AND INDICATIONS FOR IT
CL2012003584A1 (en) Pharmaceutical dosage form comprising 6-fluoro - (n-methyl-or n, n-dimethyl) -4-phenyl -4,9-dihydro-3h-spiro - (cyclohexan-1,1-pyran (3,4, b) indole) -4-amine, useful as an analgesic
GT201200321A (en) DERIVATIVES OF HETEROARIL IMIDAZOLONA AS JAK INHIBITORS
GT200500385A (en) TRICYCLE AMINOALCOHOLES, PROCEDURES FOR PREPARATION AND USE AS INFLAMMATION INHIBITORS

Legal Events

Date Code Title Description
FB Suspension of granting procedure